Seznam vědeckých a publikačních aktivit, vyžádaných přednášek a grantů a další aktivity dokládající osobnost uchazeče ABA Studie charakteru vědecké monografie v časopisech a sbornících vydané v zahraničních vydavatelstvích ABA01 Jampílek, Josef [UKOEXAF] (50% [2,18 AH]) - Kráľová, Katarína [UKOPRCUS] (50% [2,18 AH]): Application of Nanotechnology in Agriculture and Food Industry, Its Prospects and Risks Lit.: 432 zázn. In: Ecological Chemistry and Engineering S. - Vol. 22, No. 3 (2015), s. 321-361 [4,36 AH] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2015= [2014-0,553] ABA02 Kráľová, Katarína [UKOPRCUS] (70% [2,67 AH]) - Jampílek, Josef [UKOEXAF] (30% [1,14 AH]): Impact of environmental contaminants on breast cancer Lit.: 304 zázn. In: Ecological Chemistry and Engineering S. - Vol. 22, No. 1 (2015), s. 9-44 [3,81 AH] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2015= [2014-0,553] ABC Kapitoly ve vědeckých monografiích vydané v zahraničních vydavatelstvích ABC01 Doležal, Martin (40%) - Zitko, Jan (25%) - Jampílek, Josef [UKOEXAF] (35%): Pyrazinecarboxylic acid derivatives with antimycobacterial activity Lit. 108 zázn. In: Ed.: Cardona, P.J. : Understanding Tuberculosis : New approaches to fighting against drug resistance. Rijeka : InTech, 2012. - S. 233-262 [2,35 AH]. - ISBN 978-953-307-948-6 ABC02 Jampílek, Josef [UKOEXAF] (80%) - Dohnal, Jiří (20%): Investigation of carbohydrates and their derivatives as crystallization modifiers Lit. 126 zázn. In: Ed.: Chang, Ch.F. : Carbohydrates : Comprehensive studies on glycobiology and glycotechnology. Rijeka : InTech, 2012. - S. 81-116 [2,74 AH]. - ISBN 978-953-51-0864-1 ABC03 Jampílek, Josef [UKOEXAF] (80%) - Dohnal, Jiří (20%): Alaptide as transdermal permeation modifier Lit. 69 zázn. In: Eds.: Nina Dragicevic, Howard I. Maibach : Percutaneous Penetration Enhancers Chemical Methods in Penetration Enhancement : Modification of the Stratum Corneum. - Berlin : Springer, 2015. - S. 115-132 [1,38 AH]. - ISBN 978-3-662-47038-1 ABC04 Jampílek, Josef [UKOEXAF] (100%) : Azone(R) and its analogues as penetration enhancers Lit. 114 zázn. In: Eds.: Nina Dragicevic, Howard I. Maibach : Percutaneous Penetration Enhancers Chemical Methods in Penetration Enhancement : Modification of the Stratum Corneum. - Berlin : Springer, 2015. - S. 69-105 [3,21 AH]. - ISBN 978-3-662-47038-1 ACB Vysokoškolské učebnice vydané v domácích vydavatelstvích ACB01 Brusová, Hana (8%) - Dohnal, Jiří (8%) - Grafnetterová, Taťjana (4%) - Grünwaldová, Veronika (12%) - Havlíček, Jaroslav (7%) - Jampílek, Josef [UKOEXAF] (20%) - Král, Vladimír (1%) - Opatřilová, Radka (2%) - Pekárek, Tomáš (4%) - Plaček, Lukáš (7%)- Krumbholcová, Lucie (3%) - Řezáčová, Anna (6%) Setnička, Vladimír (9%) - Urbanová, Marie (9%): Moderní přístupy k farmaceutické analýze. - 1. vyd. Praha : Veterinární a farmaceutická univerzita Brno, 2010. - 500 s. [17,45 AH] Jampílek, J.: 3,48 AH Lit. 36 zázn. ISBN 978-80-7305-085-6
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ADC Vědecké práce v zahraničních karentovaných časopisech ADC01 Jampílek, Josef [UKOEXAF] (80%) - Doležal, Martin (10%) - Dvořák, Bohumír (10%): Bis(4methoxyphenyl)disulfide formation through copper catalysts Lit. 17 zázn. In: Chemical papers. - Vol. 56, No. 3 (2002), s. 147-149 Registrované v: wos Indikátor časopisu: IF (JCR) 2002=0,336 ADC02 Jampílek, Josef [UKOEXAF] (45%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Víchová, Petra (10%) - Jun, Daniel (10%) - Hanika, Jiří (5%) - O'Connor, Robert (5%) - Clynes, Martin (5%): Synthesis of(2E)2-methyl-3-(4-[4-(quinolin-2-ylmethoxy)phenyl]sulfanylphenyl)prop-2-enoic acid (VUFB 20609) and 2methyl-3-(4-[4-(quinolin-2-ylmethoxy)phenyl]sulfanylphenyl)propanoic acid (VUFB 20584) as potential antileukotrienic agents Lit. 30 zázn. In: Journal of Pharmacy and Pharmacology. - Vol. 56, No. 6 (2004), s. 783-794 Registrované v: wos Indikátor časopisu: IF (JCR) 2004=1,348 Ohlasy (3): [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5130 - SCI [o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol. 19, No. 2, 2008, s. 263 - SCI [o1] 2009 Brychtova, K. - Farsa, O. - Csollei, J.: Letters in Organic Chemistry, Vol. 6, No. 1, 2009, s. 28 SCI ADC03 Jampílek, Josef [UKOEXAF] (45%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Víchová, Petra (10%) - Raich, Ivan (5%) - Jun, Daniel (10%) - O'Connor, Robert (5%) - Clynes, Martin (5%): Preparation of2(4-[4-(Quinolin-2-ylmethoxy)phenyl]sulfanylphenyl) propionic acid (VUFB 20615) and 2-methyl-2-(4-[4(quinolin-2- ylmethoxy)phenyl]sulfanylphenyl)propionic acid (VUFB 20623) as potential antileukotrienic agents Lit. 27 zázn. In: Current Organic Chemistry. - Vol. 8, No. 13 (2004), s. 1235-1243 Registrované v: wos Indikátor časopisu: IF (JCR) 2004=2,775 Ohlasy (3): [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5130 - SCI [o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol. 19, No. 2, 2008, s. 263 - SCI [o1] 2009 Brychtova, K. - Farsa, O. - Csollei, J.: Letters in Organic Chemistry, Vol. 6, No. 1, 2009, s. 28 SCI ADC04 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Raich, Ivan (10%) Liška, František (10%): 4-substituted aryl bromides coupling with 4-methoxybenzene-1-thiol by means of copper catalysts Lit. 38 zázn. In: Chemical papers. - Vol. 59, No. 3 (2005), s. 182-186 Registrované v: wos Indikátor časopisu: IF (JCR) 2005=0,409 Ohlasy (3): [o1] 2009 Brychtova, K. - Farsa, O. - Csollei, J.: Letters in Organic Chemistry, Vol. 6, No. 1, 2009, s. 28 SCI [o1] 2010 Del Rosso, P.G. - Almassio, M.F. - Bruno, M. - Garay, R.O.: Tetrahedron Letters, Vol. 51, No. 51, 2010, s. 6733 - SCI [o1] 2012 Moosun, S. - Joule, J.A. - Bhowon, M.G. - Jhaumeer-Laulloo, S.: Phosphorus Sulfur and Silicon and the Related Elements, Vol. 187, No. 11, 2012, s. 1400 - SCI
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ADC05 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Šatínsky, Dalibor (10%) - Raich, Ivan (10%): Novel regioselective preparation of 5-chloropyrazine-2-carbonitrile from pyrazine-2-carboxamide and coupling study of substituted phenylsulfanylpyrazine- 2-carboxylic acid derivatives Lit. 41 zázn. In: Current Organic Chemistry. - Vol. 9, No. 1 (2005), s. 49-60 Registrované v: wos Indikátor časopisu: IF (JCR) 2005=3,102 Ohlasy (2): [o1] 2009 Brychtova, K. - Farsa, O. - Csollei, J.: Letters in Organic Chemistry, Vol. 6, No. 1, 2009, s. 28 SCI [o1] 2009 Hu, L.X. - Arafa, R.K. - Ismail, M.A. - Patel, A. - Munde, M. - Wilson, W.D. - Wenzler, T. Brun, R. - Boykin, D.W.: Bioorganic & Medicinal Chemistry, Vol. 17, No. 18, 2009, s. 6658 - SCI ADC06 Doležal, Martin (20%) - Pálek, Lukáš (15%) - Vinšová, Jarmila (5%) - Buchta, Vladimír (20%) Jampílek, Josef [UKOEXAF] (20%) - Kráľová, Katarína [UKOPRCUS] (20%): Substituted Pyrazinecarboxamides: Synthesis and Biological Evaluation Lit.: 27 zázn. In: Molecules. - Vol. 11, No. 4 (2006), s. 242-256 Registrované v: wos Indikátor časopisu: IF (JCR) 2006=0,841 Ohlasy (20): [o3] 2008 Martin, S. - Revathi, C. - Dayalan, A. - Mathivanan, N. - Shanmugaiya, V.: Rasayan Journal of Chemistry, Vol. 1, No. 2, 2008, s. 378-389 [o1] 2009 Ukrainets, L.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Khimiya Geterotsiklicheskikh Soedinenii, No. 9, 2009, s. 1324-1337 - SCOPUS [o1] 2009 Ukrainets, L.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Chemistry of Heterocyclic Compouds, Vol. 45, No. 9, 2009, s. 1058-1068 - SCI [o1] 2010 Lee, J.H. - Myung, P.K. - Kim, S.J. - Sung, N.D.: Journal of Applied Biological Chemistry, Vol. 53, No. 4, 2010, s. 440-445 - SCOPUS [o3] 2010 Meenakshi, S. – Malhotra, R.: Agricultural and Biological Research, Vol. 26, No. 2, 2010, s. 123-135 [o3] 2010 Tewatia, N. - Namdeo, K.P. - Jain, S.K. - Prajapati, S.K. - Singh, O. - Jain, V. - Kumar, P.: Journal of the Institution of Chemists (India), Vol. 82, No. 5, 2010, s. 148-153 [o3] 2011 Lima, C.H.S. - Bispo, M.L.F. - de Souza, M.V.N.: Pirazinamida: Um Fármaco Essencial no Tratamento da Tuberculose. In: Revista Virtual de Química, Vol. 3, No. 3, 2011, s. 159-180 [o3] 2011 Prasad, R. - Sharma, R.: 2D QSAR Analysis of pyrazinecarboxamides derivatives as an herbicidal agent. In: Journal of Computational Methods in Molecular Design, Vol. 1, No. 1, 2011, s. 7-13 [o1] 2012 Patel, N. B. - Patel, H. R.: Arabian Journal of Chemistry, Vol. 5, Iss. 1, 2012, s. 81-91 - SCI ; SCOPUS [o3] 2011 Khalil, A. - Mohamed, S. I. - Eyada, H. A. - abdel Alaziz, T. A. - Ali, G. A. M. - Mohamed ElHag: Journal of Materials Science and Engineering A, Vol. 1, Iss. 2, 2011, s. 228-235 [o1] 2012 Lo Monte, F. - Kramer, T. - Gu, J. - Anumala, U.R. - Marinelli, L. - La Pietra, V. - Novellino, E. - Franco, B. - Demedts, D. - Van Leuven, F. - Fuertes, A. - Dominguez, J.M. - Plotkin, B. - EldarFinkelman, H. - Schmidt, B.: Journalof Medicinal Chemistry, Vol. 55, No. 9, 2012, s. 4407-4424 - SCI ; SCOPUS [o1] 2012 Tewatia, N. - Abidab, Namdeo, K.P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 3, 2012, s. 1794-1798 - SCOPUS [o3] 2012 Vikramjeet J. - Balasubramanian N. - Munish A.: A Review of Biological potential of Pyrazinamide derivatives. In: Hygeia. Journal for drugs and medicines, Vol. 4, No. 1, 2012, s. 6 [o3] 2011 Sato, N.: Pyrazines. In: Science of Synthesis, Knowledge Updates, No. 4, 2011, s. 235-343 [o1] 2013 Zhang, R.Z. - Zhang, X.Z.: Indian Journal of Pure and Applied Physics, Vol. 51, No. 3, 2013, s. 164-173 - SCI ; SCOPUS [o1] 2013 Helal, M.H. - Abbas, S.Y. - Salem, M.A. - Farag, A.A. - Ammar, Y.A.: Medicinal Chemistry Research, Vol. 22, No. 11, 2013, s. 5598-5609 - SCOPUS ; SCI [o3] 2014 Parimala Vaijayanthi, S. - Mathiyalagan, N.: Antibacterial, antifungal, anti-oxidant, antiinflammatory and anti-hypertensive activities of N-chloropyrazinamide. In: International Letters of Chemistry, Physics and Astronomy, Vol. 7, 2014, s. 1-8
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[o1] 2014 Nayak, P.S. - Narayana, B. - Anthal, S. - Gupta, V.K. - Kant, R.: Molecular Crystals and Liquid Crystals, Vol. 592, No. 1, 2014, s. 199-208 - SCI ; SCOPUS [o1] 2015 Verbitskiy, E.V. - Slepukhin, P.A. - Kravchenko, M.A. - Skornyakov, S.N. - Evstigneeva, N.P. Kungurov, N.V. - Zil'Berberg, N.V. - Rusinov, G.L. - Chupakhin, O.N. - Charushin, V.N.: Bioorganic and Medicinal Chemistry Letters, Vol. 25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS [o1] 2016 Chylewska, A. - Sikorski, A. - Ogryzek, M. - Makowski, M.: Journal of Molecular Structure, Vol. 1105, 2016, s. 104 - SCI; SCOPUS ADC07 Jampílek, Josef [UKOEXAF] (75%) - Doležal, Martin (10%) - Opletalová, Veronika (10%) - Hart, Jiří (5%): 5-lipoxygenase, leukotrienes biosynthesis and potential antileukotrienic agents Lit. 102 zázn. In: Current Medicinal Chemistry. - Vol. 13, No.2 (2006), s. 117-129 Registrované v: wos Indikátor časopisu: IF (JCR) 2006=5,207 Ohlasy (18): [o1] 2006 Ward, W.O. - Delker, D.A. - Hester, S.D. - Thai, S.F. - Wolf, D.C. - Allen, J.W. - Nesnow, S.: Toxicologic Pathology, Vol. 34, No. 7, 2006, s. 878 - SCI [o1] 2006 Chen, X.X. - Sood, S. - Yang, C.S. - Li, N. - Sun, Z.: Current Cancer Drug Targets, Vol. 6, No. 7, 2006, s. 622 - SCI [o1] 2007 Di Mari, J.F. - Saada, J.I. - Mifflin, R.C. - Valentich, J.D. - Powell, D.W.: American Journal of Physiology-Gastrointestinal and Liver Physiology, Vol. 239, No. 4, 2007, s. G728 - SCI [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5130 - SCI [o1] 2007 Lin, D. - Zhang, J.Y. - Sayre, L.M.: Journal of Organic Chemistry, Vol. 72, No. 25, 2007, s. 9480 - SCI [o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol. 19, No. 2, 2008, s. 263 - SCI [o1] 2008 Fiorucci, S. - Golebiowski, J. - Cabrol-Bass, D. - Antonczak, S.: Proteins-Structure Function and Bioinformatics, Vol. 73, No. 2, 2008, s. 298 - SCI [o1] 2009 Hoffmann, E.K. - Lambert, I.H - Pedersen, S.F.: Physiological Reviews, Vol. 89, No. 1, 2009, s. 277 - SCI [o1] 2009 Gomes, A. - Fernandes, E. - Silva, A.M.S. - Pinto, D.C.G.A. - Santos, C.M.M. - Cavaleiro, J.A.S. - Lima, J.L.F.C.: Biochemical Pharmacology, Vol. 78, No. 2, 2009, s. 177 - SCI [o1] 2010 Adcock, I.M. - Marwick, J. - Casolari, P. - Contoli, M. - Chung, K.F. - Kirkham, P. - Papi, A. Caramori, G.: Current Pharmaceutical Design, Vol. 16, No. 32, 2010, s. 3573 - SCI [o1] 2011 Pontiki, E. - Hadjipavlou-Litina, D. - Litinas, K. - Nicolotti, O. - Carotti, A.: European Journal of Medicinal Chemistry, Vol. 46, No. 1, 2011, s. 200 - SCI [o1] 2011 Li, Y. - Chen, S.H. - Ou, T.M. - Tan, J.H. - Li, D. - Gu, L.Q. - Huang, Z.S.: Bioorganic & Medicinal Chemistry, Vol. 19, No. 6, 2011, s. 2083 - SCI [o1] 2011 Tan, C.M. - Chen, G.S. - Chen, C.S. - Chang, P.T. - Chern, J.W.: Bioorganic & Medicinal Chemistry, Vol. 19, No. 21, 2011, s. 6328 - SCI [o1] 2012 Gomes, A. - Couto, D. - Alves, A. - Dias, I. - Freitas, M. - Porto, G. - Duarte, J.A. - Fernandes, E.: Biofactors, Vol. 38, No. 5, 2012, s. 386 - SCI [o1] 2013 Mathew, G. - Jacob, A. - Durgashivaprasad, E. - Reddy, N.D. - Unnikrishnan, M.K.: International Immunopharmacology, Vol. 15, No. 1, 2013, s. 189 - SCI [o1] 2013 Joshi, N. - Hoobler, E.K. - Perry, S. - Diaz, G. - Fox, B. - Holman, T.R.: Biochemistry, Vol. 52, No. 45, 2013, s. 8035 - SCI [o1] 2014 Meyers, D.A. - Bleecker, E.R. - Holloway, J.W. - Holgate, S.T.: Lancet Respiratory Medicine, Vol. 2, No. 5, 2014, s. 415 - SCI [o1] 2014 Sudha, A. - Srinivasan, P.: Pharmacognosy Magazine, Vol. 10, No. 39, 2014, s. 605 - SCI ADC08 Musiol, Robert (20%) - Jampílek, Josef [UKOEXAF] (20%) - Buchta, Vladimír (5%) - Silva, Luis (10%) - Niedbala, Halina (10%) - Podeszwa, Barbara (10%) - Palka, Anna (5%) - Majerz-Maniecka, Katarzyna (5%) - Oleksyn, Barbara (5%) - Polanski, Jaroslaw(10%): Antifungal properties of new series of quinoline derivatives Lit. 20 zázn. In: Bioorganic and Medicinal Chemistry. - Vol. 14, No. 10 (2006), s. 3592-3598 Registrované v: wos Indikátor časopisu: IF (JCR) 2006=2,624
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Ohlasy (60): [o1] 2006 Metwally, K.A. - Abdel-Aziz, L.M. - Lashine, E.S.M. - Hussemy, M.I. - Badawy, R.H.: Bioorganic & Medicinal Chemistry, Vol. 14, No. 24, 2006, s. 8682 - SCI [o1] 2007 Kamal, A. - Reddy, K.S. - Khan, M.N.A. - Shetty, R.V.C.R.N.C. - Ahmed, S.K. - Kumar, K.P. Murty, U.S.N.: Letters in Drug Design & Discovery, Vol. 4, No. 8, 2007, s. 586 - SCI [o1] 2007 Bouraiou, A. - Belfaitah, A. - Bouacida, S. - Benard-Rocherulle, P. - Carboni, B.: Acta Crystallographica Section E-Structure Reports Online, Vol. 63, 2007, s. O2135 - SCI [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5130 - SCI [o1] 2008 Kaplancikli, Z.A. - Turan-Zitouni, G. - Ozdemir, A. - Revial, G.: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 23, No. 6, 2008, s. 870 - SCI [o1] 2008 Ali, I.A.I. - Fathalla, W. - El Rayes, S.M.: Arkivoc, Part 13, 2008, s. 188 - SCI [o1] 2008 Prasad, A.K. - Kumar, P. - Dhawan, A. - Chhillar, A.K. - Sharma, D. - Yadav, V. - Kumar, M. Jha, H.N. - Olsen, C.E. - Sharma, G.L. - Parmar, V.S.: Bioorganic & Medicinal Chemistry Letters, Vol. 18, No. 6, 2008, s. 2161 - SCI [o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol. 19, No. 2, 2008, s. 263 - SCI [o1] 2008 Abdel-Hafez, S.H. - Hussein, M.A.: Archiv der Pharmazie, Vol. 341, No. 4, 2008, s. 246 - SCI [o1] 2008 Gomez, C.M.M. - Kouznetsov, V.V. - Sortino, M.A. - Alvarez, S.L. - Zacchino, S.A.: Bioorganic & Medicinal Chemistry, Vol. 16, No. 17, 2008, s. 7920 - SCI [o1] 2009 Kaiser, C.R. - Pais, K.C. - de Souza, M.V.N. - Wardell, J.L. - Wardell, S.M.S.V. - Tiekink, E.R.T.: Crystengcomm, Vol. 11, No. 6, 2009, s. 1140 - SCI [o1] 2009 de Souza, M.V.N. - Pais, K.C. - Kaiser, C.R. - Peralta, M.A. - Ferreira, M.D. - Lourenco, M.C.S.: Bioorganic & Medicinal Chemistry, Vol. 17, No. 4, 2008, s. 1480 - SCI [o1] 2009 da Silva, M.A.V.R. - da Silva, M.D.M.C.R. - Ferreira, A.I.M.C.L. - Santos, A.F.L.O.M. - Galvo, T.L.P.: Journal of Chemical Thermodynamics, Vol. 41, No. 10, 2009, s. 1080 - SCI [o1] 2010 Howie, R.A. - de Souza, M.V.N. - Ferreira, M.D. - Kaiser, C.R. - Wardell, J.L. - Wardell, S.M.S.V.: Zeitschrift fur Kristallographie, Vol. 225, No. 10, 2010, s. 447 - SCI [o1] 2010 Chang, F.S. - Chen, W.C. - Wang, C.H. - Tzeng, C.C. - Chen, Y.L.: Bioorganic & Medicinal Chemistry, Vol. 18, No. 1, 2010, s. 133 - SCI [o1] 2010 Avetisyan, A.A. - Aleksanyan, I.L. - Ambartsumyan, L.P.: Russian Journal of Organic Chemistry, Vol. 46, No. 3, 2010, s. 431 - SCI [o1] 2010 Murugesan, S. - Ganguly, S. - Maga, G.: Journal of Chemical Sciences, Vol. 122, No. 2, 2010, s. 176 - SCI [o1] 2010 Fun, H.K. - Chanawanno, K. - Kobkeatthawin, T. - Chantrapromma, S.: Acta Crystallographica Section E-Structure Reports Online, Vol. 66, 2010, s. U3214 - SCI [o1] 2010 Ganguly, S. - Murugesan, S.: Journal of the Indian Chemical Society, Vol. 87, No. 7, 2010, s. 885 - SCI [o1] 2010 Gao, W.T. - Cheng, X.P. - Li, Y.: Heterocycles, Vol. 81, No. 8, 2010, s. 1930 - SCI [o1] 2010 Prabha, K. - Vennila, K.N. - Prasad, K.J.R. - Velmurugan, D.: Acta Crystallographica Section EStructure Reports Online, Vol. 66, 2010, s. U1222 - SCI [o1] 2010 Kumar, S. - Bawa, S. - Drabu, S. - Kumar, R. - Panda, B.P.: Latin American Journal of Pharmacy, Vol. 29, No. 6, 2010, s. 975 - SCI [o1] 2011 El-Agrody, A.M. - Al-Ghamdi, A.M.: Arkivoc, Part 11, 2011, s. 146 - SCI [o1] 2011 Djamel, D. - Tahar, D. - Djahida, H. - Hanane, H. - Salah, C.: Acta Crystallographica Section EStructure Reports Online, Vol. 67, 2011, s. U377 - SCI [o1] 2011 Kumar, S. - Bawa, S. - Kaushik, D. - Panda, B.P.: Archiv der Pharmazie, Vol. 344, No. 7, 2011, s. 480 - SCI [o1] 2011 Thakre, W.B. - Meshram, J.S.: Indian Journal of Heterocyclic Chemistry, Vol. 21, No. 1, 2011, s. 68 - SCI [o1] 2011 Ziemons, E. - Bourichi, H. - Mantanus, J. - Rozet, E. - Lebrun, P. - Essassi, E. - Cherrah, Y. Bouklouze, A. - Hubert, P.: Journal of Pharmaceutical and Biomedical Analysis, Vol. 55, No. 5, 2011, s. 1212 - SCI [o1] 2011 Yang, G.H. - Li, Y.X. - Yan, S.H. - Dai, L. - Zhao, B.: Acta Chimica Sinica, Vol. 69, No. 15, 2011, s. 1750 - SCI [o1] 2011 Kumar, A. - Rao, V.K.: Synlett, No. 15, 2011, s. 2162 - SCI [o1] 2011 Haggag, S.M.S. - Farag, A.A.M. - Mahmoud, M.E.: Polyhedron, Vol. 30, No. 16, 2011, s. 2732 - SCI [o1] 2011 Robak, W. - Apostoluk, W. - Ochromowicz, K.: Journal of Chemical and Engineering Data, Vol. 56, No. 11, 2011, s. 3983 - SCI
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[o1] 2011 Alshahateet, S.F. - Al-Zereini, W.A. - Alghezawi, N.M.: Journal of Chemical Crystallography, Vol. 41, No. 12, 2011, s. 1811 - SCI [o1] 2012 Thapa, P. - Lee, E.S.: Bulletin of the Korean Chemical Society, Vol. 33, No. 5, 2012, s. 1772 SCI [o1] 2012 Li, V.M. - Gavrishova, T.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 48, No. 6, 2012, s. 828 - SCI [o1] 2012 Kouznetsov, V.V. - Gomez, C.M.M. - Derita, M.G. - Svetaz, L. - del Olmo, E. - Zacchino, S.A.: Bioorganic & Medicinal Chemistry, Vol. 20, No. 21, 2012, s. 6512 - SCI [o1] 2012 Tukulula, M. - Little, S. - Gut, J. - Rosenthal, P.J. - Wan, B.J. - Franzblau, S.G. - Chibale, K.: European Journal of Medicinal Chemistry, Vol. 57, 2012, s. 267 - SCI [o1] 2012 El-Agrody, A.M. - Khattab, E.S.A.E.H. - Fouda, A.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research, Vol. 21, No. 12, 2012, s. 4213 - SCI [o1] 2013 Goncalves, R.S.B. - de Souza, M.V.N. - Wardell, J.L. - Wardell, S.M.S.V.: Zeitschrift fur Kristallographie, Vol. 228, No. 12, 2013, s. 668 - SCI [o1] 2013 Savegnago, L. - Vieira, A.I. - Seus, N. - Goldani, B.S. - Castro, M.R. - Lenardao, E.J. - Alves, D.: Tetrahedron Letters, Vol. 54, No. 1, 2013, s. 44 - SCI [o1] 2013 Derita, M. - Montenegro, I. - Garibotto, F. - Enriz, R.D. - Fritis, M.C. - Zacchino, S.A.: Molecules, Vol. 18, No. 2, 2013, s. 2051 - SCI [o1] 2013 Serrao, E. - Debnath, B. - Otake, H. - Kuang, Y.T. - Christ, F. - Debyser, Z. - Neamati, N.: Journal of Medicinal Chemistry, Vol. 56, No. 6, 2013, s. 2322 - SCI [o1] 2013 Sun, W.Q. - Yuan, G.Z. - Liu, J.X. - Ma, L. - Liu, C.B.: Spectrochimica Acta Part A-Molecular and Biomolecular Spectroscopy, Vol. 106, 2013, s. 283 - SCI [o1] 2013 Patel, R.V. - Kumari, P. - Chikhalia, K.H.: Medicinal Chemistry, Vol. 9, No. 4, 2013, s. 607 SCI [o1] 2013 De Leon, F. - Kalagara, S. - Navarro, A.A. - Mito, S.: Tetrahedron Letters, Vol. 54, No. 24, 2013, s. 3149 - SCI [o1] 2013 Vandekerckhove, S. - Tran, H.G. - Desmet, T. - D'hooghe, M.: Bioorganic & Medicinal Chemistry, Letters, Vol. 23, No. 16, 2013, s. 4643 - SCI [o1] 2013 Boechat, N. - Bastos, M.M.: Current Topics in Medicinal Chemistry, Vol. 13, No. 22, 2013, s. 2904 - SCI [o1] 2014 Gok, D. - Kasimogullari, R. - Cengiz, M. - Mert, S.: Journal of Heterocyclic Chemistry, Vol. 51, No. 1, 2014, s. 232 - SCI [o1] 2014 Yernale, N.G. - Mathada, M.B.H.: Bioinorganic Chemistry and Applications, 2014, Article No. 314963 - SCI [o1] 2014 Ahmed, A. - Dhara, S. - Singha, R. - Nuree, Y. - Sarkar, P. - Ray, J.K.: RSC Advances, Vol. 4, No. 95, 2014, s. 53141 - SCI [o1] 2014 Peng, H.K. - Lin, I.L. - Lee, C.C. - Wang, L.Y. -Tzeng, C.C. - Chang, J.G. - Yang, S.C.: Medicinal Chemistry Research, Vol. 23, No. 3, 2014, s. 1446 - SCI [o1] 2014 Patel, A.B. - Kumari, P. - Chikhalia, K.H.: Catalysis Letters, Vol. 144, No. 7, 2014, s. 1338 SCI [o1] 2014 Gavrishova, T.N. - Li, V.M. - Karpov, O.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 50, No. 8, 2014, s. 1144 - SCI [o1] 2014 Haggag, S.M.S. - Farag, A.A.M. - Refea, M.A.: Thin Solid Films, Vol. 566, 2014, s. 44 - SCI [o1] 2014 Vairavelu, L. - Prasad, K.J.R.: Journal of Chemical Sciences, Vol. 126, No. 6, 2014, s. 1902 SCI [o1] 2015 Yadav, T. - Kishore, D. - Singh, B.: British Journal of Pharmaceutical Research, Vol. 8, No. 3, 2015, Article No. 19615 - SCI [o1] 2015 Akhter, M. - Saha, R. - Tanwar, O. - Alam, M.M. - Zaman, M.S.: Medicinal Chemistry Research, Vol. 24, No. 2, 2015, s. 890 - SCI [o1] 2015 Li, Y.Q. - Chibale, K. - Smith, G.S.: Journal of Chemical Crystallography, Vol. 45, No. 4, 2015, s. 206 - SCI [o1] 2015 Tummatorn, J. - Poonsilp, P. - Nimnual, P. - Janprasit, J. - Thongsornkleeb, C. - Ruchirawat, S.: Journal of Organic Chemistry, Vol. 80, No. 9, 2015, s. 4525 - SCI [o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI [o1] 2015 Cho, S.K. - Song, J.H. - Lee, E.J. - Lee, D.H. - Hahn, J.T. - Jung, D.I.: Bulletin of the Korean Chemical Society, Vol. 36, No. 11, 2015, s. 2749 - SCI ADC09 Vinšová, Jarmila (20%) - Čermáková, Kateřina (10%) - Tomečková, Alexandra (10%) - Jampílek, Josef [UKOEXAF] (10%) - Čermák, Pavel (10%) - Kuneš, Jiří (10%) - Doležal, Martin (10%) - Štaud, František (10%) - Čečková, Martina (10%): Synthesis andantimicrobial evaluation of new 2-substituted 5,7-di-tertbutylbenzoxazoles
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Lit. 31 zázn. In: Bioorganic and Medicinal Chemistry. - Vol. 14, No. 17 (2006), s. 5850-5865 Registrované v: wos Indikátor časopisu: IF (JCR) 2006=2,624 Ohlasy (51): [o1] 2007 Janin, Y.L.: Bioorganic & Medicinal Chemistry, Vol. 15, No. 7, 2007, s. 2513 - SCI [o1] 2007 Hioki, H. - Matsushita, K. - Kubo, M. - Harada, K. - Kodama, M. - Fukuyama, Y.: Tetrahedron, Vol. 63, No. 46, 2007, s. 11324 - SCI [o1] 2008 Soni, K. - Samota, M.K. - Jhajharia, P. - Seth, G.: Phosphorus Sulfur and Silicon and the Related Elements, Vol. 183, No. 11, 2008, s. 2853 - SCI [o1] 2008 Kumar, D. - Rudrawar, S. - Chakraborti, A.K.: Australian Journal of Chemistry, Vol. 61, No. 11, 2008, s. 887 - SCI [o1] 2008 Gottumukkala, A.L. - Derridj, F. - Djebbar, S. - Doucet, H.: Tetrahedron Letters, Vol. 49, No. 18, 2008, s. 2930 - SCI [o1] 2008 Evangelio, E. - Saiz-Poseu, J. - Maspoch, D. - Wurst, K. - Busque, F. - Ruiz-Molina, D.: European Journal of Inorganic Chemistry, No. 14, 2008, s. 2285 - SCI [o1] 2008 Salcedo, A. - Neuville, L. - Zhu, J.P.: Journal of Organic Chemistry, Vol. 73, No. 9, 2008, s. 3603 - SCI [o1] 2008 Siddiqui, N. - Sarafroz, M. - Alam, M.M. - Ahsan, W.: Acta Poloniae Pharmaceutica, Vol. 65, No. 4, 2008, s. 455 - SCI [o1] 2008 Costa, S.P.G. - Oliveira, E. - Lodeiro, C. - Raposo, M.M.M.: Tetrahedron Letters, Vol. 49, No. 36, 2008, s. 5261 - SCI [o1] 2009 Heravi, M.M. - Baghernejad, B. - Oskooie, H.A.: Chinese Journal of Chemistry, Vol. 27, No. 2, 2009, s. 383 - SCI [o1] 2009 Kumar, A. - Maurya, R.A. - Ahmad, P.: Journal of Combinatorial Chemistry, Vol. 11, No. 2, 2009, s. 201 - SCI [o1] 2009 Horvati, K. - Mezo, G. - Szabo, N. - Hudecz, F. - Bosze, S.: Journal of Peptide Science, Vol. 15, No. 5, 2009, s. 391 - SCI [o1] 2009 Klimesova, V. - Koci, J. - Waisser, K. - Kaustova, J. - Mollmann, U.: European Journal of Medicinal Chemistry, Vol. 44, No. 5, 2009, s. 2293 - SCI [o1] 2009 Husain, A. - Akhter, M.S.A. - Khatoon, Y.: Indian Journal of Heterocyclic Chemistry, Vol. 19, No. 1, 2009, s. 94 - SCI [o1] 2009 Chen, W.H. - Pang, Y.: Tetrahedron Letters, Vol. 50, No. 48, 2009, s. 6683 - SCI [o1] 2010 Kumar, A. - Maurya, R.A. - Saxena, D.: Molecular Diversity, Vol. 15, No. 2, 2010, s. 341 [o1] 2010 Chauhan, P.M.S. - Sunduru, N. - Sharma, M.: Future Medicinal Chemistry, Vol. 2, No. 9, 2010, s. 1500 - SCI [o1] 2010 Kumar, A. - Sharma, S. - Maurya, R.A.: Tetrahedron Letters, Vol. 51, No. 48, 2010, s. 6226 SCI [o1] 2010 Rossi, R. - Bellina, F. - Lessi, M.: Synthesis-Stuttgart, No. 24, 2010, s. 4153 - SCI [o1] 2011 Sun, Q. - Wu, R.Z. - Cai, S.T. - Lin, Y.A. - Sellers, L. - Sakamoto, K. - He, B.A. - Peterson, B.R.: Journal of Medicinal Chemistry, Vol. 54, No. 5, 2011, s. 1139 - SCI [o1] 2011 Chari, M.A. - Shobha, D. - Sasaki, T.: Tetrahedron Letters, Vol. 52, No. 43, 2011, s. 5580 - SCI [o1] 2012 Vaillard, V.A. - Guastavino, J.F. - Buden, M.E. - Bardagi, J.I. - Barolo, S.M. - Rossi, R.A.: Journal of Organic Chemistry, Vol. 77, No. 3, 2012, s. 1519 - SCI [o1] 2012 Horvati, K. - Bacsa, B. - Szabo, N. - David, S. - Mezo, G. - Grolmusz, V. - Vertessy, B. Hudecz, F. - Bosze, S.: Bioconjugate Chemistry, Vol. 223, No. 5, 2012, s. 907 - SCI [o1] 2012 Aparaschivei, R. - Holban, M. - Sunel, V. - Popa, M. - Desbrieres, J.: Cellulose Chemistry and Technology, Vol. 46, No. 5-6, 2012, s. 306 - SCI [o1] 2012 Li, Y. - Tao, X.Y. - Lin, G.H. - Gao, W.T.: Heterocyclic Communications, Vol. 18, No. 4, 2012, s. 210 - SCI [o1] 2012 Gao, W.T. - Lin, G.H. - Li, Y. -Tao, X.Y. - Liu, R. - Sun, L.J.: Beilstein Journal of Organic Chemistry, Vol. 8, 2012, s. 1857 - SCI [o1] 2012 Abdou, W.M. - Barghash, R.F. - Sediek, A.A.: European Journal of Medicinal Chemistry, Vol. 57, 2012, s. 372 - SCI [o1] 2013 Salehzadeh, H. - Nematollahi, D. - Hesari, H.: Green Chemistry, Vol. 15, No. 9, 2013, s. 2446 SCI [o1] 2013 Nieddu, G. - Giacomelli, G.: Tetrahedron, Vol. 69, No. 2, 2013, s. 795 - SCI [o1] 2013 Protasenko, N.A. - Poddel'sky, A.I. - Bogomyakov, A.S. - Somov, N.V. - Abakumov, G.A. Cherkasov, V.K.: Polyhedron, Vol. 49, No. 1, 2013, s. 243 - SCI
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[o1] 2013 Park, H.J. - Park, M.S. - Lee, T.H. - Park, K.H.: Journal of Heterocyclic Chemistry, Vol. 50, No. 3, 2013, s. 667 - SCI [o1] 2013 Abdou, W.M. - Barghash, R.F. - Khidre, R.E.: Monatshefte fur Chemie, Vol. 144, No. 8, 2013, s. 1242 - SCI [o1] 2013 Arisoy, M. - Temiz-Arpaci, O. - Kaynak-Onurdag, F. - Ozgen, S.: Zeitschrift fur Naturforschung Section C-A Journal of Biosciences, Vol. 68, No. 11-12, 2013, s. 460 - SCI [o1] 2013 Li, A.K. - Ma, H.Y. - Huang, J.L.: Organometallics, Vol. 32, No. 24, 2013, s. 7469 - SCI [o1] 2014 Rana, D.N. - Chhabria, M.T. - Shah, N.K. - Brahmkshatriya, P.S.: Medicinal Chemistry Research, Vol. 23, No. 1, 2014, s. 381 - SCI [o1] 2014 Abdou, W.M. - Ganoub, N.A. - Barghash, R.F.: Synthetic Communications, Vol. 44, No. 18, 2014, s. 2678 - SCI [o1] 2014 Ashfaq, M. - Shah, S.S.A. - Najam, T. - Ahmad, M.M. - Tabassum, R. - Rivera, G.: Current Medicinal Chemistry, Vol. 21, No. 7, 2014, s. 931 - SCI [o1] 2014 Pardeshi, S.D. - Sonar, J.P. - Pawar, S.S. - Dekhane, D. - Gupta, S. - Zine, A.M. - Thore, S.N.: Journal of the Chilean Chemical Society, Vol. 59, No. 1, 2014, s. 2340 - SCI [o1] 2014 Rana, D.N. - Chhabria, M.T. - Shah, N.K. - Brahmkshatriya, P.S.: Medicinal Chemistr Research, Vol. 23, No. 5, 2014, s. 2228 - SCI [o1] 2014 Haider, S. - Alam, M.S. - Hamid, H. - Shafi, S. - Dhulap, A. - Hussain, F. - Alam, P. - Umar, S. Pasha, M.A.Q. - Bano, S. - Nazreen, S. - Ali, Y. - Kharbanda, C.: European Journal of Medicinal Chemistry, Vol. 81, 2014, s. 217 - SCI [o1] 2014 Aparaschivei, R. - Sunel, V. - Popa, M. - Desbrieres, J.: Journal of Heterocyclic Chemistry, Vol 51, No. 4, 2014, s. 1132 - SCI [o1] 2014 Abdou, W.M. - Ganoub, N.A. - Sabry, E.: Acta Pharmaceutica, Vol. 64, No. 3, 2014, s. 284 SCI [o1] 2014 Barghash, R.F. - Ganoub, N.A. - Abdou, W.M.: Monatshefte fur Chemie, Vol. 145, No. 10, 2014, s. 1630 - SCI [o1] 2014 Horvati, K. - Bacsa, B. - Kiss, E. - Gyulai, G. - Fodor, K. - Balka, G. - Rusvai, M. - Szabo, E. Hudecz, F. - Bosze, S.: Bioconjugate Chemistry, Vol. 25, No. 12, 2014, s. 2268 - SCI [o1] 2015 Zhang, X.X. - Lin, Y.Y. - Zhang, J. - Cao, S.: RSC Advances, Vol. 5, No. 11, 2014, s. 7908 SCI [o1] 2015 Kochem, A. - Gellon, G. - Jarjayes, O. - Philouze, C. - d'Hardemare, A.D. - van Gastel, M. Thomas, F.: Dalton Transactions, Vol. 44, No. 28, 2015, s. 12756 - SCI [o1] 2015 VenkatRamani, S. - Ghiviriga, I. - Abboud, K.A. - Veige, A.S.: Dalton Transactions, Vol. 44, No. 42, 2015, s. 18486 - SCI [o1] 2015 Khandan-Barani, K. - Maghsoodlou, M.T. - Hassanabadi, A. - Hosseini-Tabatabaei, M.R. Saffari, J. - Kangani, M.: Research on Chemical Intermediates, Vol. 41, No. 5, 2015, s. 3016 - SCI [o1] 2015 Lv, M.Y. - Zheng, H.M. - Li, Y. - Gao, W.T.: Research on Chemical Intermediates, Vol. 41, No. 10, 2015, s. 6939 - SCI [o1] 2015 Abdou, W.M. - Kamel, A.A. - Khidre, M.D.: Journal of Heterocyclic Chemistry, Vol 52, No. 6, 2015, s. 1662 - SCI [o1] 2015 Qiu, J. - Zhang, Y.D. - Hua, C.W. - Gou, X.F. - Chen, B. - Zhao, J.L.: Heterocycles, Vol. 91, No. 11, 2015, s. 2162 - SCI ADC10 Imramovský, Aleš (20%) - Polanc, Slovenko (10%) - Vinšová, Jarmila (20%) - Kočevar, Marijan (10%) - Jampílek, Josef [UKOEXAF] (15%) - Rečková, Zuzana (15%) - Kaustová, Jarmila (10%): A new modification of anti-tubercular active molecules Lit. 25 zázn. In: Bioorganic and Medicinal Chemistry. - Vol. 15, No. 7 (2007), s. 2551-2559 Registrované v: wos Indikátor časopisu: IF (JCR) 2007=2,662 Ohlasy (46): [o1] 2007 Rollas, S. - Kucukguzel, S.G.: Molecules, Vol. 12, No. 8, 2007, s. 1939 - SCI [o1] 2008 Fun, H.K. - Chantrapromma, S. - Jana, S. - Hazra, A. - Goswami, S.: Acta Crystallographica Section E-Structure Reports Online, Vol. 64, 2008, s. U4082 - SCI [o1] 2008 Turan-Zitouni, G. - Ozdemir, A. - Kaplancikli, Z.A. - Benkli, K. - Chevallet, P. - Akalin, G.: European Journal of Medicinal Chemistry, Vol. 43, No. 5, 2008, s. 985 - SCI [o1] 2009 Abdel-Rahman, H.M. - El-Koussi, N.A. - Hassan, H.Y.: Archiv der Pharmazie, Vol. 342, No. 8, 2009, s. 99 - SCI [o1] 2009 Rogoza, L.N. - Salakhutdinov, N.F. - Tolstikov, G.A.: Mini-Reviews in Organic Chemistry, Vol. 6, No. 2, 2009, s. 151 - SCI
8
[o1] 2010 Ajani, O.O. - Obafemi, C.A. - Nwinyi, O.C. - Akinpelu, D.A.: Bioorganic & Medicinal Chemistry, Vol. 18, No. 1, 2010, s. 221 - SCI [o1] 2010 Eswaran, S. - Adhikari, A.V. - Pal, N.K. - Chowdhury, I.H.: Bioorganic & Medicinal Letters, Vol. 20, No. 3, 2010, s. 1044 - SCI [o1] 2010 Abdel-Aal, W.S. - Hassan, H.Y. - Aboul-Fadl, T. - Youssef, A.F.: European Journal of Medicinal Chemistry, Vol. 45, No. 3, 2010, s. 1106 - SCI [o1] 2010 Turan-Zitouni, G. - Kaplancikli, Z.A. - Ozdemir, A.: European Journal of Medicinal Chemistry, Vol. 45, No. 5, 2010, s. 2088 - SCI [o1] 2010 Patel, N.B. - Patel, V.N. - Patel, H.R. - Shaikh, F.M. - Patel, J.C.: Acta Poloniae Pharmaceutica, Vol. 67, No. 3, 2010, s. 275 - SCI [o1] 2010 Sharma, P.C. - Jain, A. - Jain, S. - Pahwa, R. - Yar, M.S.: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 25, No. 4, 2010, s. 589 - SCI [o1] 2010 Abdel-Aziz, M. - Abdel-Rahman, H.M.: European Journal of Medicinal Chemistry, Vol. 45, No. 8, 2010, s. 3388 - SCI [o1] 2010 Chauhan, P.M.S. - Sunduru, N. - Sharma, M.: Future Medicinal Chemistry, Vol. 2, No. 9, 2010, s. 1500 - SCI [o1] 2010 Wiles, J.A. - Bradbury, B.J. - Pucci, M.J.: Expert Opinion on Therapeutic Patents, Vol. 20, No. 10, 2010, s. 1319 - SCI [o1] 2010 Patel, N.B. - Patel, J.C. - Patel, V.N.: Chinese Journal of Chemistry, Vol. 28, No. 10, 2010, s. 1997 - SCI [o1] 2010 Mantu, D. - Luca, M.C. - Moldoveanu, C. - Zbancioc, G. - Mangalagiu, I.I.: European Journal of Medicinal Chemistry, Vol. 45, No. 11, 2010, s. 5168 - SCI [o1] 2011 Jiang, X.L. - Cui, Y.B. - Cao, S.H.: Zhongguo Kangshengsu Zazhi, Vol. 36, No. 4, 2011, s. 263 - SCI [o1] 2011 Joshi, R.S. - Mandhane, P.G. - Badadhe, P.V. - Gill, C.H.: Ultrasonics Sonochemistry, Vol. 18, No. 3, 2011, s. 738 - SCI [o1] 2011 Khidre, R.E. - Abu-Hashem, A.A. - El-Shazly, M.: European Journal of Medicinal Chemistry, Vol. 46, No. 10, 2011, s. 5064 - SCI [o1] 2012 Shaquiquzzaman, M. - Khan, S.A. - Amir, M. - Alam, M.M.: Saudi Pharmaceutical Journal, Vol. 20, No. 2, 2012, s. 154 - SCI [o1] 2012 Gaikwad, N.D. - Patil, S.V. - Bobade, V.D.: Bioorganic & Medicinal Chemistry Letters, Vol. 22, No. 10, 2012, s. 3454 - SCI [o1] 2012 Malhotra, M. - Sharma, S. - Deep, A.: Medicinal Chemistry Research, Vol. 21, No. 7, 2012, s. 1244 - SCI [o1] 2012 Malhotra, M. - Sharma, S. - Deep, A.: Acta Poloniae Pharmaceutica, Vol. 69, No. 4, 2012, s. 644 - SCI [o1] 2012 Gaikwad, N.D. - Patil, S.V. - Bobade, V.D.: European Journal of Medicinal Chemistry, Vol. 54, 2012, s. 302 - SCI [o1] 2012 Wang, S. - Jia, X.D. - Liu, M.L. - Lu, Y. - Guo, H.Y.: Bioorganic & Medicinal Chemistry Letters, Vol. 22, No. 18, 2012, s. 5975 - SCI [o1] 2012 Sarnpitak, P. - Tsirulnikov, S. - Krasavin, M.: Tetrahedron Letters, Vol. 53, No. 48, 2012, s. 6543 - SCI [o1] 2012 Judge, V. - Narasimhan, B. - Ahuja, M.: Medicinal Chemistry Research, Vol. 21, No. 12, 2012, s. 3957 - SCI [o1] 2012 Shaquiquzzaman, M. - Khan, S.A. - Amir, M. - Alam, M.M.: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 27, No. 6, 2012, s. 831 - SCI [o1] 2013 Rudrapal, M. - Satyanandam, R.S. - Swaroopini, T.S. - Lakshmi, T.N. - Jaha, S.K. - Zaheera, S.: Medicinal Chemistry Research, Vol. 22, No. 6, 2013, s. 2846 - SCI [o1] 2013 Matei, L. - Bleotu, C. - Baciu, I. - Draghici, C. - Ionita, P. - Paun, A. - Chifiriuc, M.C. - Sbarcea, A. - Zarafu, I.: Bioorganic & Medicinal Chemistry, Vol. 21, No. 17, 2013, s. 5361 - SCI [o1] 2013 Hagar, M. - Soliman, S.M. - Ibid, F. - El Ashry, E.H.: Journal of Moleular Structure, Vol. 1049, 2013, s. 188 - SCI [o1] 2013 Anbazhagan, R. - Sankaran, K.R.: Journal of Moleular Structure, Vol. 1050, 2013, s. 80 - SCI [o1] 2013 Refat, H.M. - Fadda, A.A.: European Journal of Medicinal Chemistry, Vol. 70, 2013, s. 426 SCI [o1] 2014 Refat, H.M. - Fadda, A.A.: Synthetic Communications, Vol. 44, No. 15, 2014, s. 2154 - SCI [o1] 2014 Bhat, M.A.: Acta Poloniae Pharmaceutica, Vol. 71, No. 5, 2014, s. 770 - SCI [o1] 2014 Malhotra, M. - Sharma, R. - Rathee, D. - Phogat, P. - Deep, A.: Arabian Journal of Chemistry, Vol. 7, No. 5, 2014, s. 671 - SCI
9
[o1] 2014 dos Reis, F.D. - Gatti, I.C. - Garcia, H.C. - de Oliveira, V.E. - de Oliveira, L.F.C.: Journal of Physical Chemistry A, Vol. 118, No. 49, 2014, s. 11528 - SCI [o1] 2015 Saha, R. - Alam, M.M. - Akhter, M.: RSC Advances, Vol. 5, No. 17, 2015, s. 12820 - SCI [o1] 2015 Mathew, B. - Suresh, J. - Ahsan, M.J. - Mathew, G.E. - Usman, D. - Subramanyan, P.N.S. Safna, K.F. - Maddela, S.: Infectious Disorders - Drug Targets, Vol. 15, No. 2, 2015, s. 88 - SCI [o1] 2015 Anbazhagan, R. - Sankaran, K.R.: Spectrochimica Acta Part A-Molecular and Biomolecular Spectroscopy, Vol. 135, 2015, s. 993 - SCI [o1] 2015 Kamble, R.D. - Hese, S.V. - Meshram, R.J. - Kote, J.R. - Gacche, R.N, - Dawane, B.S.: Medicinal Chemistry Research, Vol. 24, No. 3, 2015, s. 1088 - SCI [o1] 2015 Casanova, B.B. - Muniz, M.N. - de Oliveira, T. - de Oliveira, L.F. - Machado, M.M. Fuentefria, A.M. - Gosmann, G. - Gnoatto, S.C.B.: Molecules, Vol. 20, No. 5, 2015, s. 9241 - SCI [o1] 2015 Refat, H.M. - Fadda, A.A.: Heterocycles, Vol. 91, No. 6, 2015, s. 1226 - SCI [o1] 2015 Yurttas, L. - Kaplancikli, Z.A. - Canturk, Z. - Gencer, H.K.: Phosphorus Sulfur and Silicon and the Related Elements, Vol. 190, No. 7, 2015, s. 1191 - SCI [o1] 2015 El-Faham, A. - Farooq, M. - Khattab, S.N. - Abutaha, N. - Wadaan, M.A. - Ghabbour, H.A. Fun, H.K.: Molecules, Vol. 20, No. 8, 2015, s. 14655 - SCI [o1] 2015 Dikkar, A.B. - Pethe, G.B. - Aswar, A.S.: Russian Journal of Physical Chemistry A, Vol. 89, No. 12, 2015, s. 2203 - SCI ADC11 Musiol, Robert (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Richardson, Des R. (10%) Kalinowski, Danuta (10%) - Podeszwa, Barbara (10%) - Finster, Jacek (10%) - Niedbala, Halina (10%) Palka, Anna (10%) - Polański, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (10%): Investigating biological activity spectrum for novel quinoline analogues Lit.: 32 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 15, No. 3 (2007), s. 1280-1288 Registrované v: wos Indikátor časopisu: IF (JCR) 2007=2,662 Ohlasy (74): [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5120-5130 - SCI [o1] 2008 Gabriele, B. - Mancuso, R. - Salerno, G. - Lupinacci, E. - Ruffulo, G. - Costa, M.: J. Org. Chem., Vol. 73, No. 13, 2008, s. 4971-4977 - SCI [o1] 2008 Mendelez-Homez, C.M. - Kouznetsov, V.V. - Sortino, M.A. - Alvarez, S.L. - Zacchino, S.A.: Bioorg. Med. Chem., Vol. 16, No. 17, 2008, s. 7908-7920 - SCI [o1] 2008 Madapa, S. - Tusi, Z. - Batra, S.: Current Organic Chemistry, Vol. 12, No. 13, 2008, s. 11161183 - SCI [o1] 2008 Shindoh, N. - Tokuyama, H. - Takemoto, Y. - Takasu, K.: Journal of Organic Chemistry, Vol. 73, No. 19, 2008, s. 7451-7456 - SCI [o3] 2008 Batra, M.K. - Batra, C. - Ojha, K.G.: Medicinal Chemistry Research, Vol. 17, No. 9, 2008, s. 604-617 [o1] 2009 Schmidt, F. - Champy, P. - Séon-Méniel, B. - Franck, X. - Raisman-Vozari, R. - Figadere, B.: PLoS ONE, Vol. 4, No. 7, 2009, S. Article no. e6215 - SCOPUS [o1] 2009 Lee, C.H. - Lee, H.S.: Journal of the Korean Society for Applied Biological Chemistry, Vol. 52, No. 4, 2009, s. 331-335 - SCI [o1] 2010 Garcia-Santos, I. - Sanmartin, J. - Garcia-Deibe, A.M. - Fondo, M. - Gómez, E.: Inorganica Chimica Acta, Vol. 363, No. 1, 2010, s. 193-198 - SCI [o1] 2010 Chang, F.S. - Chen, W. - Wang, C. - Tzeng, C.C. - Chen, Y.L.: Bioorganic & Medicinal Chemistry, Vol. 18, No. 1, 2010, s. 124-133 - SCI [o1] 2009 Malakyan, M.G. - Badzhinyan, S.A. - Vardevanyan, L.A. - Grigoryan, D.S. - Egiazaryan, D.É. Avetisian, A.A. - Aleksanyan, I.L. - Ambartsumyan, L.P. - Sargsyan, K.S.: Pharmaceutical Chemistry Journal, Vol. 43, No. 1, 2009, . 7-10 -SCI [o1] 2009 Rajakumar, P. - Raja, R. - Selvam, S. - Rengasamy, R. - Nagaraj, S.: Bioorganic & Medicinal Chemistry Letters, Vol. 19, No. 13, 2009, s. 3466-3470 - SCI [o1] 2009 Shen, M.G. - Cai, C. - Yi, W.B.: Journal of Hetecyclic Chemistry Chemistry, Vol. 46, No. 4, 2009, s. 796-799 - SCI [o1] 2009 Erenler, R. - Uno, M. - Goud, T.V. - Biellmann, J.F.: Journal of Chemical Research-S, No. 7, 2009, s. 459-464 - SCI [o1] 2009 Barluenga, J. - Rodriguez, F. - Fananas, F.J.: Chemistry - An Asian Journal, Vol. 4, No. 7, 2009, s. 1036-1048 - SCI
10
[o1] 2010 Broch, S. - Aboab, B. - Anizon, F. - Moreau, P.: European Journal of Medicinal Chemistry, Vol. 45, No. 4, 2010, s. 1657-1662 - SCI [o1] 2010 Bhatt, H.G. - Agrawal, Y.K.: Medicinal Chemistry Research, Vol. 19, No. 4, 2010, s. 392-402 SCI [o1] 2010 Pinheiro, L.M.V. - Ventura, M.C.M.M. - Moita, M.L.C.J.: Journal of Molecular Liquids, Vol. 154, No. 2-3, 2010, s. 102-110 - SCI [o1] 2010 Rajakumar, P. - Raja, R.: Tetrahedron Letters, Vol. 51, No. 33, 2010, s. 4365-4370 - SCI [o3] 2009 Chang, F.S.: Synthesis and Antiproliferative Evaluations of 2-Phenylvinylquinoline (2Styrylquinoline) and 2-Furanylvinylquinoline Derivatives. Kaohsiung City : Kaohsiung Medical University, 2009, S. 151 [o3] 2008 Chao, S.T.: Syntheses of Quinolino-fused Bicyclo [2.2.2] octadienes and Sesquibicyclo [2.2.2] octadienes from Friedländer Reaction. Taichung : Thunghai University, 2008, S. 156 [o3] 2010 Rachid, O.: Synthese de bromocétones quinoléiques précurseurs de Produits d´intéret biologique. Batna : Université de Batna, 2010, S. 10, 71 [o1] 2011 Yang, G.H. - Li, Y.X. - Yan, S.H. - Dai, L. - Zhao, B.: Acta Chimica Sinica, Vol. 69, No. 15, 2011, s. 1743-1750 - SCI [o1] 2011 Saugues, E. - Nauton, L. - Théry, V. - Anizon, F. - Moreau, P.: Bioorganic Chemistry, Vol. 39, No. 4, 2011, s. 143-150 - SCOPUS [o1] 2011 Zhang, W.X. - Dai, Y.S. - Wang, X.R. - Zhang, W.: Tetrahedron Letters, Vol. 52, No. 46, 2011, s. 6122-6126 - SCOPUS [o3] 2011 Reis, D.C.: Estudo do perfil farmacológico de novas tiossemicarbazonas e novos complexos de bismuto(III) e antimônio(III). Belo Horizonte : [s.n.], 2011, S. 6 [o1] 2011 Thakre, W. B. - Meshram, J. S.: Indian Journal of Heterocyclic Chemistry, Vol. 21, Iss. 1, 2011, s. 65-68 - SCI [o1] 2011 El-Agrody, A. M. - Al-Ghamdi, A. M.: Arkivoc, Part 11, 2011, s. 134-146 - SCI [o1] 2012 Peng, H.K. - Lin, C.K. - Yang, S.Y. - Tseng, C.K. - Tzeng, C.C. - Lee, J.C. - Yang, S.C.: Bioorganic and Medicinal Chemistry Letters, Vol. 22, Iss. 2, 2012, s. 1107-1110 - SCI ; SCOPUS [o1] 2012 Tyagi, R. - Singh, B. - Kishore, D.: Journal of Chemical Sciences, Vol. 124, Iss. 2, 2012, s. 431435 - SCI ; SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, Iss. 6, 2012, s. 2928-2936 - SCOPUS [o3] 2011 Li Runlai - Li Shuan - Zhang Zhenming - Ma Xiaobo - Wu Qiong: Study on Synthetic Process of 5,7-dinitro-8-hydroxy-2-Methylquinoline. In: Chemical Industry Times, Vol. 25, Iss. 9, 2011, s. 1-8 [o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied Photosynthesis. Rijeka : InTech, 2012, S. 1-22 [o3] 2011 Pandey, H. - Mehta, P. - Pathak, A.K. - Soni, H.: 2D-QSAR study of 4-(4-alkoxylphenyl)-3ethyl-4H-1,2,4-triazoles as open-chain analogues of 7-alkoxyl-4,5-dihydro[1,2,4]triazolo[4,3-a] quinolines. In: Journal of Pharmacy Research,Vol. 4, No. 5, 2011, s. 1349-1352 [o3] 2011 Soto-Lopez, A. F. - Meneses, J. P. - Saez-Vega, J. - Camargo, M.: Cytotoxicity evaluation of new styrylquinoline analogues in leukemoid jurkat cells. In: Actualidades Biologicas, Vol.33, No. 95, 2011, s. 165-172 [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o1] 2012 Li, V.M. - Gavrishova, T.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 48, No. 6, 2012, s. 823-828 - SCOPUS [o1] 2012 El-Agrody, A.M. - Khattab, E.S.A.E.H. - Fouda, A.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research, Vol. 21, No. 12, 2012, s. 4200-4213 - SCI [o1] 2012 Kouznetsov V.V. - Meléndez Gómez C.M. - Derita M.G. - Svetaz L. - del Olmo E. - Zacchino S.A.: Bioorganic & Medicinal Chemistry, Vol. 20, No. 21, 2012, s. 6506-6512 - SCI ; SCOPUS [o3] 2011 Yang Z. - Fang Z. - Wang Z.X.: Synthesis of - 2,5 - dihydro - 3,6 -dimethoxy - 2 isopropylpyrazine. In: Chemical Industry Times, Vol. 24, No. 9, 2011, s. 6-8 [o1] 2013 Sun, W. - Yuan, G. - Liu, J. - Ma, L. - Liu, C.: Spectrochimica Acta - Part A: Molecular and Biomolecular Spectroscopy, Vol. 106, 2013, s. 275-283 - SCOPUS [o1] 2013 El-Agrody, A.M. - Abd-Rabboh, H.S.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research, Vol. 22, Iss. 3, 2013, s. 1339-1355 - SCI ; SCOPUS [o3] 2013 Kondaiah, S. - Nagarajareddy, G. - Rajesh, D. - Mallikarjuna Rao, R. - Sree Ramulu, J.: Synthesis, Structural Characterization and Anti-bacterial Activity of some Novel Schiff Base Ligans and their Vanadium (IV) Metal Complexes. In: IJPI s Journal of Drug Chemistry, Vol 3, No. 12, 2013, Nestr. http://ijpijournals.com/Articles/PDF/379.pdf
11
[o3] 2013 Sales, E.S. - Schneider, J.M.F.M. – Merlo, A.A.: Síntese Tricomponente de Novos Materiais Funcionais Quinolínicos. In: XIX Encontro da Quimica de Regiao Sul. Zborník. Tubarao : Universidade do Sul de Santa Catarina, 2012, Nestr.http://ijpijournals.com/Articles/PDF/379.pdf [o3] 2011 Shridhar Bhat - Curtis Chong, R. - Jun Liu, O - Sup Joong Shim: Quinoline compounds as inhibitors of angiogenesis, human methionine aminopeptidase, and sirt1, and methods of treating disorders. In: Patent EP2350012 A2, 2011, http://www.google.com/patents/EP2350012A2?cl=en [o3] 2011 Li P. - Wang F. - Lin Z.Y. - Ma, C. - Huang H.H.: Synthesis of 7-Nitro-8-quinolinol. In: Chinese Journal of Synthetic Chemistry, Vol. 19, No. 5, 2011, s. 656-658 [o1] 2013 Celik, I. - Akkurt, M. - Gezegen, H. - Kazak, C.: Acta Crystallographica Section E: Structure Reports Online, Vol. 69, No. 6, 2013, s. o956 - SCI; SCOPUS [o1] 2013 Bompart, D. - Núnez-Durán, J. - Rodríguez, D. - Kouznetsov, V.V. - Meléndez Gómez, C.M. Sojo, F. - Arvelo, F. - Visbal, G. - Alvarez, A. - García-Marchán, Y.: Bioorganic and Medicinal Chemistry, Vol. 21, No. 14, 2013, s. 4426-4431- SCI; SCOPUS [o1] 2013 Kuroda, Y. - Shindoh, N. - Takemoto, Y. - Takasu, K.: Synthesis (Germany), Vol. 45, No. 16, 2013, s. 2328-2329 - SCI; SCOPUS [o1] 2013 Fahmy, H.H. - Khalifa, N.M. - Abou El-Ella, D.A. - Ismail, M.A. - Mostafa, N.M. - Hamdy, A.A.: Life Science Journal, Vol. 10, No. 4, 2013, s. 362-368 - SCI; SCOPUS [o1] 2013 Devi, K. - Asmat, K. - Agrawal, M. - Sharma, S. - Dwivedi, J.: Journal of Chemical Sciences, Vol. 125, No. 5, 2013, s. 1093-1101 - SCI [o1] 2013 Hoda H. - Fahmy, Nagy M. - Khalifa, Dalal A. - Abou El Ella, Mohamed A. - Ismail, Noha M. Abdelhamid A. Hamdy: Life Science Journal, Vol. 10, No. 4, 2013, s. 362-368 - SCOPUS [o1] 2013 Han, J. - Li, L. - Shen, Y. - Chen, J. - Deng, H. - Shao, M. - Lu, X. - Zhang, H. - Cao, W.: European Journal of Organic Chemistry, No. 36, 2013, s. 8323-8329 - SCI; SCOPUS [o1] 2014 Lam, K.H. - Gambari, R. - Lee, K.K.H. - Chen, Y.X. - Kok, S.H.L. - Wong, R.S.M. - Lau, F.Y. Cheng, C.H. - Wong, W.Y. - Bian, Z.X. - Chan, A.S.C. - Tang, J.C.O. - Chui, C.H.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No.1, 2014, s. 367-370 - SCI; SCOPUS [o3] 2013 Li Shuan, Z.Z. - Qi, J. - Wang, T. - Zhao, H.: Study on synthesis of 8-hydroxyquinoline by doebnermiller method. In: Speciality Petrochemicals, No. 4, 2013, s. 22-24 [o1] 2014 Rahmati, A. - Eskandari-Vashareh, M.: Journal of Chemical Sciences, Vol. 126, No. 1, 2014, s. 169-176 - SCI; SCOPUS [o1] 2014 Islam, R. - Hossain, M.I. - Okamoto, Y. - Nagamatsu, T. - Anraku, K. - Okawara, T.: Heterocycles, Vol. 89, No. 3, 2014, s. 693-708 - SCOPUS [o1] 2014 Zhang, S. - Wang, Y. - Feng, C. - Yang, T. - Ji, M.ab: Dongnan Daxue Xuebao (Ziran Kexue Ban)/Journal of Southeast University (Natural Science Edition), Vol. 44, No. 1, 2014, s. 129-132 SCOPUS [o1] 2014 Peng, H.K. - Lin, I.L. - Lee, C.C. - Wang, L.Y. - Tzeng, C.C. - Chang, J.G. - Yang, S.C.: Medicinal Chemistry Research, Vol. 23, No. 3, 2014, s. 1437-1446 - SCI; SCOPUS [o3] 2014 Liu, J.O. - Shim, J.S. - Chong, C.R. - Bhat, S.: Quinoline compounds as inhibitors of angiogenesis, human methionine aminopeptidase, and SIRT1, and methods of treating disorders. United States Patent No. US 8,729,097 B2. [s.l.] : TheUnited States Patent and Trademark Office, 2014, S. 1 [o3] 2014 Desai, N.C. - Dodiya, A.M.: Microwave-Induced Synthesis of Various Quinoline Derivatives: Green Methodologies in Organic Synthesis. In: Green Chemistry: Synthesis of Bioactive Heterocycles. New Delhi : Springer, 2014, S. 163-200 [o1] 2014 Gao, Q. - Liu, S. - Wu, X. - Wu, A.: Organic Letters, Vol. 16, No. 17, 2014, s. 4582-4585 - SCI; SCOPUS [o1] 2014 Ahmed, A. - Dhara, S. - Singha, R. - Nuree, Y. - Sarkar, P.: RSC Advances, Vol. 4, No. 95, 2014, s. 53137-53141 - SCOPUS [o1] 2015 Qi, J.J. - Li, S.A. - Zhang, Z.M. - Wang, T. - Zhao, H.B. - Wang, X. - Yin, F.J.: Asian Journal of Chemistry, Vol. 27, No. 2, 2015, s. 435-440 - SCI; SCOPUS [o1] 2015 Shah, A. - Raj, D.: Journal of Saudi Chemical Society, Vol. 19, No. 1, 2015, s. 73-82 - SCI [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCOPUS [o1] 2015 Shadrikova, V.A. - Golovin, E.V. - Zatonskii, G.V. - Klimochkin, Yu.N.: Russian Journal of Organic Chemistry, Vol. 51, No. 1, 2015, s. 130-131 - SCI; SCOPUS [o3] 2015 Baluja, S.: Dissociation Constants of Some Quinoline Derivatives in Mixed Solvent mixture. In: International Letters of Chemistry, Physics and Astronomy, International Letters of Chemistry, Physics and Astronomy, Vol. 9, No. 1, 2015,s. 32-36 [o3] 2015 Alias, M. - Ismael, S. - Mousa, S.A.: Synthesis, Characterization and Theoretical Study of Some Mixed-ligand Complexes of 2-Quinoline Carboxylic Acid and 4,4/-dimethyl,2,2/-Bipyridyl with Some Transition Metal Ions. In: Journal of Al-Nahrain University, Vol. 18, No. 1, 2015, s. 28-38
12
[o1] 2014 Khalifa, N.M. - Eweas, A. - Al-Omar, M.A. - Hozzein, W.: Journal of Pure and Applied Microbiology, Vol. 8, 2014, s. 629-637 - SCI; SCOPUS [o1] 2014 Yan, X. - Yu, Y. - Ji, P. - He, H. - Qiao, C.: European Journal of Medicinal Chemistry, Vol. 102, Art. No. 8024, 2015, s. 180-187 - SCOPUS [o1] 2015 Gao, Q. - Liu, S. - Wu, X. - Zhang, J. - Wu, A.: Journal of Organic Chemistry, Vol. 80, No. 11, 2015, s. 5984-5991 - SCI; SCOPUS [o1] 2015 Chung, P.Y. - Bian, Z.X. - Pun, H.Y. - Chan, D. - Chan, A.S.C. - Chui, C.H. - Tang, J.C.O. Lam, K.H.: Future Medicinal Chemistry, Vol. 7, No. 7, 2015, s. 947-967 - SCOPUS [o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI; SCOPUS ADC12 Podeszwa, Barbara (10%) - Niedbala, Halina (10%) - Polanski, Jaroslaw (10%) - Musiol, Robert (10%) - Tabak, Dominik (5%) - Finster, Jacek (5%) - Serafin, Karol (5%) - Wietrzyk, Joanna (5%) - Boryczkka, Stanislaw (5%) - Mól, Wojciech (5%) - Jampílek, Josef [UKOEXAF] (10%) - Dohnal, Jiří (5%) Kalinowski, Danuta S. (10%) - Richardson, Des Robert (5%): Investigating the antiproliferative activity of quinoline-5,8-diones and styrylquinolinecarboxylic acids on tumor cell lines Lit. 35 zázn. In: Bioorganic & Medicinal Chemistry Letters. - Vol. 17, No. 22 (2007), s. 6138-6141 Registrované v: wos Indikátor časopisu: IF (JCR) 2007=2,604 Ohlasy (17): [o1] 2009 Li, Y.Q. - Zheng, D. - Li, J. - Han, L. - Cui, X.L. - Lang, L. - Li, M.G. - Wang, Z.Y. - Zhao, J.Y. - Huang, X.S.: Journal of Antibiotics, Vol. 62, No. 11, 2009, s. 648 - SCI [o1] 2010 Sliman, F. - Blairvacq, M. - Durieu, E. - Meijer, L. - Rodrigo, J. - Desmaele, D.: Bioorganic & Medicinal Chemistry Letters, Vol. 20, No. 9, 2010, s. 2805 - SCI [o1] 2011 Paretzki, A. - Das, H.S. - Weisser, F. - Scherer, T. - Bubrin, D. - Fiedler, J. - Nycz, J.E. - Sarkar, B.: European Journal of Inorganic Chemistry, No. 15, 2011, s. 2421 - SCI [o1] 2011 Khodairy, A. - Abass, M.: Chemistry of Heterocyclic Compounds, Vol. 47, No. 5, 2011, s. 621 SCI [o1] 2012 Li, V.M. - Gavrishova, T.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 48, No. 6, 2012, s. 828 - SCI [o1] 2012 Al-Ghamdi, A.M. - Abd El-Wahab, A.H.F. - Mohamed, H.M. - El-Agrody, A.M.: Letters in Drug Design & Discovery, Vol. 9, No. 5, 2012, s. 470 - SCI [o1] 2012 Stein, A.L. - Bilheri, F.N. - da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry-A European Journal, Vol. 18, No. 34, 2012, s. 10608 - SCI [o1] 2013 Keyari, C.M. - Kearns, A.K. - Duncan, N.S. - Eickholt, E.A. - Abbott, G. - Beall, H.D. - Diaz, P.: Journal of Medicinal Chemistry, Vol. 56, No. 10, 2013, s. 3806-3819 - SCI [o1] 2014 Keshipour, S. - Shaabani, A. - Pedarpour, M. - Sarvary, A.: Research on Chemical Intermediates, Vol. 40, No. 1, Spec. Iss., 2014, s. 156 - SCI [o1] 2014 Bassyouni, F.A. - Abu-Baker, S.M. - Mahmoud, K. - Moharam, M. - El-Nakkady, S.S. - Rehim, M.A.: RSC Advances, Vol. 4, No. 46, 2014, s. 24141 - SCI [o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: European Journal of Pharmaceutical Sciences, Vol. 51, 2014, s. 203 - SCI [o1] 2014 Gavrishova, T.N. - Li, V.M. - Karpov, O.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 50, No. 8, 2014, s. 1144 - SCI [o1] 2015 Yadav, T. - Kishore, D. - Singh, B.: British Journal of Pharmaceutical Research, Vol. 8, No. 3, 2015, Article No. 19615 - SCI [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3819 - SCI [o1] 2015 Gavrishova, T.N. - Budyka, M.F. - Potashova, N.I. - Karpov, O.N.: Russian Journal of Organic Chemistry, Vol. 51, No. 6, 2015, s. 873 - SCI [o1] 2015 Kumar, N.S. - Rao, L.C. - JagadeeshBabu, N. - Kumar, V.D. - Murthy, U.S.N. - Meshram, H.M.: Synlett, Vol. 26, No. 13, 2015, s. 1814 - SCI [o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI ADC13 Vinšová, Jarmila (20%) - Imramovský, Aleš (20%) - Buchta, Vladimír (10%) - Čečková, Martina (10%) - Doležal, Martin (10%) - Štaud, František (10%) - Jampílek, Josef [UKOEXAF] (10%) - Kaustová, Jarmila (10%): Salicylanilide acetates: synthesis and antibacterial evaluation Lit. 14 zázn. In: Molecules. - Vol. 12, No. 1 (2007), s. 1-12
13
Registrované v: wos Indikátor časopisu: IF (JCR) 2007=0,940 Ohlasy (6): [o1] 2008 Pyka, A.: Journal of Liquid Chromatography & Related Technologies, Vol. 31, No. 13, 2008, s. 1958 - SCI [o1] 2009 Skala, P. - Machacek, M. - Vejsova, M. - Kubicova, L. - Kunes, J. - Waisser, K.: Journal of Heterocyclic Chemistry, Vol. 46, No. 5 , 2009, s. 880 - SCI [o1] 2013 Kang, S. - Min, H.J. - Kang, M.S. - Jung, M.G. - Kim, S.: Bioorganic & Medicinal Chemistry Letters, Vol. 23, No. 6, 2013, s. 1751 - SCI [o1] 2013 Nuta, D.C. - Chifiriuc, M.C. - Draghici, C. - Limban, C. - Missir, A.V. - Morusciag, L.: Farmacia, Vol. 61, No. 5, 2013, s. 974 - SCI [o1] 2015 Dank, C. - Kirchknopf, B. - Mastalir, M. - Kahlig, H. - Felsinger, S. - Roller, A. - Arion, V.B. Gstach, H.: Molecules, Vol. 20, No. 1, 2015, s. 1711 - SCI [o1] 2015 Diller, D.J. - Connell, N.D. - Welsh, W.J.: Journal of Computer-Aided Molecular Design, Vol. 29, No. 11, 2015, s. 1024 - SCI ADC14 Doležal, Martin (20%) - Čmedlová, Pavlína (15%) - Pálek, Lukáš (15%) - Vinšová, Jarmila (5%) Kuneš, Jiří (5%) - Buchta, Vladimír (10%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek, Josef [UKOEXAF] (15%): Synthesis and antimycobacterialevaluation of substituted pyrazinecarboxamides Lit.: 27 zázn., 1 obr., 3 tab. In: European Journal of Medicinal Chemistry. - Vol. 43, No. 5 (2008), s. 1105-1113 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=2,882 Ohlasy (31): [o3] 2008 Haruaki, T.: Expert Opinion on Drug Discovery, Vol. 3, No. 1, 2008, s. 21-49 [o3] 2009 Hopper, D.W. - Clemens, J.J. - Kwon, S.: Chapter 6.1 Six-membered ring systems: pyridine and benzo derivatives. In: Progress in Heterocyclic Chemistry, Volume 21. Amsterdam : Elsevier, 2009, S. 330-414 [o1] 2009 Manlove, A. - Groziak, M.P.: Progress in Heterocyclic Chemistry, Vol. 21, 2009, s. 375-414 SCOPUS [o1] 2010 Dunklevy, J.D. - Soole, K.L. - Perkins, M.V. - Dennis, E.G. - Keyzers, R.A. - Kalua, C.M. Boss, P.K.: Plant Molecular Biology, Vol. 74, No. 1-2, 2010, s. 77-89 - SCI [o1] 2010 Abdel-Aziz, M. - Abdel-Rahman, H.M.: European Journal of Medicinal Chemistry, Vol. 45, No. 8, 2010, s. 3384-3388 - SCI [o1] 2010 Yesilel, O.Z. - Mutlu, A. - Darcan, C. - Buyukgungor, O.: Journal of Molecular Structure, Vol. 964, No. 1-3, 2010, s. 39-46 - SCOPUS [o1] 2010 Chauhan, P.M.S. - Sunduru, N. - Sharma, M.: Future Medicinal Chemistry, Vol. 2, No. 9, 2010, s. 1469-1500 - SCOPUS [o1] 2010 Lee, J.H. - Myung, P.K. - Kim, S.J. - Sung, N.D.: Journal of Applied Biological Chemistry, Vol. 53, No. 4, 2010, s. 440-445 - SCOPUS [o3] 2010 Yafei, L.I. - Liqun, J.I.N. - Zhiqiang, L.I.U. - Yuguo, Z.: Chinese Journal of Modern Applied Pharmacy, Vol. 27, No. 4, 2010, s. 307-312 [o3] 2010 Tewatia, N. - Namdeo, K.P. - Jain, S.K. - Prajapati, S.K. - Singh, O. - Jain, V. - Kumar, P.: Journal of the Institution of Chemists (India), Vol. 82, No. 5, 2010, s. 148-153 [o3] 2011 Lima, C.H.S. - Bispo, M.L.F. - de Souza, M.V.N.: Pirazinamida: Um Fármaco Essencial no Tratamento da Tuberculose. In: Revista Virtual de Química, Vol. 3, No. 3, 2011, s. 159-180 [o3] 2011 Prasad, R. - Sharma, R.: 2D QSAR Analysis of Pyrazinecarboxamides derivatives as an herbicidal agent. In: Journal of Computational Methods in Molecular Design, Vol. 1, No. 1, 2011, s. 7-13 [o1] 2011 Dib-Bellahouel, S. - Fortas, Z.: African Journal of Biotechnology, Vol. 10, No. 47, 2011, s. 9694-9699 - SCOPUS [o3] 2011 Vikramjeet J. - Balasubramanian N. - Munish A.: A Review of Biological potential of Pyrazinamide derivatives. In: Hygeia : Journal for Drugs and Medicines, Vol. 4, Iss. 1, 2012, s. 1-6 [o3] 2012 Ghetiya: Pyrazine derivatives. In: Studies on heterocyclic compounds, Pp. 17, 2012, http://ir.inflibnet.ac.in:8080/bitstream/10603/3890/7/07_part%20a.pdf [o1] 2012 Bispo, M.D.L.F. - Gonçalves, R.S.B. - Lima, C.H.D.S. - Cardoso, L.N.D.F. - Lourenço, M.C.S. - De Souza, M.V.N.: Journal of Heterocyclic Chemistry , Vol. 49, Iss. 6, 2012, s. 1317-1322 - SCOPUS [o3] 2010 Li, Y. - Kinley L.J.L. - Liu Z. - Yu-Guo Z.: Pyrazinamide research progress. In: Chinese Journal of Modern Applied Pharmacy, Vol. 27, Iss. 4, 2010, s. 307-312
14
[o1] 2013 Nayak, P.S. - Narayana, B. - Samshuddin, S. - Sarojini, B.K.: MolBank, Vol. 2013, Iss. 2, 2013, Nestr. - SCOPUS [o3] 2012 Asif, M.: Recent Efforts for the Development of Antitubercular Drug Containing Diazine Ring. In: Medicinal Chemistry, Vol. 2, Iss. 7, 2012, s. 151-167 [o3] 2013 Blochin I.V. - Ageev, A.V. - Artošenko J.M. - Chlytin, N.V. - Tormozov, V.A.: Sintez 2metoksi-3-T-pirazinov v ionnoj židkosti. In: Izvestja Tulskogo Gosudarstvennoho Universiteta, Jestestvennye Nauki, 2013, s. 163 [o1] 2013 Achelle, S. - Baudequin, C. - Plé, N.: Dyes and Pigments, Vol. 98, No. 3, 2013, s. 575-600 - SCI ; SCOPUS [o1] 2013 Miniyar, P.B. - Murumkar, P.R. - Patil, P.S. - Barmade, M.A. - Bothara, K.G.: Reviews in Medicinal Chemistry, Vol. 13, No. 11, 2013, s. 1607-1625 - SCI [o1] 2014 Ma, W.J. - Gao, Z.Y. - Zhu, S. - Wu, B.L.: Polyhedron, Vol. 73, May 2014, s. 59-66 - SCOPUS [o1] 2013 Darcan, C. - Kaygusuz, Ö. - Korkmaz, T.: Journal of Pure and Applied Microbiology, Vol. 7, No. 4, 2013, s. 2747-2756 - SCOPUS [o1] 2014 Konar, S. - Saha, U. - Dolai, M. - Chatterjee, S.: Journal of Molecular Structure, Vol. 1075, 2014, s. 286-291 - SCOPUS [o1] 2015 Verbitskiy, E.V. - Slepukhin, P.A. - Kravchenko, M.A. - Skornyakov, S.N. - Evstigneeva, N.P. Kungurov, N.V. - Zil'Berberg, N.V. - Rusinov, G.L. - Chupakhin, O.N. - Charushin, V.N.: Bioorganic and Medicinal Chemistry Letters, Vol.25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS [o1] 2015 Benzon, K.B. - Varghese, H.T. - Panicker, C.Y. - Pradhan, K. - Tiwary, B.K. - Nanda, A.K. Alsenoy, C.V.: Spectrochimica Acta - Part A: Molecular and Biomolecular Spectroscopy, Vol. 151, July, 2015, s. 965-979 - SCOPUS [o3] 2015 Mohammad Asif: Anti-tubercular activity of some six membered heterocycle compounds. In: Chemistry International, Vol. 1, No. 3, 2015, s. 134-163 [o3] 2015 Elidrissi, B. - Ousaa, A. - Ghamali, M. - Chtita,S. - Ajana, M.A. - Bouachrine - Lakhlifi, T.: The biological activity of pyrazinecarboxamides derivatives as an herbicidal agent: combining DFT and QSAR studies. In: Journal of Computational Methods in Molecular Design, Vol. 5, No. 2, 2015, s. 83-91 [o3] 2015 Shaikh, A.R. - Gonsalves, S.I. - Nikam, A. - Kshirsagar, S.J. - Thombare, Y.: Predicting Pyrazinecarboxamides Derivatives as an Herbicidal Agent: 3d Qsar by kNN-MFA and Multiple linear regression Approach. In: World Applied Sciences Journal, Vol. 33, No. 6, 2015, s. 980-989 [o1] 2016 Chylewska, A. - Sikorski, A. - Ogryzek, M. - Makowski, M.: Journal of Molecular Structure, Vol. 1105, 2016, s. 104 - SCI; SCOPUS ADC15 Jampílek, Josef [UKOEXAF] (50%) - Brojerová, Eliška (25%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Jun, Daniel (5%): Preparation and antiplatelet activity of glycidic acid derivatives Lit. 30 zázn. In: Chemical papers. - Vol. 62, No. 3 (2008), s. 281-287 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=0,758 ADC16 Jampílek, Josef [UKOEXAF] (25%) - Rečková, Zuzana (20%) - Imramovský, Aleš (20%) - Raich, Ivan (20%) - Vinšová, Jarmila (10%) - Dohnal, Jiří (5%): Study of stability of new mutual prodrugs with antimycobacterial activity Lit. 45 zázn. In: Current Organic Chemistry. - Vol. 12, No. 8 (2008), s. 667-674 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=3,184 ADC17 Musilek, Kamil (30%) - Jampílek, Josef [UKOEXAF] (30%) - Dohnal, Jiří (5%) - Jun, Daniel (10%) Gunn-Moore, Frank (5%) - Doležal, Martin (5%) - Kuča, Kamil (15%): RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker Lit. 39 zázn. In: Analytical and Bioanalytical Chemistry. - Vol. 391, No. 1 (2008), s. 367-372 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=3,328 ADC18 Musiol, Robert (20%) - Tabak, Dominik (10%) - Niedbala, Halina (5%) - Podeszwa, Barbara (5%) Kráľová, Katarína [UKOPRCUS] (15%) - Dohnal, Jiří (5%) - Finster, Jacek (10%) - Mencel, Agnieszka (5%) - Polanski, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (15%): Investigating biological activity
15
spectrum for novel quinoline analogues 2: Hydroxyquinolinecarboxamides with photosynthesis-inhibiting activity Lit.: 44 zázn., 4 obr., 2 tab., 1 schéma In: Bioorganic & Medicinal Chemistry. - Vol. 16, No. 8 (2008), s. 4490-4499 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=3,075 Ohlasy (20): [o1] 2009 Qui, C.M. - Zheng, Q.W. - Hua, R.M.: Tetrahedron, Vol. 65, No. 7, 2009, s. 1316-1320 SCOPUS; SCI [o1] 2010 Achrem-Achremowicz, J. - Kepczynska, E. - Zylewski, M. - Janeczko, Z.: Biomedical Chromatography, Vol. 24, No. 3, 2010, s. 261-267 - SCI [o1] 2010 Rahimizadeh, M. - Pordel, M. - Bakavoli, M. - Eshghi, H.: Dyes and Pigments, Vol. 86, No. 3, 2010, s. 266-270 - SCI [o1] 2011 Khodairy, A. - Abass, M.: Khimiya Geterotsiklicheskikh Soedinenii, No. 5, 2011, s. 736-749 SCOPUS [o3] 2011 Pan, S.M.: The Synthesis and Characterization of Quinoline-Metallic Complexes and Study Material for Military Sensor. [S.l.] : National Defense University, 2011, S. 150 [o3] 2011 Gagliardi, S. - Del Sordo, S. - Mailland, F. - Legora, M.A.: Secondary 8 hydroxyquinoline 7 carboxamide derivatives for use as antifungal agents. Patent WO 2011080265, S. 51 [o1] 2011 Khodairy, A. - Abass, M.: Chemistry of Heterocyclic Compounds, Vol. 47, No. 5, 2011, s. 611621 - SCI [o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied Photosynthesis. Rijeka : InTech, 2012, S. 1-22 [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o1] 2013 Nycz J.E. - Malecki G.J.: Journal of Molecular Structure, Vol. 1032, 2013, s. 159-168 SCOPUS [o1] 2013 El-Agrody, A.M. - Abd-Rabboh, H.S.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research, Vol. 22, No. 3, 2013, s. 1339-1355 - SCI; SCOPUS [o3] 2013 Shet Prakash, M. - Vaidya, V. P. - Mahadevan, K.M. - Shivananda, M.K. - Suchetan, P.A. Sunitha, M.: Synthesis characterization and antimicrobial activities of some novel carboxamides derived from napthofurans and 1,2,4-triazoles.In: National Conference on Challenges and Opportunities of Chemical Sciences in 21st Century. [S.l.] : [s.n.], 2013, Nestr. [o1] 2014 Lam, K.H. - Gambari, R. - Lee, K.K.H. - Chen, Y.X. - Kok, S.H.L. - Wong, R.S.M. - Lau, F.Y. Cheng, C.H. - Wong, W.Y. - Bian, Z.X., Chan, A.S.C. - Tang, J.C.O. - Chui, C.H.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No.1, 2014, s. 367-370 - SCI; SCOPUS [o1] 2014 El-Agrody, A.M. - Afifi, T.H.: Heterocycles, Vol. 89, No. 7, 2014, s. 1557-1584 - SCOPUS [o1] 2014 Ariyasu, S. - Mizuseda, Y. - Hanaya, K. - Aoki, S.: Chemical and Pharmaceutical Bulletin, Vol. 62, No. 7, 2014, s. 642-648 - SCI; SCOPUS [o1] 2014 Khalifa, N.M. - Eweas, A. - Al-Omar, M.A. - Hozzein, W.: Journal of Pure and Applied Microbiology, Vol. 8, 2014, s. 629-637 - SCOPUS [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCOPUS [o1] 2015 Chung, P.Y. - Bian, Z.X. - Pun, H.Y. - Chan, D. - Chan, A.S.C. - Chui, C.H. - Tang, J.C.O. Lam, K.H.: Future Medicinal Chemistry, Vol. 7, No. 7, 2015, s. 947-967 - SCOPUS [o1] 2015 Fang, F.Q. - Guo, H.S. - Zhang, J. - Ban, L.Y. - Liu, J.W. - Yu, P.Y.: Molecular Medicine Reports, Vol. 12, No. 6, 2015, s. 8070 - SCI; SCOPUS ADC19 Opletalová, Veronika (20%) - Kalinowski, Danuta S. (15%) - Vejsová, Marcela (15%) - Kuneš, Jiří (10%) - Pour, Milan (10%) - Jampílek, Josef [UKOEXAF] (10%) - Buchta, Vladimír (10%) - Richardson, Rhonda (10%): Identification and characterization of thiosemicarbazones with antifungal and antitumor effects: cellular iron chelation mediating cytotoxic activity Lit. 58 zázn. In: Chemical Resarch in Toxicology. - Vol. 21, No. 9 (2008), s. 1878-1889 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=3,491
16
ADC20 Palek, Lukáš (25%) - Dvořák, Jaroslav (15%) - Svobodová, Michaela (15%) - Buchta, Vladimír (15%) Jampílek, Josef [UKOEXAF] (15%) - Doležal, Martin (15%): Synthesis, antimycobacterial and antifungal evaluation of3-arylaminopyrazine-2,5-dicarbonitriles Lit. 16 zázn. In: Archiv der Pharmazie. - Vol. 341, No. 1 (2008), s. 61-65 Registrované v: wos Indikátor časopisu: IF (JCR) 2008=1,429 Ohlasy (3): [o1] 2009 Ukrainets, I.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Chemistry of Heterocyclic Compounds, Vol. 45, No. 9, 2009, s. 1068 - SCI [o1] 2010 Walkiewcz, R. - Chazan, R. - Grubek-Jaworska, H.: Biocybernetics and Biomedical Engineering, Vol. 30, No. 2, 2010, s. 14 - SCI [o1] 2010 Abdel-Aziz, M. - Abdel-Rahman, H.M.: European Journal of Medicinal Chemistry, Vol. 45, No. 8, 2010, s. 3388 - SCI ADC21 Brychtová, Kateřina (25%) - Slabá, Barbora (10%) - Plaček, Lukáš (15%) - Jampílek, Josef [UKOEXAF] (20%) - Raich, Ivan (25%) - Csöllei, Jozef (5%): Coupling reactions of alphabromocarboxylate with non-aromatic N-heterocycles Lit. 25 zázn. In: Molecules. - Vol. 14, No. 8 (2009), s. 3019-3029 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=1,738 ADC22 Doležel, Jan (20%) - Hiršová, Petra (15%) - Opletalová, Veronika (20%) - Dohnal, Jiří (5%) - Vejsová, Marcela (10%) - Kuneš, Jiří (10%) - Jampílek, Josef [UKOEXAF] (20%): Rhodanineacetic Acid Derivatives as Potential Drugs: Preparation, Hydrophobic Properties and Antifungal Activity of (5Arylalkylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)acetic Acids Lit. 63 zázn. In: Molecules. - Vol. 14, No. 10 (2009), s. 4197-4212 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=1,738 ADC23 Imramovský, Aleš (20%) - Vinšová, Jarmila (20%) - Ferriz, Juana Monreal (10%) - Doležal, Rafael (10%) - Jampílek, Josef [UKOEXAF] (20%) - Kaustová, Jarmila (10%) - Kunc, Filip (10%): New antituberculotics originated from salicylanilides with promising in vitro activity against atypical mycobacterial strains Lit. 25 zázn. In: Bioorganic & Medicinal Chemistry Letters. - Vol. 17, No. 10 (2009), s. 3572-3579 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=2,822 ADC24 Imramovský, Aleš (20%) - Vinšová, Jarmila (20%) - Ferriz, Juana Monreal (20%) - Buchta, Vladimír (20%) - Jampílek, Josef [UKOEXAF] (20%): Salicylanilide esters of N-protected amino acids as novel antimicrobial agents Lit. 19 zázn. In: Bioorganic & Medicinal Chemistry Letters. - Vol. 17, No. 2 (2009), s. 348-351 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=2,650 ADC25 Jampílek, Josef [UKOEXAF] (15%) - Musiol, Robert (15%) - Finster, Jacek (5%) - Peško, Matúš [UKOPREEF] (10%) - Carroll, James (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Vejsová, Marcela (10%) - O Mahony, Jim (5%) - Coffey, Aidan (5%) - Dohnal, Jiří (5%) - Polanski, Jaroslaw (10%): Investigating Biological Activity Spectrum for Novel Styrylquinazoline Analogues Lit.: 70 zázn., 1 obr., 2 tab. In: Molecules. - Vol. 14, No. 10 (2009), s. 4246-4265 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=1,738
17
Ohlasy (18): [o3] 2011 Vijaychand, A. - Manjula, S.N. - Barath, E.N. - Divya, B.: Medicinal and biological significance of quinazoline a highly important scaffold for drug discovery: a review. In: International Journal of Pharma and Bio Sciences, Vol. 2, No. 1, 2011, s. 780-809 [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS [o1] 2012 Stein, A.L. - Bilheri, F.N. - Da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry - A European Journal, Vo. 18, No. 34, 2012, s. 10602-10608 - SCI ; SCOPUS [o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied Photosynthesis. Rijeka : InTech, 2012, S. 1-22 [o1] 2012 Wang, Y.K. - Jin, J. - Zhu, L.N. - Zhang, Y. - Chen, X.G. - Gao, X.Q. - Xu, B.L.: Yaoxue Xuebao, Vol. 47, No. 9, 2012, s. 1164-1178 - SCOPUS [o3] 2012 Samira, I. - Patel, S. - Hasmin, M. - Patel, S.: Biological Profile of Quinazoline. In: International Journal of Pharmaceutical and Chemical Sciences, Vol. 1, No. 4, 2012, s. 1527 [o3] 2012 Wangy, Y.K. - Jin, J. - Zhu, L.N. - Zhang, Y. - Chen, X.G. - Gao, X.Q. - Xu, B.L.: Synthesis and antitumor activity of novel 2-(1-substituted-piperidin -4-ylamino)quinazolines as antitumor agents. In: Acta Pharmaceutica Sinica, Vol.47, No. 9, 2012, s. 1178 [o1] 2013 Li, Y. - De Kock, C. - Smith, P.J. - Guzgay, H. - Hendricks, D.T. - Naran, K. - Mizrahi, V. Warner D.F. - Chibale, K. - Smith, G.S.: Organometallics, Vol. 32, No. 1, 2013, s. 141-150 - SCI ; SCOPUS [o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: Journal of Pharmaceutical Sciences, Vol. 51, No. 1, 2014, s. 196-203 - SCI ; SCOPUS [o3] 2014 Indubhushan - Choudhary, A.N. - Kothiyal, P.: Synthesis and evaluation of quinazolinthione derivatives as antibacterial agents. In: International Journal of Pharmacy, Vol. 4, No. 3, 2014, s. 135 [o1] 2014 Lakshmi, K. - Rama Rao, N. - Basaveswararao, M.V.: Rasayan Journal of Chemistry, Vol. 7, No. 1, 2014, s. 44-54 - SCOPUS [o1] 2014 Aly, S.A. - Alganzory, H.H. - Salem, T.A.: Journal of Chemical and Pharmaceutical Research, Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCI ; SCOPUS [o1] 2015 Kumar, D. - Jadhavar, P.S. - Nautiyal, M. - Sharma, H. - Meena, P.K. - Adane, L. - Pancholia, S. - Chakraborti, A.K.: RSC Advances, Vol. 5, No. 39, 2015, s. 30819-30825 - SCOPUS [o1] 2015 Lakshmi, K. - Rama Rao, N. - Basaveswara Rao, M.V.: Journal of Environmental Biology, Vol. 36, No. 4, 2015, s. 909-918 - SCI ; SCOPUS [o3] 2015 Wani, Z.A. - Pathania, A.S. - Mahajan, G. - Behl, A. - Mintoo, M.J. - Guru, S.K. - Viswanath, V. - Malik, F. - Kamal, A. - Mondhe, D.M.: Anticancer activity of a novel quinazolinone-chalcone derivative through cell cycle arrest inpancreatic cancer cell line. In: Journal of Solid Tumors, Vol. 5, No. 2, 2015, s. 84 [o3] 2014 Krastina, G. - Ravina, I. - Mierina, I. - Zicane, D. - Turks, M. - Tetere, Z. - Leonciks, A.: Synthesis of novel quinazolinone-1,2,3-triazole conjugates. In: Journal of Chemical and Pharmaceutical Research, Vol. 6, No. 12, 2014, s.13 ADC26 Jampílek, Josef [UKOEXAF] (10%) - Musiol, Robert (10%) - Peško, Matúš [UKOPREEF] (10%) Kráľová, Katarína [UKOPRCUS] (10%) - Vejsová, Marcela (10%) - Carroll, James (10%) - Coffey, Aidan (5%) - Finster, Jacek (5%) - Tabak, Dominik (5%) - Niedbala,Halina (5%) - Kozik, Violetta (5%) Polanski, Jaroslaw (5%) - Csöllei, Jozef (5%) - Dohnal, Jiří (5%): Ring-substituted 4-Hydroxy-1Hquinolin-2-ones: Preparation and Biological Activity Lit.: 39 zázn., 2 obr., 2 tab. In: Molecules. - Vol. 14, No. 3 (2009), s. 1145-1159 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=1,738 Ohlasy (16): [o3] 2010 Ibrahim, M.A. - Hassanin, H.M. - Gabr, Y.A.A. - Alnamer, Y.A.S.: European Journal of Chemistry, Vol. 1, No. 3, 2010, s. 195-199 [o1] 2011 Ukrainets, I.V. - Golik, N.Y.U. - Bevz, O.V. - Gorokhova, O.V.: Khimiya Geterotsiklicheskikh Soedinenii, No. 7, 2011, s. 1018-1023 - SCOPUS [o1] 2011 Ukrainets, I. V. - Golik, N. Y. - Bevz, O. V. - Gorokhova, O. V.: Chemistry of Heterocyclic Compounds, Vol. 47, No. 2, 2011, s. 833-837 - SCI
18
[o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o3] 2012 Teixeira R.R. - Pereira J.L. - Pereira W.L: Photosynthetic inhibitors. In: Applied Photosynthesis. Rijeka : Intech, 2012, S. 1-22 [o1] 2012 Abass, M. - Mohamed, E.H.A. - Mayas, A.S. - Ibrahim, A.H.: Journal of Chemical Sciences, Vol. 124, No. 5, 2012, s. 1033-1041 - SCI [o1] 2013 El-Agrody, A.M. - Abd-Rabboh, H.S.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research, Vol. 22, No. 3, 2013, s. 1339-1355 - SCI ; SCOPUS [o1] 2014 Bhat, S.I. - Trivedi, D.R.: RSC Advances, Vol. 4, No. 22, 2014, s. 11300-11304 - SCI ; SCOPUS [o1] 2014 El-Agrody, A.M. - Afifi, T.H.: Heterocycles, Vol. 89, No. 7, 2014, s. 1557-1584 - SCOPUS [o1] 2014 Prajapati, S.M. - Patel, K.D. - Vekariya, R.H. - Panchal, S.N. - Patel, H.D.: RSC Advances, Vol. 4, No. 47, 2014, s. 24463-24476 - SCI ; SCOPUS [o1] 2014 Aly, S.A. - Alganzory, H.H. - Salem, T.A.: Journal of Chemical and Pharmaceutical Research, Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS [o1] 2014 Khalifa, N.M. - Eweas, A. - Al-Omar, M.A. - Hozzein, W.: Journal of Pure and Applied Microbiology, Vol. 8, No. 1, 2014, s. 629-637 - SCOPUS [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCOPUS [o3] 2015 Ruat, M. - Faure, H. - Gorojankina, T.: Use of quinolinone derivatives as a research tool. US Patent US8957091, http://www.google.com/patents/US8957091 [o1] 2015 Fang, F.Q. - Guo, H.S. - Zhang, J. - Ban, L.Y. - Liu, J.W. - Yu, P.Y.: Molecular Medicine Reports, Vol. 12, No. 6, 2015, s. 8070 - SCI; SCOPUS ADC27 Opatřilová, Radka (5%) - Jampílek, Josef [UKOEXAF] (20%) - Raich, Ivan (20%) - Kačerová, Sandra (15%) - Pekárek, Tomáš (15%) - Dohnal, Jiří (5%) - Csöllei, Jozef (5%) - Havlíček, Jaroslav (15%): Synthesis, Characterization and Physico-chemical Properties of New 2-(4-Arylpiperazine-1-yl)-1-(3methylbenzofuran-2-yl)ethanoles as Potential Antihypertensive Agents Lit. 24 zázn. In: Current Organic Chemistry. - Vol. 13, No. 10 (2009), s. 965-975 Registrované v: wos Indikátor časopisu: IF (JCR) 2009=2,879 ADC28 Brychtová, Kateřina (20%) - Opatřilová, Radka (5%) - Raich, Ivan (10%) - Kalinowski, Danuta S. (10%) - Dvořáková, Lenka (10%) - Plaček, Lukáš (10%) - Csöllei, Jozef (5%) - Richardson, Des R. (10%) - Jampílek, Josef [UKOEXAF] (20%): Investigating the activity of 2-substituted alkyl-6-(2,5dioxopyrrolidin-1-yl)hexanoates as skin penetration enhancers Lit. 44 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 18, No. 24 (2010), s. 8556-8565 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=2,978 ADC29 Brychtová, Kateřina (35%) - Jampílek, Josef [UKOEXAF] (20%) - Opatřilová, Radka (10%) - Raich, Ivan (20%) - Farsa, Oldřich (10%) - Csöllei, Jozef (5%): Synthesis, physico-chemical properties and penetration activity ofalkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1-yl)hexanoates as potential transdermal penetration enhancers Lit. 47 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 18, No. 1 (2010), s. 73-79 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=2,978 ADC30 Doležal, Martin (20%) - Zitko, Jan (15%) - Osička, Zdeněk (10%) - Kuneš, Jiří (5%) - Vejsová, Marcela (10%) - Buchta, Vladimír (5%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek, Josef [UKOEXAF] (15%): Synthesis,Antimycobacterial, Antifungal and Photosynthesis-Inhibiting Activity of Chlorinated N-phenylpyrazine-2-carboxamides Lit.: 28 zázn., 2 obr., 2 tab., 1 schéma In: Molecules. - Vol. 15, No. 12 (2010), s. 8567-8581
19
Registrované v: wos Indikátor časopisu: IF (JCR) 2010=1,988 Ohlasy (8): [o3] 2012 Tewatia, N. - Abida - Namdeo, K. P.: Synthesis and antimicrobial activity of pyrazine carboxamide derivatives. In: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 3, 2012, s.1794-1798 [o1] 2012 Bentabed-Ababsa G. - Hamza-Reguig S. - Derdour A. - Domingo L.R. - Sáez J.A. - Roisnel T. Dorcet V. - Nassar E. - Mongin F.: Organic & Biomoecular Cheistry, Vol. 10, No. 42, 2012, s. 8434-8444 - SCI [o1] 2013 Chan, J.G.Y. - Chan, H.-K. - Prestidge, C.A. - Denman, J.A.b , Young, P.M. - Traini, D.: European Journal of Pharmaceutics and Biopharmaceutics, Vol. 83, No. 2, 2013, s. 285-292 - SCI ; SCOPUS [o3] 2014 Parimala Vaijayanthi, S. - Mathiyalagan, N.: Antibacterial, antifungal, anti-oxidant, antiinflammatory and anti-hypertensive activities of N-chloropyrazinamide. In: International Letters of Chemistry, Physics and Astronomy, Vol. 7, 2014, s. 1-8 [o1] 2014 Nayak, P.S. - Narayana, B. - Anthal, S. - Gupta, V.K. - Kant, R.: Molecular Crystals and Liquid Crystals, Vol. 592, No. 1, 2014, s. 199-208 - SCI ; SCOPUS [o1] 2015 Verbitskiy, E.V. - Slepukhin, P.A. - Kravchenko, M.A. - Skornyakov, S.N. - Evstigneeva, N.P. Kungurov, N.V. - Zil'Berberg, N.V. - Rusinov, G.L. - Chupakhin, O.N. - Charushin, V.N.: Bioorganic and Medicinal Chemistry Letters, Vol.25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS [o1] 2016 Chylewska, A. - Sikorski, A. - Ogryzek, M. - Makowski, M.: Journal of Molecular Structure, Vol. 1105, 2016, s. 104 - SCI; SCOPUS [o1] 2015 Apostolov, S. - Vastag, G. - Matijevic, B. - Petrovic, S.: Journal of Liquid Chromatography and Related Technologies, Vol. 38, No. 18, 2015, s. 1698 - SCI; SCOPUS ADC31 Mrozek-Wilczkiewicz, Anna (10%) - Kalinowski, Danuta S. (10%) - Musiol, Robert (10%) - Finster, Jacek (5%) - Szurko, Agnieszka (10%) - Serafin, Katarzyna (5%) - Knas, Magdalena (5%) Kamalapuram, Sishir K. (5%) - Kovacevic, Zaklina (10%) - Jampílek, Josef [UKOEXAF] (10%) Ratuszna, Alicja (5%) - Rzeszowska-Wolny, Joanna (5%) - Richardson, Des R. (5%) - Polanski, Jaroslaw (5%): Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones Lit. 25 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 18, No. 7 (2010), s. 2664-2671 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=2,978 ADC32 Musiol, Robert (15%) - Jampílek, Josef [UKOEXAF] (15%) - Nycz, Jacek E. (5%) - Peško, Matúš [UKOPREEF] (10%) - Carroll, James (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Vejsova, Marcela (10%) - O Mahony, Jim (5%) - Coffey, Aidan (5%) - Mrozek,Anna (5%) - Polanski, Jaroslaw (10%): Investigating the Activity Spectrum for Ring-Substituted 8-Hydroxyquinolines Lit.: 48 zázn., 3 tab. In: Molecules. - Vol. 15, No. 1 (2010), s. 288-304 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=1,988 Ohlasy (15): [o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied Photosynthesis. Rijeka : InTech, 2012, S. 1-22 [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS [o1] 2012 Stein, A.L. - Bilheri, F.N. - Da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry - A European Journal, Vol. 18, No. 34, 2012, s. 10602-10608 - SCOPUS [o3] 2012 Panda, B.K.: Synthesis, characterization and photophysical properties of quinolin-8-olato chelated osmium(II) organometallics bearing a pendant imine-phenol motif and electrogeneration of trivalent analogue. In: Open Journal ofInorganic Chemistry, Vol. 2, No. 3, 2012, s. 49-57 [o1] 2013 Li, Y. - De Kock, C. - Smith, P.J. - Guzgay, H. - Hendricks, D.T. - Naran, K. - Mizrahi, V. Warner D.F. - Chibale, K. - Smith, G.S.: Organometallics, Vol. 32, No. 1, 2013, s. 141-150 - SCI
20
[o1] 2013 Novakova, J. - Vlkova, E. - Bonusova, B. - Rada, V. - Kokoska, L.: Anaerobe, Vol. 22, 2013, s. 134-136 - SCI ; SCOPUS [o1] 2013 Vandekerckhove, S. - Tran, H.G. - Desmet, T. - D'Hooghe, M.: Bioorganic and Medicinal Chemistry Letters, Vol. 23, No. 16, 2013, s. 4641-4643 - SCI ; SCOPUS [o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: Journal of Pharmaceutical Sciences, Vol. 51, No. 1, 2014, s. 196-203 - SCI ; SCOPUS [o3] 2012 Kaiss, R.I. - Noor, F.A.-A.: Synthesis and study some mixed ligands complexes from folic acid with 1,10-phenanthroline and 8-hydroxyquinoline. In: Journal of University of Anbar for Pure Science, Vol. 6, No. 3, 2012, s. 67-74 [o1] 2014 Muscia, G.C. - Hautmann, S. - Buldain, G.Y. - Asís, S.E. - Gütschow, M.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No. 6, 2014, s. 1545-1549 - SCI [o1] 2014 De O Freitas, L.B. - Borgati, T.F. - De Freitas, R.P. - Ruiz, A.L.T.G. - Marchetti, G.M. - De Carvalho, J.E. - Da Cunha, E.F.F. - Ramalho, T.C. - Alves, R.B: European Journal of Medicinal Chemistry, Vol. 84, September, 2014, s. 595-604 - SCI ; SCOPUS [o1] 2014 Ariyasu, S. - Mizuseda, Y. - Hanaya, K. - Aoki, S.: Chemical and Pharmaceutical Bulletin, Vol. 62, No. 7, 2014, s. 642-648 - SCOPUS [o1] 2014 Aly, S.A. - Alganzory, H.H. - Salem, T.A.: Journal of Chemical and Pharmaceutical Research, Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS [o3] 2015 Siddiqi, H. - Faizi, S. - Naz, S. - Zahir, E.: Synthesis of Mannich Bases of 8-Hydroxyquinoline. In: Journal of Basic and Applied Sciences, Vol. 11, 2015, s. 539-543 ADC33 Oktábec, Zbyněk (15%) - Kos, Jiří (10%) - Mandelová, Zuzana (10%) - Havelková, Lenka (5%) Pekárek, Tomáš (10%) - Řezáčová, Anna (10%) - Plaček, Lukáš (10%) - Tkadlecová, Marcela (5%) Havlíček, Jaroslav (5%) - Dohnal, Jiří (5%) - Jampílek, Josef [UKOEXAF] (15%): Preparation and properties of new Co-crystals of ibandronate with gluco- or galactopyranoside derivatives Lit. 25 zázn. In: Molecules. - Vol. 15, No. 12 (2010), s. 8973-8987 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=1,988 ADC34 Otevřel, Jan (10%) - Mandelová, Zuzana (5%) - Peško, Matúš [UKOPREEF] (10%) - Guo, Jiahui (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Šeršeň, František [UKOPRCUS] (10%) - Vejsová, Marcela (5%) - Kalinowski, Danuta S. (5%) - Kovacevic, Zaklina (5%)- Coffey, Aidan (5%) - Csöllei, Jozef (10%) - Richardson, Des R. (5%) - Jampílek, Josef [UKOEXAF] (10%): Investigating the Spectrum of Biological Activity of Ring-Substituted Salicylanilides and Carbamoylphenylcarbamates Lit.: 62 zázn., 2 obr., 2 tab. In: Molecules. - Vol. 15, No. 11 (2010), s. 8122-8142 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=1,988 Ohlasy (4): [o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied Photosynthesis. Rijeka : InTech, 2012, S. 1-22 [o1] 2012 Krátky, M. - Vinšová, J.: Molecules, Vol. 17, No. 8, 2012, s. 9426-9442 - SCI ; SCOPUS [o1] 2013 Kang, S. - Min, H.-J. - Kang, M.-S. - Jung, M.-G. - Kim, S.: Bioorganic and Medicinal Chemistry Letters, Vol. 23, No. 6, 2013, s. 1748-1751 - SCI ; SCOPUS [o3] 2013 Madhavan, M.S. - Varghese, H.T. - Panicker, C.Y. - Mathew, S.: Natural Bond Orbital (NBO) Analysis of Certain Salicylanilide Derivatives. In: Material Science Research India, Vol. 10, 2013, s. 37-50 ADC35 Skórska-Stania, Agnieszka (20%) - Sliwa, Magdalena (20%) - Musilek, Kamil (10%) - Kuča, Kamil (10%) - Jampílek, Josef [UKOEXAF] (10%) - Musiol, Robert (10%) - Oleksyn, Barbara (10%) - Dohnal, Jiří (10%): Selected AChE reactivators in different crystalline environment: salts and enzyme Lit. 24 zázn. In: Structural Chemistry. - Vol. 21, No. 3 (2010), s. 495-501 Registrované v: wos Indikátor časopisu: IF (JCR) 2010=1,727 ADC36 Imramovský, Aleš (20%) - Peško, Matúš [UKOPREEF] (15%) - Ferriz, Juana Monreal (10%) Kráľová, Katarína [UKOPRCUS] (25%) - Vinšová, Jarmila (10%) - Jampílek, Josef [UKOEXAF] (20%): Photosynthesis-Inhibiting efficiency of 4-chloro-2-(chlorophenylcarbamoyl)phenyl alkylcarbamates
21
Lit.: 38 zázn., 1 obr., 1 tab., 1 schéma In: Bioorganic & Medicinal Chemistry Letters. - Vol. 21, No. 15 (2011), s. 4564-4567 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=2,554 Ohlasy (1): [o3] 2013 Madhavan, M.S. - Varghese, H.T. - Panicker, C.Y. - Mathew, S.: Natural Bond Orbital (NBO) Analysis of Certain Salicylanilide Derivatives. In: Material Science Research India, Vol. 10, 2013, s. 37-50 ADC37 Imramovský, Aleš (25%) - Peško, Matúš [UKOPREEF] (15%) - Kráľová, Katarína [UKOPRCUS] (15%) - Vejsova, Marcela (10%) - Stolaříková, Jiřina (10%) - Vinsova, Jarmila (10%) - Jampílek, Josef [UKOEXAF] (15%): Investigating Spectrum of BiologicalActivity of 4-and 5-Chloro-2-hydroxy-N-[2(arylamino)-1-alkyl-2-oxoethyl]benzamides Lit.: 41 zázn., 2 obr., 2 tab. In: Molecules. - Vol. 16, No. 3 (2011), s. 2414-2430 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=2,386 Ohlasy (3): [o1] 2012 Balkrishna, S.J. - Kumar, S.: Synthesis, Vol. 44, No. 9, 2012, s. 1417-1426 - SCI ; SCOPUS [o1] 2014 Güell, I. - Ribas, X.: Journal of Organic Chemistry, Vol. 2014, No. 15, 2014, s. 3188-3195 - SCI [o1] 2015 Mahesh, B. - Mohan, G. - Kabeer, S.A. - Venkateswarulu, N. - Vijaya, T. - Reddy, C.S.: Synthetic Communications, Vol. 45, No. 7, 2015, s. 838-846 - SCI ; SCOPUS ADC38 Kos, Jiří (15%) - Pěntáková, Monika (5%) - Oktábec, Zbyněk (10%) - Krejčík, Lukáš (5%) Mandelová, Zuzana (5%) - Haroková, Pavla (5%) - Hrušková, Jana (5%) - Pekárek, Tomáš (5%) Dammer, Ondrej (5%) - Tkadlecová, Marcela (5%) - Havlíček, Jaroslav(5%) - Vinšová, Jarmila (5%) Král, Vladimír (5%) - Dohnal, Jiří (5%) - Jampílek, Josef [UKOEXAF] (15%): Crystallization products of risedronate with carbohydrates and their substituted derivatives Lit. 32 zázn. In: Molecules. - Vol. 16, No. 5 (2011), s. 3740-3760 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=2,386 ADC39 Mandelová, Zuzana (15%) - Opatřilová, Radka (5%) - Raich, Ivan (15%) - Havlíček, Jaroslav (10%) Kačerová, Sandra (10%) - Pekárek, Tomáš (10%) - Tkadlecová, Marcela (10%) - Stašková, Petra (5%) Dohnal, Jiří (5%) - Csöllei, Jozef (5%) - Jampílek, Josef [UKOEXAF] (10%): Synthesis, PhysicoChemical Properties and DFT Calculations of New 2-(4-Arylpiperazine-1-yl)-1-(3-ethylbenzofuran-2yl)ethanols As Potential Antihypertensive Agents Lit. 34 zázn. In: Current Organic Chemistry. - Vol. 15, No. 7 (2011), s. 1081-1096 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=3,064 ADC40 Mrózek, Lech (15%) - Dvořáková, Lenka (15%) - Mandelová, Zuzana (5%) - Rárová, Lucie (10%) Řezáčová, Anna (5%) - Plaček, Lukáš (5%) - Opatřilová, Radka (5%) - Dohnal, Jiří (5%) - Paleta, Oldřich (5%) - Král, Vladimír (5%) - Drašar, Pavel (10%) - Jampílek, Josef [UKOEXAF] (15%): Investigation of new acyloxy derivatives of cholic acid and their esters as drug absorption modifiers Lit. 57 zázn. In: Steroids. - Vol. 76, No. 10-11 (2011), s. 1082-1097 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=2,892 ADC41 Opletalová, Veronika (15%) - Doležel, Jan (15%) - Kráľová, Katarína [UKOPRCUS] (25%) - Peško, Matúš [UKOPREEF] (15%) - Kunes, Jiří (15%) - Jampílek, Josef [UKOEXAF] (15%): Synthesis and Characterization of (Z)-5-Arylmethylidene-rhodanines with Photosynthesis-Inhibiting Properties Lit.: 58 zázn., 1 obr., 2 tab. In: Molecules. - Vol. 16, No. 6 (2011), s. 5207-5227 Registrované v: wos Indikátor časopisu:
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IF (JCR) 2011=2,386 Ohlasy (7): [o1] 2011 Jacobine, A.M. - Posner, G.H.: Journal of Organic Chemistry, Vol. 76, No. 19, 2011, s. 81218125 - SCI ; SCOPUS [o1] 2013 Han, L. - Wu, T. - Zhou, Z.: Scientific World Journal, Vol. 2013, 2013, Art. No. 543768 - SCI ; SCOPUS [o1] 2014 Guiheneuf, S. - Paquin, L., - Carreaux, F. - Durieu, E. - Roisnel, T. - Meijer, L. - Bazureau, J.P.: Molecular Diversity, Vol. 18, No. 2, 2014, s. 375-388 - SCI; SCOPUS [o1] 2014 Zapol'skii, V.A. - Namyslo, J.C. - Gjikaj, M. - Kaufmann, D.E.: Beilstein Journal of Organic Chemistry, Vol. 10, Art. No. 170, 2014, s. 1638-1644 - SCI; SCOPUS [o1] 2014 Ramesh, V. - Ananda Rao, B. - Sharma, P. - Swarna, B. - Thummuri, D. - Srinivas, K. - Naidu, V.G.M. - Jayathirtha Rao, V.: European Journal of Medicinal Chemistry, Vol. 83, August, 2014, s. 569580 - SCI; SCOPUS [o1] 2014 Jadav, S.S. - Sinha, B.N. - Hilgenfeld, R. - Pastorino, B. - de Lamballerie, X. - Jayaprakash, V.: European Journal of Medicinal Chemistry, Vol. 89, 2014, s. 172-178 - SCOPUS [o3] 2014 Guihéneuf, S. - Paquin, L. - Carreaux,F. - Durieu, E. - Bénédetti, H. - Le Guével, R.l. - Corlu,A. - Meijer, L. - Bazureau J.: Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects. In: Current Microwave Chemistry, Vol. 1, No. 1, 2014, s. 40 ADC42 Pejchal, Vladimír (20%) - Štěpánková, Šárka (20%) - Padělková, Zdeňka (20%) - Imramovský, Aleš (20%) - Jampílek, Josef [UKOEXAF] (20%): 1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes Lit. 49 zázn. In: Molecules. - Vol. 16, No. 9 (2011), s. 7565-7582 Registrované v: wos Indikátor časopisu: IF (JCR) 2011=2,386 ADC43 Bobáľ, Pavel (20%) - Sujan, Josef (20%) - Otevřel, Jan (20%) - Imramovský, Aleš (10%) - Padělková, Zdeňka (10%) - Jampílek, Josef [UKOEXAF] (20%): Microwave-assisted synthesis of new substituted anilides of quinaldic acid Lit. 44 zázn. In: Molecules. - Vol. 17, No. 2 (2012), s. 1292-1306 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (3): [o1] 2013 Ju, L. - Yao, J.Z. - Wu, Z.H. - Liu, Z.X. - Zhang, Y.H.: Journal of Organic Chemistry, Vol. 78, No. 21, 2013, s. 10831 - SCI [o1] 2014 Lukasik, N. - Wagner-Wysiecka, E.: Current Organic Synthesis, Vol. 11, No. 4, 2014, s. 604 SCI [o1] 2015 Latimer, D. - Wiebe, M.: Green Chemistry Letters and Reviews, Vol. 8, No. 2, 2015, s. 42 - SCI ADC44 Brychtová, Kateřina (20%) - Dvořáková, Lenka (10%) - Opatřilová, Radka (5%) - Raich, Ivan (10%) Kačerová, Sandra (10%) - Plaček, Lukáš (5%) - Kalinowski, Danuta S. (10%) - Richardson, Des R. (10%) - Jampílek, Josef [UKOEXAF] (20%): Investigationof substituted 6-aminohexanoates as skin penetration enhancers Lit. 55 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 20, No. 1 (2012), s. 86-95 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,903 Ohlasy (1): [o1] 2013 Marepally, S. - Boakye, C.H.A. - Shah, P.P. - Etukala, J.R. - Vemuri, A. - Singh, M.: PLoS ONE, Vol. 8, No. 12, 2013, Article No. UNSP e82581 - SCI ADC45 Cieslik, Wioleta (20%) - Jampílek, Josef [UKOEXAF] (15%) - Musiol, Robert (15%) - Nycz, Jacek E. (10%) - Vejsová, Marcela (10%) - Machura, Barbara (10%) - Wolff, Mariusz (10%) - Polanski, Jaroslaw (10%): Contribution to investigation of antimicrobial activity of styrylquinolines Lit. 56 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 20, No. 24 (2012), s. 6960-6968
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Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,903 Ohlasy (5): [o1] 2013 Radchatawedchakoon, W. - Promthong, N. - Sakee, U.: Letters in Organic Chemistry, Vol. 10, No. 9, 2013, s. 644 - SCI; SCOPUS [o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: European Journal of Pharmaceutical Sciences, Vol. 51, 2014, s. 203 - SCI; SCOPUS [o1] 2014 Muscia, G.C. - Hautmann, S. - Buldain, G.Y. - Asis, S.E. - Gutschow, M.: Bioorganic & Medicinal Chemistry Letters, Vol. 24, No. 6, 2014, s. 1549 - SCI; SCOPUS [o1] 2015 Xiao, J.C. - Huang, Y. - Song, Z.L. - Feng, W.H.: RSC Advances, Vol. 5, No. 10, 2015, s. 99098 - SCI; SCOPUS [o1] 2015 Huang, L. - Fei, T.H. - Hu, K. - Liu, F.M.: Journal of Heterocyclic Chemistry, Vol. 52, No. 3, 2015, s. 906 - SCI; SCOPUS ADC46 Fajkusová, Dagmar (25%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (5%) - Guo, Jiahui (5%) - Oktábec, Zbyněk (5%) - Vejsová, Marcela (5%) - Kollár, Peter (5%) - Coffey, Aidan (10%) Csöllei, Jozef (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Anti-infective and herbicidal activity of N-substituted 2-aminobenzothiazoles Lit.: 50 zázn., 5 obr., 2 tab. In: Bioorganic & Medicinal Chemistry. - Vol. 20, No. 24 (2012), s. 7059-7068 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,903 Ohlasy (3): [o1] 2013 Zhao, J.W. - Huang, H.W. - Wu, W.Q. - Chen, H.J. - Jiang, H.F.: Organic Letters, Vol. 15, No. 11, 2013, s. 2604-2607 - SCI [o1] 2015 Keri, R.S. - Patil, M.R. - Patil, S.A. - Budagupi, S.: European Journal of Medicinal Chemistry, Vol. 89, January, 2015, s. 207-251 - SCI ; SCOPUS [o1] 2015 Seddighi, M. - Shirini, F. - Mamaghani, M.: Comptes Rendus Chimie, Vol. 18, No. 5, 2015, s. 573-580 - SCI ; SCOPUS ADC47 Goněc, Tomáš (15%) - Bobáľ, Pavel (5%) - Sujan, Josef (5%) - Peško, Matúš [UKOPREEF] (10%) Guo, Jiahui (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Pavlacká, Lenka (5%) - Veselý, Libor (5%) Kreckova, Eva (5%) - Kos, Jiří (5%) - Coffey, Aidan (5%) - Kollár, Peter [UKOEXAF] (5%) Imramovský, Aleš (5%) - Plaček, Lukaš (5%) - Jampílek, Josef [UKOEXAF] (10%): Investigating the Spectrum of Biological Activity of Substituted Quinoline-2-Carboxamides and Their Isosteres Lit.: 61 zázn., 4 obr., 3 tab. In: Molecules. - Vol. 17, No. 1 (2012), s. 613-644 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (9): [o1] 2013 Tian, T. - Zhong, W.H. - Meng, S. - Meng, X.B. - Li, Z.J.: Journal of Organic Chemistry, Vol. 78, No. 2, 2013, s. 728-732 - SCI; SCOPUS [o1] 2013 Mamidi, N. - Manna, D.: Journal of Organic Chemistry, Vol.78, No. 6, 2013, s. 2386-2396 SCI; SCOPUS [o1] 2014 Hassan, W.M.I. - Moustafa, H. - Hamed, M.N.H. - Ali, L.I. - Halim, S.A.: Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy, Vol. 117, 2014, s. 587-597 - SCI; SCOPUS [o1] 2014 Babjak, M. - Caletková, O. - Ďurišová, D. - Gracza, T.: Synlett, Vol. 25, No. 18, 2014, Art. No. st-2014-b0535-1, s. 2579-2584 - SCI; SCOPUS [o1] 2014 Keri, R.S. - Patil, S.A.: Biomedicine and Pharmacotherapy, Vol. 68, No. 8, 2014, s. 1161-1175 SCI; SCOPUS [o1] 2015 Funder, E.D. - Trads, J.B. - Gothelf, K.V.: Organic and Biomolecular Chemistry, Vol. 13, No. 1, 2015, s. 185-198 - SCI ; SCOPUS [o3] 2015 Baluja, S.: Dissociation Constants of Some Quinoline Derivatives in Mixed Solvent mixture. In: International Letters of Chemistry, Physics and Astronomy, International Letters of Chemistry, Physics and Astronomy, Vol. 9, No. 1, 2015, s. 32-36 [o3] 2015 Boyarshinov V.D. - Mikhalev A.I. - Yushkova T.A. - Konshina T.A. - Ukhov S.V.: Synthesis and biological activity quinoline-2-carboxamides. In: Pharmaceutical Sciences, Fundamental Research, No. 2, 2015, s. 1715-1719
24
[o1] 2015 Xie, H. - Liao, Y. - Chen, S. - Chen, Y. - Deng, G.-J.: Organic and Biomolecular Chemistry, Vol. 13, No. 25, 2015, s. 6944-6948 - SCI; SCOPUS ADC48 Imramovský, Aleš (16%) - Štěpánková, Šárka (14%) - Vančo, Ján [UKOEXAF] (14%) - Pauk, Jozef (14%) - Monreal-Ferriz, Juana (14%) - Vinšová, Jarmila (14%) - Jampílek, Josef [UKOEXAF] (14%): Acetylcholinesterase-inhibiting activity of salicylanilide N-alkylcarbamates and their molecular docking Lit. 50 zázn. In: Molecules. - Vol. 17, No. 9 (2012), s. 10142-10158 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (7): [o1] 2014 Das, R.N. - Roy, K.: Industrial & Engineering Chemistry Research, Vol. 53, No. 2, 2014, s. 1032 - SCI [o1] 2014 Lo, R. - Ganguly, B.: Molecular Biosystems, Vol. 10, No. 9, 2013, s. 2383 - SCI [o1] 2014 Varadaraju, K.R. - Kumar, J.R. - Mallesha, L. - Muruli, A. - Mohana, K.N.S. - Mukunda, C.K. Sharanaiah, U.: International Journal of Alzheimer's Disease, Vol. 2013, art.no. 653962 - SCOPUS [o1] 2015 Gocer, H. - Akincioglu, A. - Goksu, S. - Gulcin, I. - Supuran, C.T.: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 30, No. 2, 2015, s. 320 - SCI [o1] 2015 Thangnipon, W. - Suwanna, N. - Jantrachotechatchawan, C. - Ngampramuan, S. - Tuchinda, P. Nobsathian, S.: Archives of Pharmacal Research, Vol. 38, No. 7, 2015, s. 1388 - SCI [o1] 2015 Basant, N. - Gupta, S. - Singh, K.P.: Journal of Molecular Liquids, Vol. 209, 2015, s. 412 - SCI [o1] 2015 Kose, L.P. - Gulcin, I. - Goren, A.C. - Namiesnik, J. - Martinez-Ayala, A.L. - Gorinstein, S.: Industrial Crops and Products, Vol. 74, 2015, s. 721 - SCI ADC49 Jampílek, Josef [UKOEXAF] (60%) - Brychtová, Kateřina (40%): Azone analogues: classification, design, and transdermal penetration principles Lit. 238 zázn. In: Medicinal Research Reviews. - Vol. 32, No. 5 (2012), s. 907-947 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=9,583 ADC50 Serda, Maciej (20%) - Mrozek-Wilczkiewicz, Anna (10%) - Peško, Matúš [UKOPREEF] (10%) Kráľová, Katarína [UKOPRCUS] (10%) - Vejsova, Marcela (10%) - Musiol, Robert (10%) - Ratuszna, Alicja (10%) - Polanski, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (10%): Investigation of the Biological Properties of (Hetero)Aromatic Thiosemicarbazones Lit.: 55 zázn., 4 obr., 3 tab. In: Molecules. - Vol. 17, No. 11 (2012), s. 13483-13502 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (4): [o1] 2014 Pino-Cuevas, A. - Carballo, R. - Vázquez-López, E.M.: Acta Crystallographica Section E: Structure Reports Online, Vol. 70, No. 9, 2014, s. o926 - SCOPUS [o1] 2014 Carballo, R. - Pino-Cuevas, A. - Ezequiel, M. - Vazquez-Lopez, E.M.: Acta Crystallographica Section E: Structure Reports Online, Vol. 70, No. 9, 2014, s. o970 S - SCOPUS [o1] 2014 Paiva, R.O. - Kneipp, L.F. - Goular, C.M. - Albuquerque, M.A. - Echevarria, A.: Ciencia e Agrotecnologia, Vol. 38, No. 6, 2014, s. 531-537 - SCOPUS; SCI [o1] 2015 Cui, J. - Lin, Q. - Gan, C. - Zhan, J. - Su, W. - Zhao, D. - Qi, B. - Huang, Y.: Steroids, Vol. 98, Art. No. 7766, 2015, s. 138-142 - SCOPUS ADC51 Vaculiková, Eliška (30%) - Grünwaldová, Veronika (20%) - Král, Vladimír (15%) - Dohnal, Jiří (10%) Jampílek, Josef [UKOEXAF] (25%): Primary Investigation of the Preparation of Nanoparticles by Precipitation Lit. 30 zázn. In: Molecules. - Vol. 17, No. 9 (2012), s. 11067-11078 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (1):
25
[o1] 2015 Pinjari, D.V. - Prasad, K. - Gogate, P.R. - Mhaske, S.T. - Pandit, A.B.: Ultrasonics Sonochemistry, Vol. 23, 2015, s. 191 - SCI ADC52 Vaculiková, Eliška (30%) - Grünwaldová, Veronika (20%) - Král, Vladimír (15%) - Dohnal, Jiří (10%) Jampílek, Josef [UKOEXAF] (25%): Preparation of candesartan and atorvastatin nanoparticles by solvent evaporation Lit. 46 zázn. In: Molecules. - Vol. 17, No. 11 (2012), s. 13221-13234 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,428 Ohlasy (5): [o1] 2013 Anarjan, N. - Tan, C.P.: Molecules, Vol. 18, No. 1, 2013, s. 777 - SCI [o1] 2015 Yeom, D.W. - Song, Y.S. - Kim, S.R. - Lee, S.G. - Kang, M.H. - Lee, S. - Choi, Y.W.: International Journal of Nanomedicine, Vol. 10, 2015, s. 3878 - SCI [o1] 2015 Sezgin-Bayindir, Z. - Antep, M.N. - Yuksel, N.: AAPS PharmSciTech, Vol. 16, No. 1, 2015, s. 117 - SCI [o1] 2015 Agrawal, A.G. - Kumar, A. - Gide, P.S.: Drug Development and Industrial Pharmacy, Vol. 41, No. 4, 2015, s. 604 - SCI [o1] 2015 Hennig, R. - Ohlmann, A. - Staffel, J. - Pollinger, K. - Haunberger, A. - Breunig, M. - Schweda, F. - Tamm, E.R. - Goepferich, A.: Journal of Controlled Release, Vol. 22, 2015, s. 274 - SCI ADC53 Zitko, Jan (25%) - Jampílek, Josef [UKOEXAF] (20%) - Dobrovolný, Lukáš (25%) - Svobodová, Michaela (10%) - Kuneš, Jiří (10%) - Doležal, Martin (10%): Synthesis and antimycobacterial evaluation of N-substituted 3-aminopyrazine-2,5-dicarbonitriles Lit. 23 zázn. In: Bioorganic & Medicinal Chemistry Letters. - Vol. 22, No. 4 (2012), s. 1598-1601 Registrované v: wos Indikátor časopisu: IF (JCR) 2012=2,338 ADC54 Coufalová, Lenka (10%) - Mrózek, Lech (10%) - Rárová, Lucie (10%) - Plaček, Lukáš (10%) Opatřilová, Radka (10%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Paleta, Oldřich (5%) - Král, Vladimír (10%) - Drašar, Pavel (10%) - Jampílek, Josef [UKOEXAF] (10%): New propanoyloxy derivatives of 5 beta-cholan-24-oic acid as drug absorption modifiers Lit.: 68 zázn., 4 obr., 5 schém, 2 tab. In: Steroids. - Vol. 78, No. 5 (2013), s. 435-453 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,716 Ohlasy (5): [o1] 2013 Perrone, D. - Bortolini, O. - Fogagnolo, M. - Marchesi, E. - Mari, L. - Massarenti, C. Navacchia, M.L. - Sforza, F. - Varani, K. - Capobianco, M.L.: New Journal of Chemistry, Vol. 37, No. 1, 2013, s. 3559-3567 - SCI [o1] 2014 Ojewole, E. - Kalhapure, R. - Akamanchi, K. - Govender, T.: Drug Development and Industrial Pharmacy, Vol. 40, No. 5, 2014, s. 657-668 - SCOPUS [o1] 2014 Yang, Y.X. - Zheng, L.T. - Shi, J.J. - Gao, B. - Chen, Y.K. - Yang, H.C. - Chen, H.L. - Li, Y.C. - Zhen, X.C.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No. 4, 2014, s. 1222-1227 - SCI ; SCOPUS [o1] 2015 Poša, M. - Bjedov, S. - Škoric, D. - Sakač, M.: Biochimica et Biophysica Acta - General Subjects, Vol. 1850, No. 7, 2015, s. 1345-1353 - SCOPUS [o1] 2015 Moghimipour, E. - Ameri, A. - Handali, S.: Molecules, Vol. 20, No. 8, 2015, s. 14451-14473 SCOPUS ADC55 Čulen, Martin (25%) - Řezáčová, Anna (25%) - Jampílek, Josef [UKOEXAF] (25%) - Dohnal, Jiří (25%): Designing a Dynamic Dissolution Method: A Review of Instrumental Options and Corresponding Physiology of Stomach and Small Intestine Lit. 111 zázn. In: Journal of Pharmaceutical Sciences. - Vol. 102, No. 9 (2013), s. 2995-3017 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=3,007
26
Ohlasy (6): [o1] 2014 Zhao, Y. - Bettinger, J. - Caritis, S. - Venicataramanan, R.: American Journal of Health-System Pharmacy, Vol. 71, No. 13, 2014, s. 1127 - SCI [o1] 2014 Nokhodchi, A. - Asare-Addo, K.: Expert Opinion on Drug Delivery, Vol. 11, No. 9, 2014, s. 1418 - SCI [o1] 2014 Hens, B. - Brouwers, J. - Anneveld, B. - Corsetti, M. - Symillides, M. - Vertzoni, M. - Reppas, C. - Turner, D.B. - Augustijns, P.: European Journal of Pharmaceutical Sciences, Vol. 63, 2014, s. 242 SCI [o1] 2014 Rhee, K.H. - Park, J.S. - Cho, M.J.: Yonsei Medical Journal, Vol. 55, No. 6, 2014, s. 1466 - SCI [o1] 2014 Wu, P. - Chen, L.D. - Wu, X. - Chen, X.D.: Journal of Food Engineering, Vol. 142, 2014, s. 178 - SCI [o1] 2015 Wuyts, B. - Riethorst, D. - Brouwers, J. - Tack, J. - Annaert, P. - Augustijns, P.: European Journal of Pharmaceutical Sciences, Vol. 67, 2015, s. 135 - SCI ADC56 Goněc, Tomáš (10%) - Kos, Jiří (5%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%) Govender, Rodney (5%) - Keltošová, Stanislava (5%) - Chambel, Barbara (5%) - Pereira, Diogo (5%) Kollár, Peter (5%) - Imramovský, Aleš (5%) – O´Mahony, Jim (5%) - Coffey, Aidan (5%) - Čížek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Antibacterial and herbicidal activity of ring-substituted 2-hydroxynaphthalene-1-carboxanilides Lit.: 60 zázn., 3 obr., 1 tab. In: Molecules. - Vol. 18, No. 8 (2013), s. 9397-9419 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,095 Ohlasy (1): [o1] 2015 Kotb, E.R. - Anwar, M.M. - Syam, Y.M. - Bagato, O. - AbdelMoaz, S.: International Journal of Pharmacy and Technology, Vol. 7, No. 1, 2015, s. 8237-8273 - SCOPUS ADC57 Goněc, Tomáš (10%) - Kos, Jiří (10%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (10%) - Tengler, Jan (10%) - Bobáľ, Pavel (5%) - Kollár, Peter (5%) - Čížek, Alois (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Antimycobacterial and herbicidal activity of ring-substituted 1-hydroxynaphthalene-2-carboxanilides Lit.: 50 zázn., 5 obr., 1 schéma, 1 tab. In: Bioorganic & Medicinal Chemistry. - Vol. 21, No. 21 (2013), s. 6531-6541 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,951 Ohlasy (3): [o1] 2014 Xu, S. - Li, D. - Pei, L. - Yao, H. - Wang, C. - Cai, H. - Yao, H. - Wu, X. - Xu, J.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No. 13, 2014, s. 2811-2814 - SCOPUS; SCI [o1] 2014 Chaaban, I. - El Khawass, E.S.M. - Abd El Razik, H.A. - El Salamouni, N.S. - RedondoHorcajo, M. - Barasoain, I. - Díaz, J.F. - Yli-Kauhaluoma, J. - Moreira, V.M.: European Journal of Medicinal Chemistry, Vol. 87, November, 2014, s.805-813 - SCOPUS; SCI [o1] 2015 Brahmachari, G.: ACS Sustainable Chemistry and Engineering, Vol. 3, No. 9, 2015, s. 20582066 - SCOPUS; SCI ADC58 Imramovský, Aleš (10%) - Pejchal, Vladimír (9%) - Štěpánková, Šárka (9%) - Vorčáková, Katarína (9%) - Vančo, Ján [UKOEXAF] (9%) - Šimůnek, Petr (9%) - Královec, Karel (9%) - Brůčková Lenka (9%) - Mandíková, Jana (9%) - Trejtnar, František (9%) - Jampílek, Josef [UKOEXAF] (9%): Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors Lit. 60 zázn. In: Bioorganic & Medicinal Chemistry Letters. - Vol. 21, No. 7 (2013), s. 1735-1748 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,095 Ohlasy (4): [o1] 2014 Du, X.J. - Bian, Q. - Wang, H.X. - Yu, S.J. - Kou, J.J. - Wang, Z.P. - Li, Z.M. - Zhao, W.G.: Organic & Biomolecular Chemistry, Vol. 12, No. 29, 2014, s. 5434 - SCI [o1] 2014 Gundogdu-Karaburun, N.: Letters in Drug Design & Discovery, Vol. 11, No.6, 2014, s. 823 SCI
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[o1] 2015 Keri, R.S. - Patil, M.R. - Patil, S.A. - Budagupi, S.: European Journal of Medicinal Chemistry, Vol. 89, 2015, s. 251 - SCOPUS [o1] 2015 Hroch, L. - Aitken, L. - Benek, O. - Dolezal, M. - Kuca, K. - Gunn-Moore, F. - Musilek, K.: Current Medicinal Chemistry, Vol. 22, No. 6, 2015, s. 747 - SCI ADC59 Kos, Jiří (20%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (5%) - Tengler, Jan (5%) - Goněc, Tomáš (5%) - Bobáľ, Pavel (5%) - Kauerová, Tereza (5%) - Oravec, Michal (5%) - Kollár, Peter (5%) - Čížek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) Jampílek, Josef [UKOEXAF] (10%): Antibacterial and herbicidal activity of ring-substituted 3hydroxynaphthalene-2-carboxanilides Lit.: 55 zázn., 3 obr., 1 schéma, 1 tab. In: Molecules. - Vol. 18, No. 7 (2013), s. 7977-7997 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,095 ADC60 Mrózek, Lech (20%) - Coufalová, Lenka (10%) - Rárová, Lucie (10%) - Plaček, Lukáš (5%) Opatřilová, Radka (10%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Paleta, Oldřich (10%) - Král, Vladimír (5%) - Drašar, Pavel (5%) - Jampílek, Josef [UKOEXAF] (10%): New polyfluorothiopropanoyloxy derivatives of 5 beta-cholan-24-oic acid designed as drug absorption modifiers Lit.: 67 zázn., 4 obr., 2 schémy, 1 tab. In: Steroids. - Vol. 78, No. 9 (2013), s. 832-844 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,716 Ohlasy (2): [o1] 2014 Ojewole, E. - Kalhapure, R. - Akamanchi, K. - Govender, T.: Drug Development and Industrial Pharmacy, Vol. 40, No. 5, 2014, s. 657-668 - SCI; SCOPUS [o1] 2015 Poša, M. - Bjedov, S. - Škoric, D. - Sakač, M.: Biochimica et Biophysica Acta - General Subjects, Vol. 1850, No. 7, 2015, s. 1345-1353 - SCOPUS; SCI ADC61 Otevřel, Jan (10%) - Bobáľ, Pavel (5%) - Zadražilová, Iveta (10%) - Govender, Rodney (5%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (5%) - Kolečkárová, Petra (5%) - Maršálek, Petr (5%) - Imramovský, Aleš (5%) - Coffey, Aidan (5%) – O´Mahony, Jim (5%) - Kollár, Peter (5%) - Čížek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Antimycobacterial and photosynthetic electron transport inhibiting activity of ring-substituted4-arylamino-7chloroquinolinium chlorides Lit.: 68 zázn., 3 obr., 1 schéma, 1 tab. In: Molecules. - Vol. 18, No. 9 (2013), s. 10648-10670 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,095 ADC62 Pauk, Karel (25%) - Zadražilová, Iveta (20%) - Imramovský, Aleš (10%) - Vinšová, Jarmila (5%) Pokorná, Michaela (10%) - Masaříková, Martina (5%) - Čížek, Alois (5%) - Jampílek, Josef [UKOEXAF] (20%): New derivatives of salicylamides: Preparationand antimicrobial activity against various bacterial species Lit. 44 zázn. In: Bioorganic & Medicinal Chemistry. - Vol. 21, No. 21 (2013), s. 6574-6581 Registrované v: wos Indikátor časopisu: IF (JCR) 2013=2,951 Ohlasy (1): [o1] 2015 Rajamuthiah, R. - Fuchs, B.B. - Conery, A.L. - Kim, W. - Jayamani, E. - Kwon, B. - Ausubel, F.M. - Mylonakis, E.: PLoS ONE, Vol. 10, No. 4, Article No. UNSP e0124595 - SCI ADC63 Tengler, Jan (20%) - Kapustíková, Iva (20%) - Stropnický, Ondřej (20%) - Mokrý, Petr (10%) - Oravec, Michal (5%) - Csöllei, Jozef (5%) - Jampílek, Josef [UKOEXAF] (20%): Synthesis of new (arylcarbonyloxy)aminopropanol derivatives and the determination of their physico-chemical properties Lit. 36 zázn. In: Central European Journal of Chemistry. - Vol. 11, No. 11 (2013), s. 1757-1767 Registrované v: wos
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Indikátor časopisu: IF (JCR) [2013-1,329] ADC64 Goněc, Tomáš (15%) - Kos, Jiří (5%) - Nevin, Eoghan (5%) - Govender, Rodney (5%) - Peško, Matúš [UKOPREEF] (10%) - Tengler, Jan (5%) - Kushkevych, Ivan (5%) - Šťastná, Vendula (5%) - Oravec, Michal (10%) - Kollár, Peter (5%) – O´Mahony, Jim (5%) - Kráľová, Katarína [UKOPRCUS] (10%) Coffey, Aidan (5%) - Jampílek, Josef [UKOEXAF] (10%): Preparation and Biological Properties of RingSubstituted Naphthalene-1-Carboxanilides Lit.: 46 zázn., 3 obr., 4 tab. In: Molecules. - Vol. 19, No. 7 (2014), s. 10386-10409 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2014=2,416 ADC65 Imramovský, Aleš (25%) - Peško, Matúš [UKOPREEF] (25%) - Kráľová, Katarína [UKOPRCUS] (25%) - Jampílek, Josef [UKOEXAF] (25%): Synthesis and photosynthetic electron transport inhibition of 2-substituted 6-fluorobenzothiazoles Lit.: 39 zázn., 2 obr., 1 schéma, 1 tab. In: Monatshefte für Chemie. - Vol. 145, No. 11 (2014), s. 1817-1824 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2014=1,222 ADC66 Jampílek, Josef [UKOEXAF] (100%) : Recent advances in design of potential quinoxaline antiinfectives Lit. 267 zázn. In: Current Medicinal Chemistry. - Vol. 21, No. 38 (2014), s. 4347-4373 Registrované v: wos Indikátor časopisu: IF (JCR) 2014=3,853 ADC67 Krompiec, Stanislav (10%) - Malarz, Joanna (10%) - Pietraszuk, Cezary (10%) - Powala, Beata (5%) Rogalski, Szymon (5%) - Malecki, Jan G. (5%) - Penkala, Mateusz (5%) - Filapek, Michal (5%) - Musiol, Robert (5%) - Jampílek, Josef [UKOEXAF] (5%) - Vejsova, Marcela (5%) - Polanski, Jaroslaw (5%) Paluch, Marian (5%) - Pawlus, Sebastian (5%) - Danikiewicz, Witold (5%) - Kania, Magdalena (5%) Marcol, Beata (5%): New strategy for the synthesis of 3,4,5-trisubstituted isoxazolines from allylcompounds Lit. 78 zázn. In: Current Organic Chemistry. - Vol. 18, No. 17 (2014), s. 2280-2296 Registrované v: wos Indikátor časopisu: IF (JCR) 2014=2,157 ADC68 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (20%) - Musiol, Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Anto, P. L. (10%) - Van Alsenoy, Christian (10%): Spectroscopic (FT-IR, FT-Raman) investigations and quantum chemical calculations of 4-hydroxy-2-oxo1,2-dihydroquinoline-7-carboxylic acid Lit. 61 zázn. In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 121 (2014), s. 404-414 Registrované v: wos Indikátor časopisu: IF (JCR) 2014=2,353 ADC69 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (20%) - Musiol, Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Anto, P. L. (10%) - Van Alsenoy, Christian (10%): Vibrational spectroscopic, H-1 NMR and quantum chemical computational study of 4-hydroxy-2-oxo-1, 2dihydroquinoline-8-carboxylic acid Lit. 70 zázn. In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 121 (2014), s. 445-456 Registrované v: wos Indikátor časopisu: IF (JCR) 2014=2,353 Ohlasy (1):
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[o1] 2015 Al-Otaibi, J.S. - Ai-Wabli, R.I.: Spectrochimica Acta Part A-Molecular and Biomolecular Spectroscopy, Vol. 137, 2015, s. 15 - SCI ADC70 Vaculiková, Eliška (14%) - Plachá, Daniela (14%) - Pisárčik, Martin [UKOFACH] (15%) - Peikertová, Pavlína (14%) - Dedková, Kateřina (14%) - Devínsky, Ferdinand [UKOFACH] (15%) - Jampílek, Josef [UKOEXAF] (14%): Preparation of Risedronate Nanoparticles by Solvent Evaporation Technique Lit. 30 zázn. In: Molecules. - Vol. 19, No. 11 (2014), s. 17848-17861 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2014=2,416 SJR (SCOPUS) [2014-0,650] SNIP (SCOPUS) [2014-1,220] Ohlasy (2): [o1] 2015 Rawat, P. - Manglani, K. - Gupta, S. - Kalam, A. - Vohora, D. - Ahmad, F.J. - Talegaonkar, S.: Pharmaceutical Research, Vol. 32, No. 10, 2015, s. 3158 - SCOPUS; SCI [o1] 2015 Sun, D.Q. - Xue, A.Y. - Zhang, B. - Lou, H.Y. - Shi, H.Y. - Zhang, X.M.: Journal of Pharmacy and Pharmacology, Vol. 67, No. 12, 2015, s. 1662 - SCI ADC71 Goněc, Tomáš (20%) - Zadražilová, Iveta (5%) - Nevin, Eoghan (5%) - Krauerová, Tereza (5%) Peško, Matúš [UKOPREEF] (10%) - Kos, Jiří (5%) - Oravec, Michal (5%) - Kollár, Peter (5%) - Coffey, Aidan (10%) - O Mahony, Jim (5%) - Cizek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) Jampílek, Josef [UKOEXAF] (10%): Synthesis and Biological Evaluation of N-Alkoxyphenyl-3hydroxynaphthalene-2-carboxanilides Lit.: 48 zázn., 3 obr., 1 tab. In: Molecules. - Vol. 20, No. 6 (2015), s. 9767-9787 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2015= [2014-2,416] ADC72 Kos, Jiří (10%) - Nevin, Eoghan (10%) - Šoral, Michal (10%) - Kushkevych, Ivan (10%) - Goněc, Tomáš (5%) - Bobáľ, Pavel (10%) - Kollár, Peter (5%) - Coffey, Aidan (5%) – O´Mahony, Jim (10%) Liptaj, Tibor (10%) - Kráľová, Katarína [UKOPRCUS] (5%)- Jampílek, Josef [UKOEXAF] (10%): Synthesis and antimycobacterial properties of ring-substituted 6-hydroxynaphthalene-2-carboxanilides Lit.: 42 zázn., 4 obr., 1 tab. In: Bioorganic & Medicinal Chemistry. - Vol. 23, No. 9 (2015), s. 2035-2043 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2015= [2014-2,793] Ohlasy (1): [o1] 2015 Xiao, Z.P. - Wei, W. - Wang, P.F. - Shi, W.K. - Zhu, N. - Xie, M.Q. - Sun, Y.W. - Li, L.X. Xie, Y.X. - Zhu, L.S. - Tang, N. - Ouyang, H. - Li, X.H. - Wang, G.C. - Zhu, H.L.: European Journal of Medicinal Chemistry, Vol. 102, Art.No. 8061, 2015, s. 631-638 - SCOPUS ADC73 Kos, Jiří (20%) - Zadražilová, Iveta (5%) - Nevin, Eoghan (10%) - Šoral, Michal (10%) - Goněc, Tomáš (5%) - Kollár, Peter (5%) - Oravec, Michal (5%) - Coffey, Aidan (5%) - O Mahony, Jim (5%) - Liptaj, Tibor (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Ringsubstituted 8-hydroxyquinoline-2-carboxanilides as potential antimycobacterial agents Lit.: 50 zázn.,3 obr., 1 tab. In: Bioorganic and Medicinal Chemistry. - Vol 23, No. 15 (2015), s. 4188-4196 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) 2015= [2014-2,793] ADC74 Peško, Matúš [UKOPREEF] (40%) - Kos, Jiří (20%) - Kráľová, Katarína [UKOPRCUS] (20%) Jampílek, Josef [UKOEXAF] (20%): Inhibition of photosynthetic electron transport by 6hydroxynaphthalene-2-carboxanilides Lit. 48 zázn., 2 obr., 1 tab. In: Indian Journal of Chemistry Section B-Organic Chemistry Including Medicinal Chemistry. - Vol. 54, No. 12 (2015), s. 1511-1517 Registrované v: wos Indikátor časopisu: IF (JCR) 2015= [2014-0,387]
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ADC75 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (10%) - Musiol, Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Van Alsenoy, Christian (10%) - War, Javeed Ahmad (10%) - Manojkumar, T. K. (10%): Vibrational spectroscopic studies and molecular docking study of 2[(E)-2-phenylethenyl]quinoline-5-carboxylic acid Lit. 47 zázn. In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 150 (2015), s. 190-199 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-2,353] ADC76 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (10%) - Musiol, Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Van Alsenoy, Christian (10%) - War, Javeed Ahmad (10%) - Al-Saadi, Abdulaziz A. (10%): Vibrational spectroscopic and molecular docking study of (2E)-N(4-chloro-2-oxo-1,2-dihydroquinolin-3-yl)-3-phenylprop-2-enamide Lit. 65 zázn. In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 151 (2015), s. 335-349 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-2,353] ADC77 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (10%) - Musiol, Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Van Alsenoy, Christian (10%) - War, Javeed Ahmad (10%) - Srivastava, S. K. (10%): Molecular structure,FT-IR, FT-Raman, NBO, HOMO and LUMO, MEP, NLO and molecular docking study of 2-[(E)-2-(2-bromophenyl)ethenyl]quinoline-6-carboxylic acid Lit. 65 zázn. In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 151 (2015), s. 184-197 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-2,353] ADC78 Zdražilová, Iveta (25%) - Pospíšilová, Šárka (25%) - Masariková, Martina (5%) - Imramovský, Aleš (5%) - Ferriz, Juana Monreal (5%) - Vinšová, Jarmila (5%) - Čížek, Alois (10%) - Jampílek, Josef [UKOEXAF] (20%): Salicylanilide carbamates: Promising antibacterial agents with high in vitro activity against methicillin-resistant Staphylococcus aureus (MRSA) Lit. 70 zázn. In: European Journal of Pharmaceutical Sciences. - Vol. 77 (2015), s. 197-207 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-3,350] ADC79 Jampílek, Josef [UKOEXAF] (100%) : Potential of agricultural fungicides for antifungal drug discovery Lit. 45 zázn. In: Expert Opinion on Drug Discovery. - Vol. 11, No. 1 (2016), s. 1-9 Indikátor časopisu: IF (JCR) [2014-3,539] ADD Vědecké práce v domácích karentovaných časopisech ADD01 Kučerová-Chlupáčová, Marta (20%) - Opletalová, Veronika (20%) - Jampílek, Josef [UKOEXAF] (20%) - Doležel, Jan (20%) - Dohnal, Jiří (5%) - Pour, Milan (5%) - Kuneš, Jiří (5%) - Vořišek, Viktor (5%): New hydrophobicity constants of substituents in pyrazine rings derived from RP-HPLC study Lit. 29 zázn. In: Collection of Czechoslovak Chemical Communications. - Vol. 73, No. 1 (2008), s. 1-18 Registrované v: wos Indikátor časopisu: IF (JCR) [2008-0,784] ADD02 Oktábec, Zbyněk (50%) - Jampílek, Josef [UKOEXAF] (50%): Stručná historie chemoterapie = Brief history of chemotherapy Lit. 77 zázn. In: Chemické listy. - Roč. 107, č. 2 (2013), s. 150-158 Registrované v: wos Indikátor časopisu: IF (JCR) [2013-0,196]
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ADD03 Černíková, Aneta (50%) - Jampílek, Josef [UKOEXAF] (50%): Strukturní modifikace léčiv ovlivňující biodostupnost a terapeutický účinek = Structure modification of drugs or prodrugs influencing their bioavailability and therapeutic effect Lit. 70 zázn. In: Chemické listy. - Roč. 108, č. 1 (2014), s. 7-16 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-0,272] ADD04 Pěntáková, Monika (50%) - Jampílek, Josef [UKOEXAF] (50%): Patentová historie přípravku Viagra(R) = Patent history of Viagra(R) preparation Lit. 14 zázn. In: Chemické listy. - Roč. 109, č. 6 (2015), s. 415-417 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-0,272] ADD05 Vaculiková, Eliška (50%) - Plachá, Daniela (25%) - Jampílek, Josef [UKOEXAF] (25%): Toxikologie nanoforem nosičů léčiv = Toxicology of drug nanocarriers Lit. 74 zázn. In: Chemické listy. - Roč. 109, č. 5 (2015), s. 346-352 Registrované v: wos Indikátor časopisu: IF (JCR) [2014-0,272] ADE Vědecké práce v zahraničních nekarentovaných časopisech ADE01 Doležal, Martin (30%) - Jampílek, Josef [UKOEXAF] (30%) - Osička, Zdeněk (5%) - Kuneš, Jiří (10%) - Buchta, Vladimír (20%) - Víchová, Petra (5%): Substituted 5-aroylpyrazine-2-carboxylic acid derivatives: synthesis and biological activity Lit. 21 zázn. In: Il Farmaco. - Vol. 58, No. 11 (2003), s. 1105-1111 ADE02 Jampílek, Josef [UKOEXAF] (25%) - Doležal, Martin (15%) - Kuneš, Jiří (10%) - Buchta, Vladimír (10%) - Silva, Luis (20%) - Kráľová, Katarína [UKOPRCUS] (20%): Quinaldine Derivatives: Preparation and Biological Activity Lit.: 35 zázn. In: Medicinal Chemistry. - Vol. 1, No. 6 (2005), s. 591-599 Ohlasy (25): [o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5120-5130 - SCI [o1] 2008 Prasad, A.K. - Kumar, P. - Dhawan, A. - Chillar, A.K. - Sharma, D. - Parmar, V.S.: Bioorganic and Medicinal Chemistry Letters, Vol. 18, No. 6, 2008, s. 2156-2161 - SCI [o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol. 19, 2008, s. 257-263 - SCI [o1] 2009 Sahidhara, K.V. - Kumar, A. - Bhatia, G. - Khan, M.M. - Khanna, A.K. - Saxena, J.K.: European Journal of Medicinal Chemistry, Vol. 44, No. 4, 2009, s. 1813-1818 - SCI [o1] 2010 Ramli, Y. - Slimani, R. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystalographica Section E-Structure Reports Online, Vol. 66, Part. 4, 2010, s. O992-U3649 - SCI [o1] 2010 Musiol, R. - Serda, M. - Hensel-Bielówska, S. - Polanski, J.: Current Medicinal Chemistry, Vol. 17, No. 18, 2010, s. 1960-1973 - SCI [o1] 2010 Ramli, Y. - Slimani, R. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystalographica Section E-Structure Reports Online, Vol. 66, Part. 7, 2010, s. O1767-U268 - SCI [o1] 2010 Tang, W.J. - Sun, Y.W. - Xu, L.J. - Wang, T.L. - Fan, Q.H. - Lam, K.H. - Chan, A.S.C.: Organic and Biomolecular Chemistry, Vol. 8, No. 15, 2010, s. 3464-3471 - SCI [o1] 2010 Ramli, Y. - Moussaif, A. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystallographica, Section E- Structure Reports Online, Vol. E66, No. 8, 2010, s. o1922-U379 - SCI [o1] 2010 Zhong, Q-D. - Xue, Y-Z. - Yan, H. - Song, X-Q. - Zhong, R-G.: Bioorganic & Medicinal Chemistry Letters, Vol. 20, No. 18, 2010, s. 5532-5535 - SCI [o1] 2011 Ramli, Y. - Moussaif, A. - Zouihri, H. - Bourichi, H. - Essassi, E.M.: Acta Crystallographica Section E: Structure Reports Online, Vol. 67, Part. 6, 2011, s. O1374-NIL_362 - SCI [o1] 2011 Loh, W.S. - Fun, H.K. - Kayarmar, R. - Viveka, S. - Nagaraja, G.K.: Acta Crystallographica Section E: Structure Reports Online, Vol. 67, Part. 2, 2011, s. O405-NIL_990 - SCI
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[o1] 2012 Štefane, B. - Požgan, F. - Sosič, I. - Gobec, S.: Tetrahedron Letters, Vol. 53, Iss. 15, 2012, s. 1964-1967 - SCOPUS [o1] 2012 Ramli, Y. - Zouihri, H. - Azougagh, M. - Moussaif, A. - Essassi, E.M.: Acta Crystallographica Section E: Structure Reports Online, Vol. 68, No. 2, 2012, s. o396 - SCI ; SCOPUS [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS [o3] 2010 Serda, M. - Musiol, R. - Polanski, J.: New thiosemicarbazones based on quinoline scaffold as anticancer iron chelators. In: International Electronic Conference on Synthetic Organic Chemistry, 2010,http://www.sciforum.net/presentation/441 [o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.: Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS [o1] 2012 Armitage M. - Bret G. - Choudary B.M. - Kingswood M. - Loft M. - Moore S. - Smith S. Urquhart M.W.: Organic Process Research & Development, Vol. 16, No. 10, 2012, s. 1626-1634 - SCI ; SCOPUS [o3] 2011 Wang, L.X. - Sheng, J. - Wang, X.H.: Synthesis and crystal structure of 4- (4-bromophenyl)-9)4-chlorophenyl) -2,3,6,7 tetrahydro-6, 6-dimethyl-4H-cyclopenta[b]quinoline-1,8 (5H, 9H)-dione. In: Journal of Xuzhou Normal University(Natural Science Edition), Vol. 29, No. 4, 2011, s. 58-62 [o3] 2011 Chen, G.M. - Wu, Z.B. - Hu, D.Y. - Yang, S. - Bao, W.Y.: Research Progress on Synthesis and Bioactivity of Quinoline and Its Derivative Fine Chemical Intermediates. In: Fine Chemical Intermediates, Vol. 41, No. 2, 2011, s. 6-10 [o1] 2014 Moustafa, A.H. - Said, S.A. - Haikal, A.E.F.Z. - Abu-El-Halawa, R. - Abd-El Kader, R.T.: Nucleosides, Nucleotides and Nucleic Acids, Vol. 33, No. 3, 2014, s. 111-128 - SCOPUS [o1] 2014 Bassyouni, F.A. - Abu-Baker, S.M. - Mahmoud, K. - Moharam, M. - El-Nakkady, S.S. - Rehim, M.A.: RSC Advances, Vol. 4, No. 46, 2014, s. 24131-24141 - SCOPUS [o1] 2014 Vairavelu, L. - Rajendra Prasad, K.J.: Journal of Chemical Sciences, Vol. 126, No. 6, 2014, s. 1893-1902 - SCOPUS [o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.: International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCOPUS [o1] 2015 Liu, Y.A. - Zhang, J.A. - Zhang, L.J. - Zou, X.Z. - Li, N. - Li, Y.: Inorganic Chemistry Communications, Vol. 57, Art. No. 5970, 2015, s. 40-43 - SCOPUS ADE03 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (20%) - Buchta, Vladimír (20%): Antimicrobial evaluation of some arylsulfanylpyrazinecarboxylic acid derivatives Lit. 25 zázn. In: Medicinal Chemistry. - Vol. 3, No. 3 (2007), s. 277-280 ADE04 Vinšová, Jarmila (30%) - Imramovský, Aleš (20%) - Jampílek, Josef [UKOEXAF] (30%) - MonrealFerriz, Juana (10%) - Doležal, Martin (10%): Recent advances on isoniazide derivatives Lit. 85 zázn. In: Anti-Infective Agents in Medicinal Chemistry. - Vol. 7, No. 1 (2008), s. 12-31 ADE05 Musiol, Robert (25%) - Jampílek, Josef [UKOEXAF] (25%) - Podeszwa, Barbara (10%) - Finster, Jacek (%10) - Tabak, Dominik (10%) - Dohnal, Jiří (10%) - Polanski, Jaroslaw (10%): RP-HPLC determination of lipophilicity in series of quinoline derivatives Lit. 52 zázn. In: Central European Journal of Chemistry. - Vol. 7, No. 3 (2009), s. 586-597 ADE06 Kráľová, Katarína [UKOPRCUS] (60%) - Ostrovský, Ivan [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (30%): Metabolomics - useful tool for study of plant responses to abiotic stresses = Metabolomika - uzyteczne narzedzie do oceny wplywu czynników abiotycznych na rosliny Lit.: 150 zázn. In: Ecological Chemistry and Engineering S. - Vol. 19, No. 2 (2012), s. 133-161 Ohlasy (6): [o1] 2013 D'Alessandro, A. - Taamalli, M. - Gevi, F. - Timperio, A.M. - Zolla, L. - Ghnaya, T.: Journal of Proteome Research, Vol. 12, No. 11, 2013, s. 4979-4997 - SCI ; SCOPUS [o3] 2013 Zhong G. - Wang, Y.-Z. - Zhang, J. - Jin, H. - Zhang, J.-Y. - Xiao, Y.: Advances in metabolomics research on genus Panax plants. In: Lishizhen Medicine and Materia Medica Research, Vol. 24, No. 9, 2013, s. 2234-2237 [o1] 2014 Beck, J.J. - Smith, L. - Baig, N.: Phytochemical Analysis, Vol. 25, No. 4, 2014, s. 331-341 - SCI ; SCOPUS [o1] 2014 Boestfleisch, C. - Wagenseil, N.B. - Buhmann, A.K. - Seal, C.E. - Wade, E.M. - Muscolo, A. Papenbrock, J.: AoB Plants, Vol. 13, No. 6, 2014, s. plu046 - SCI
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[o1] 2015 Mishra, A. - Patel, M.K. - Jha, B.: Journal of Functional Foods, Vol. 13, 2015, s. 21-31 SCOPUS [o1] 2014 Turi, C.E. - Axwik, K.E. - Smith, A. - Jones, A.M.P. - Saxena, P.K. - Murch, S.J.: Plant Signaling and Behavior, Vol. 9, No. 4, 2014, Art. No. e28645 - SCI ; SCOPUS ADE07 Černíková, Aneta (25%) - Opatřilová, Radka (25%) - Bobáľ, Pavel (25%) - Jampílek, Josef [UKOEXAF] (25%): Antimicrobial evaluation of some arylsulfanylpyrazinecarboxylic acid derivatives Lit. 38 zázn. In: ADMET & DMPK. - Vol. 2, No. 4 (2014), s. 248-253 ADE08 Malík, Ivan (30%) - Govender, Rodney (10%) - Sedlárová, Eva (10%) - Csöllei, Jozef (10%) - Coffey, Aidan (10%) - O Mahony, Jim (10%) - Stanzel, Lukáš (10%) - Jampílek, Josef [UKOEXAF] (10%): The in vitro investigation ofortho-/meta-/para-alkoxyphenylcarbamic acid esters containing substituted Nphenylpiperazin-1-yl fragment against Mycobacterium tuberculosis H37Ra Lit. 20 zázn. In: Journal of Microbiology, Biotechnology and Food Sciences. - Vol. 3, No. 5 (2014), s. 395-397 ADE09 Malík, Ivan (25%) - Govender, Rodney (25%) - Sedlárová, Eva (10%) - Csöllei, Jozef (10%) - Coffey, Aidan (10%) - O Mahony, Jim (10%) - Jampílek, Josef [UKOEXAF] (10%): The in vitro evaluation of ortho-/meta-/para-alkoxyphenylcarbamic acid esterscontaining 4-(4-fluorophenyl)piperazin-1-yl moiety against Mycobacterium tuberculosis H37Ra Lit. 21 zázn. In: Journal of Microbiology, Biotechnology and Food Sciences. - Vol. 3, No. 6 (2014), s. 491-493 ADE10 Malík, Ivan (30%) - Govender, Rodney (20%) - Sedlárová, Eva (10%) - Csöllei, Jozef (10%) - Coffey, Aidan (10%) - O Mahony, Jim (10%) - Jampílek, Josef [UKOEXAF] (10%): The in vitro evaluation of ortho-/meta-/para-alkoxyphenylcarbamic acid estersbearing 4-(2-fluoro-/2-methylphenyl)piperazin-1-yl moiety against Mycobacterium tuberculosis H37Ra Lit. 27 zázn. In: Journal of Microbiology, Biotechnology and Food Sciences. - Vol. 3, No. 4 (2014), s. 286-288 ADE11 Opatřilová, Radka (50%) - Jampílek, Josef [UKOEXAF] (50%): Rapid Screening of Mupirocin Skin Permeation Modification by Micronized and Nanonized Alaptide Lit. 43 zázn. In: ADMET & DMPK. - Vol. 2, No. 1 (2014), s. 56-62 ADE12 Vaculiková, Eliška (40%) - Plachá, Daniela (20%) - Čech-Barabaszová, Karla (20%) - Jampílek, Josef [UKOEXAF] (20%): Cimetidine Nanoparticles Study Lit. 10 zázn. In: Advanced Science, Engineering and Medicine. - Vol. 6, No. 4 (2014), s. 477-481 ADE13 Černíková, Aneta (60%) - Jampílek, Josef [UKOEXAF] (50%): Permeation of Indomethacin through Skin Using Nanonized Alaptide Lit. 43 zázn. In: ADMET & DMPK. - Vol. 3, No. 4 (2015), s. 344-350 ADF Vědecké práce v domácích nekarentovaných časopisech ADF01 Kráľová, Katarína (60%) - Jampílek, Josef [UKOEXAF] (30%) - Ostrovský, Ivan (10%): Metabolomika vo výskume fytoterapeutík = Metabolomics in research of phytotherapeutics Lit. 43 zázn. In: Česká a slovenská farmacie. - Roč. 61, č. 1-2 (2012), s. 21-25 ADF02 Černíková, Aneta (34%) - Opatřilová, Radka (33%) - Jampílek, Josef [UKOEXAF] (33%): Rapid informative screening of nano-alaptide as potential transdermal permeation enhancer of acetylsalicylic acid and paracetamol Lit. 29 zázn. In: Military Medical Science Letters. - Vol. 83, No. 1 (2014), s. 34-39 ADM Vědecké práce v zahraničních časopisech registrovaných v databázích Web of Science nebo SCOPUS ADM01 Brezovská, Monika (45%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (45%): A review of HPLC methods used for determining the presence of meloxicam Lit. 44 zázn. In: Current Pharmaceutical Analysis. - Vol. 9, No. 1 (2013), s. 69-76 Registrované v: wos, scopus
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Indikátor časopisu: IF (JCR) [2013-0,771] SJR (SCOPUS) [2013-0,275] SNIP (SCOPUS) [2013-0,686] Ohlasy (2): [o1] 2015 Yang, W.J. - Li, J. - Gao, J.H. - Huang, Z.Y. - Tang, C.W.: Current Pharmaceutical Analysis, Vol. 11, No. 3, 2015, s. 172 - SCI [o1] 2015 Sim, A. - Cho, Y. - Kim, D. - Witt, M. - Birdwell, J.E. - Kim, B.J. - Kim, S.: Fuel, Vol. 140, 2015, s. 723 - SCI ADM02 Jampílek, Josef [UKOEXAF] (100%) : Transdermal application of drugs and techniques affecting skin barrier Lit. 45 zázn. In: Journal of Bioequivalence and Bioavailability. - Vol. 5, No. 6 (2013), s. 233-235 Registrované v: scopus Indikátor časopisu: SJR (SCOPUS) [2013-0,163] SNIP (SCOPUS) [2013-0,358] Ohlasy (1): [o1] 2015 Han, T. - Das, D.B.: European Journal of Pharmaceutics and Biopharmaceutics, Vol. 89, 2015, s. 328 - SCOPUS ADM03 Opatřilová, Radka (20%) - Černíková, Aneta (20%) - Coufalová, Lenka (20%) - Dohnal, Jiří (20%) Jampílek, Josef [UKOEXAF] (20%): In Vitro Permeation of Micronized and Nanonized Alaptide from Semisolid Formulations Lit. 45 zázn. In: The Scientific World Journal [elektronický zdroj]. - Vol. 2013, (2013), Art. No. 787283, s. [8 s.] [online] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) [2013-1,219] SJR (SCOPUS) [2013-0,407] SNIP (SCOPUS) [2013-0,578] ADM04 Tengler, Jan (20%) - Kapustíková, Iva (10%) - Peško, Matúš [UKOPREEF] (10%) - Govender, Rodney (10%) - Keltošová, Stanislava (10%) - Mokrý, Petr (5%) - Kollár, Peter (5%) - O Mahony, Jim (5%) Coffey, Aidan (5%) - Kráľová, Katarína [UKOPRCUS](10%) - Jampílek, Josef [UKOEXAF] (10%): Synthesis and Biological Evaluation of 2-Hydroxy-3-[(2-aryloxyethyl)amino]propyl4[(Alkoxycarbonyl)amino]benzoates Lit.: 49 zázn., 3 obr., 1 tab. In: The Scientific World Journal [elektronický zdroj]. - Vol. 2013 (2013), Art. No. 274570 [13 s.] [online] Registrované v: scopus, wos Indikátor časopisu: IF (JCR) [2013-1,219] SJR (SCOPUS) [2013-0,407] SNIP (SCOPUS) [2013-0,578] Ohlasy (2): [o1] 2014 Bado, O. - Frydrych, M. - Kolmanová, E. - Dlouhá, M.: Ceska a Slovenska Farmacie, Vol. 63, No. 4, 2014, s. 167-173 - SCOPUS [o1] 2015 Romano, B. - Plano, D. - Encío, I. - Palop, J.A. - Sanmartín, C.: Bioorganic and Medicinal Chemistry, Vol. 23, No. 8, 2015, s. 1716-1727 - SCOPUS ADM05 Bojňanská, Erika (25%) - Kalina, Michal (10%) - Pařízek, Ladislav (5%) - Bartoníčková, Eva (5%) Opravil, Tomáš (15%) - Veselý, Michal (10%) - Pekař, Miloslav (5%) - Jampílek, Josef [UKOEXAF] (25%): Determination of critical parameters of drug substance influencing dissolution: a case study Lit. 20 zázn. In: BioMed Research International. - Vol. 2014 (2014), Art. No. 929248, s. [9 s.] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) [2014-1,579] SJR (SCOPUS) [2014-0,613] SNIP (SCOPUS) [2014-0,576]
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ADM06 Imramovský, Aleš (30%) - Kozic, Jan (10%) - Peško, Matúš [UKOPREEF] (15%) - Stoláriková, Jirina (10%) - Vinšová, Jarmila (10%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek, Josef [UKOEXAF] (10%): Synthesis and antimycobacterial andphotosynthesis-inhibiting evaluation of 2-[(E)-2-Substitutedethenyl]-1,3-benzoxazoles Lit.: 55 zázn., 4 obr., 1 schéma, 1 tab. In: The Scientific World Journal [elektronický zdroj]. - Vol. 2014 (2014), Art. No. 705973 [11 s.] [online] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) [2014-1,219] SJR (SCOPUS) [2014-0,350] SNIP (SCOPUS) [2014-0,531] ADM07 Vaverková, Veronika (20%) - Vrána, Oldřich (10%) - Adam, Vojtěch (10%) - Pekárek, Tomáš (20%) Jampílek, Josef [UKOEXAF] (20%) - Babula, Petr (20%): The study of naphthoquinones and their complexes with DNA by using Raman spectroscopy and surface enhanced Raman spectroscopy: new insight into interactions of DNA with plant secondary metabolites Lit. 95 zázn. In: BioMed Research International. - Vol. 2014 (2014), Art. No. 461393, s. [12 s.] Registrované v: wos, scopus Indikátor časopisu: IF (JCR) [2014-1,579] SJR (SCOPUS) [2014-0,613] SNIP (SCOPUS) [2014-0,576] Ohlasy (1): [o1] 2016 Gasior-Glogowska, M. - Malek, K. - Zajac, G. - Baranska, M.: Analyst, Vol. 141, No. 1, 2016, s. 296 ADM08 Cieslik, Wioleta (20%) - Spaczynska, Ewelina (10%) - Jampílek, Josef [UKOEXAF] (15%) - Malarz, Katarzyna (10%) - Tabak, Dominik (5%) - Nevin, Eoghan (10%) - O Mahony, Jim (5%) - Coffey, Aidan (5%) - Mrozek-Wilczkiewicz, Anna (5%) - Musiol, Robert(15%): Investigation of the Antimycobacterial Activity of 8-Hydroxyquinolines Lit. 47 zázn. In: Medicinal Chemistry. - Vol. 11, No. 8 (2015), s. 771-779 Registrované v: scopus Indikátor časopisu: IF (JCR) [2014-1,363] SJR (SCOPUS) [2014-0,381] SNIP (SCOPUS) [2014-0,618] ADM09 Jampílek, Josef [UKOEXAF] (18%) - Záruba, Kamil (17%) - Oravec, Michal (18%) - Kuneš, Martin (17%) - Babula, Petr (5%) - Ulbrich, Pavel (5%) - Brezániová, Ingrid (5%) - Opatřilová, Radka (5%) Triska, Jan (5%) - Suchý, Pavel (5%): Preparation of silica nanoparticles loaded with nootropics and their in vivo permeation through blood-brain barrier Lit. 34 zázn. In: BioMed Research International. - Vol. 2015 (2015), Art. No. 812673, s. [9 s.] Registrované v: scopus, wos Indikátor časopisu: IF (JCR) [2014-1,579] SJR ( [2014-0,613] SNIP (SCOPUS) [2014-0,576] ADM10 Kráľová, Katarína [UKOPRCUS] (60%) - Perina, V. (5%) - Waisser, Karel (5%) - Jampílek, Josef [UKOEXAF] (30%): Structure-Activity Relationships of N-benzylsalicylamides for Inhibition of Photosynthetic Electron Transport Lit.: 53 zázn., 3 obr., 1 tab. In: Medicinal Chemistry. - Vol. 11, No. 2 (2015), s. 156-164 Registrované v: wos, scopus Indikátor časopisu: IF (JCR) [2014-1,363] SJR (SCOPUS) [2014-0,381] SNIP (SCOPUS) [2014-0,618]
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ADM11 Zdražilová, Iveta (25%) - Pospíšilová, Šárka (20%) - Pauk, Karel (10%) - Imramovský, Aleš (10%) Vinšová, Jarmila (5%) - Čížek, Alois (10%) - Jampílek, Josef [UKOEXAF] (20%): In vitro bactericidal activity of 4- and5-chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA Lit. 40 zázn. In: BioMed Research International. - Vol. 2015 (2015), s. [8 s.], Art.No. 349534 Registrované v: scopus, wos Indikátor časopisu: IF (JCR) [2014-1,579] SJR ( [2014-0,613] SNIP (SCOPUS) [2014-0,576] AED Vědecké práce v domácích recenzovaných vědeckých sbornících AED01 Jampílek, Josef [UKOEXAF] (50%) - Doležal, Martin (25%) - Deigner, Hans Peter (25%): Optimization of Sphingosine Synthesis by Tkaczuk-Thornton Method Lit. 8 zázn. In: Folia Pharmaceutica Universitatis Carolinae, Roč. 27-28. - Praha : Karolinum, 2002. - S. 69-75 AED02 Jampílek, Josef [UKOEXAF] (50%) - Doležal, Martin (25%) - Kuneš, Jiří (25%): Quinlukast Azaanalogues Preparation Lit. 9 zázn. In: Folia Pharmaceutica Universitatis Carolinae, Roč. 31-32. - Praha : Karolinum, 2004. - S. 27-32 AED03 Doležal, Martin (20%) - Opletalová, Veronika (20%) - Bagi-Krinková, Jana (10%) - Jampílek, Josef [UKOEXAF] (10%) - Kučerová-Chlupáčová, Marta (10%) - Palek, Lukáš (10%) - Kešetovičová, Diana (10%) - Zitko, Jan (10%): Development of New Antituberculous Active Pyrazines Evaluated in Cooperation with TAACF Program within a Perion of 15 years Lit. 20 zázn. In: Folia Pharmaceutica Universitatis Carolinae, Roč. 39. - Praha : Karolinum, 2010. - S. 31-40 BCI Skripta a učební texty BCI01 Jampílek, Josef [UKOEXAF] (80%) - Opatřilová, Radka (10%) - Liška, Ivo (10%): Návody do cvičení z analytické chemie : Vybrané instrumentální metody. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2007. - 74 s. Lit. 13 zázn. ISBN 978-80-7305-007-8 BCI02 Dohnal, Jiří (10%) - Grafnetterová, Taťjana (10%) - Grünwaldová, Veronika (10%) - Havlíček, Jaroslav (10%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (10%) - Pekárek, Tomáš (10%) - Plaček, Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%): Moderní přístupy k farmaceutické analýze : 1. Analýza chirálních léčiv. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2008. - 122 s. Lit. 10 zázn. ISBN 978-80-7305-056-6 BCI03 Liška, Ivo (80%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (10%): Návody do cvičení z analytické chemie : Kvalitativní anorganická analýza. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2008. - 67 s. Lit. 43 zázn. ISBN 978-80-7305-044-3 BCI04 Opatřilová, Radka (80%) - Jampílek, Josef [UKOEXAF] (10%) - Liška, Ivo (10%): Návody do cvičení z analytické chemie : Kvantitativní analýza. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2008. - 82 s. Lit. 21 zázn. ISBN 978-80-7305-027-6 BCI05 Dohnal, Jiří (10%) - Grafnetterová, Taťjana (10%) - Grünwaldová, Veronika (10%) - Havlíček, Jaroslav (10%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (10%) - Pekárek, Tomáš (10%) - Plaček, Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%): Moderní přístupy k farmaceutické analýze : 2. Strukturní analýza léčiv. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2009. - 105 s. Lit. 12 zázn. ISBN 978-80-7305-058-0
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BCI06 Dohnal, Jiří (10%) - Grafnetterová, Taťjana (5%) - Grünwaldová, Veronika (10%) - Havlíček, Jaroslav (10%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (5%) - Pekárek, Tomáš (10%) - Plaček, Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%) - Brusová, Hana (10%): Moderní přístupy k farmaceutické analýze : 3. Farmaceutická analýza v pevné fázi. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2009. - 159 s. Lit. 33 zázn. ISBN 978-80-7305-075-7
Další ukazatele publikační činnosti ve vědeckých časopisech Publikace s IF >1,000 a zároveň z nich jako první nebo korespondující autor Publikace v karentovaných časopisech (ADC, ADD) Součet IF všech vědeckých prací h-index
81 49 84 214 17 (Web of Science – Core Collection; ke dni 5.2.2016) 19 (Web of Science – All Databases; ke dni 5.2.2016)
Práce, které nebyly zařazené do seznamu kontroly AK UK – na základě kritérii VR FaF UK ke splnění podmínek získání vědecko-pedagogického titulu „profesor“ se nevyžadují: AGJ Patenty a přihlášky patentů 1. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and NIEDBALA, Halina and PAŁKA, Anna and PODESZWA, Barbara and POLAŃSKI, Jarosław (Uniwersytet Śląski v Katowicach). Pochodne chinoliny wykazujące aktywność jako herbicydy i algicydy, ich prekursory, sposoby wytwarzania oraz ich stosowanie. P 375678 A1, 13.06.2005. 2. MUSIOŁ, Robert and JAMPÍLEK, Josef and BUCHTA, Vladimír and NIEDBALA, Halina and PAŁKA, Anna and PODESZWA, Barbara and POLAŃSKI, Jarosław (Uniwersytet Śląski v Katowicach). Pochodne chinoliny wykazujące aktywność jako fungicydy oraz ich stosowanie. P 375805, 20.06.2005. 3. SVOBODA, Martin a JAMPÍLEK, Josef a ŠEBEK, Pavel (Zentiva). Farmaceutická kompozice clopidogrel hydrogenbromidu. CZ 298349 B6, 25.07.2007. 4. SVOBODA, Martin a JAMPÍLEK, Josef a KAČÍRKOVÁ, Martina a TOMÁŠEK, Václav a LEHOCKÝ, Mikuláš (Zentiva). Farmaceutická kompozice s obsahem tolterodinu. CZ 298448 B6, 24.08.2007. 5. MUSIOŁ, Robert and JAMPÍLEK, Josef and BUCHTA, Vladimír and KRÁĽOVÁ, Katarína and FINSTER, Jacek and PODESZWA, Barbara and TABAK, Dominik and POLAŃSKI, Jarosław (Uniwersytet Śląski v Katowicach). Analogi chinazoliny jako fungicydy i herbicydy oraz ich zastosowanie. P 379252, 21.03.2006. 6. SVOBODA, Martin and JAMPÍLEK, Josef and KAČÍRKOVÁ, Martina and TOMÁŠEK, Václav and LEHOCKÝ, Mikuláš and HEJTMÁNKOVÁ, Ludmila and VOSÁTKA, Václav (Zentiva). Crystalline Tolterodine Tartarate and a Pharmaceutical Composition Containing the Same. WO/2008/017278 A3, 28.08.2008. 7. KRÁL, Vladimír a JAMPÍLEK, Josef a HAVLÍČEK, Jaroslav a BRUSOVÁ, Hana a PEKÁREK, Tomáš (Zentiva). Lékové formy inhibitorů tyrosinových kináz. PV 2009-8, 13.01.2009. 8. KRÁL, Vladimír a BRUSOVÁ, Hana a HAVLÍČEK, Jaroslav a Tkadlecová, Marcela a JAMPÍLEK, Josef a PEKÁREK, Tomáš (Zentiva). Příprava, stabilizace a využití polymorfů imatinib mesylatu pro vývoj lékových forem. PV 2009-570, 26.08.2009. 9. KRÁL, Vladimír and JAMPÍLEK, Josef and HAVLÍČEK, Jaroslav and BRUSOVÁ, Hana and PEKÁREK, Tomáš (Zentiva). Dosage Forms of Tyrosine Kinase Inhibitors. WO/2010/081443 A2, 22.07.2010. 10. KRÁL, Vladimír and BRUSOVÁ, Hana and JAMPÍLEK, Josef and HAVLÍČEK, Jaroslav and PEKÁREK, Tomáš and TKADLECOVÁ, Marcela (Zentiva). Imatinib Mesylate Polymorphs Generated by Crystallization in Aqueous Inorganic Salt Solutions. WO/2011/023146 A1, 03.03.2011. 11. MUDRA, Petr a POKORNÝ, Vít a PEŠEK, Václav a PONCAR, Pavel a BÁRTA, Jaroslav a ŘEZÁČOVÁ, Anna a JAMPÍLEK, Josef a DOHNAL, Jiří a KRÁL, Vladimír (Zentiva & Ústav organické chemie a biochemie AV ČR). Simulátor trávicího traktu. CZ 302422 B6, 30.03.2011.
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12. KRÁL, Vladimír a OKTÁBEC, Zbyněk a JAMPÍLEK, Josef a BRUSOVÁ, Hana a PEKÁREK, Tomáš a ŘEZÁČOVÁ, Anna a DOHNAL, Jiří (Zentiva). Příprava, stabilizace a využití nových polymorfů imatinib mesylatu pro vývoj lékových forem. PV 2011-228, 19.04.2011. 13. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a ŘEZÁČOVÁ, Anna a OKTÁBEC, Zbyněk a PÁVEK, Petr a KRÁL, Vladimír a DOHNAL, Jiří (VFU Brno). Způsob ovlivnění rozpustnosti alaptidu, ovlivnění jeho prostupu přes membrány a jeho farmaceutické kompozice pro humánní a veterinární aplikace. PV 2011232, 20.04.2011. 14. KRÁL, Vladimír and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and PEKÁREK, Tomáš and PROKSA, Bohumil and DOHNAL, Jiří and MALOVÍKOVÁ, Anna and EBRINGEROVÁ, Anna and ŘEZÁČOVÁ, Anna (Zentiva). Pectin Complexes of Steroids and Pharmaceutical Compositions Based Thereon. WO/2011/063774 A2, 03.06.2011. 15. KRÁL, Vladimír and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and PEKÁREK, Tomáš and PROKSA, Bohumil and DOHNAL, Jiří and MALOVÍKOVÁ, Anna and EBRINGEROVÁ, Anna and ŘEZÁČOVÁ, Anna (Zentiva). Pectin Complexes of Sartans and Pharmaceutical Compositions Based Thereon. WO/2011/063775 A2, 03.06.2011. 16. KRÁL, Vladimír a RAK, Jakub a ZAGORA, Jiří a GRÜNWALDOVÁ, Veronika a ŘEZÁČOVÁ, Anna a JAMPÍLEK, Josef a KŮTKOVÁ, Božena (Zentiva). Příprava, stabilizace a využití nanočástic API pro vývoj moderních lékových forem. PV 2011-353, 13.06.2011. 17. MUDRA, Petr and POKORNÝ, Vít and PEŠEK, Václav and PONCAR, Pavel and BÁRTA, Jaroslav and ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef and DOHNAL, Jiří and KRÁL, Vladimír (Zentiva & Institute of Organic Chemistry and Biochemistry of Academy of Sciences of the Czech Republic). Digestive Tract Simulator. WO/2011/069472 A1, 16.06. 2011. 18. KRÁL, Vladimír a KRÁLOVÁ, Jarmila a FLIEGER, Miroslav a JAMPÍLEK, Josef a ŘEZÁČOVÁ, Anna a DOHNAL, Jiří a OKTÁBEC, Zbyněk a ZÁRUBA, Kamil a GRÜNWALDOVÁ, Veronika a POUČKOVÁ, Pavla a MARTÁSEK, Pavel (Zentiva). Způsob podávání léčiv ve formě nanočástic umožňující průchod hematoencefalickou bariéru. PV 2011-366, 21.06.2011. 19. KRÁL, Vladimír a OKTÁBEC, Zbyněk a JAMPÍLEK, Josef a PEKÁREK, Tomáš a PROKSA, Bohumil a DOHNAL, Jiří a MALOVÍKOVÁ, Anna a EBRINGEROVÁ, Anna a ŘEZÁČOVÁ, Anna (Zentiva). Způsob zvýšení rozpustnosti farmaceuticky aktivních látek a cílený (kontrolovaný) transport do střeva. CZ 302789 B6, 29.09.2011. 20. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující glukokortikoidy. PV 2012-72, 01.02.2012. 21. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a ČERNÍKOVÁ, Aneta a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující antimikrobiální chemoterapeutika. PV 2012-511, 26.07.2012. 22. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and COUFALOVÁ, Lenka and ČERNÍKOVÁ, Aneta and DOHNAL, Jiří (University of Veterinary and Pharmaceutical Sciences Brno). Utilization of Alaptide as Transdermal Penetration Modifier in Pharmaceutical Compositions for Human and Veterinary Applications Containing Anti-Inflammatory Drugs and/or Antimicrobial Chemotherapeutics. WO/2013/020527 A1, 14.02.2013. 23. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující léčiva centrálního a/nebo vegetativního nervového systému a/nebo pohlavní hormony, resp. modulátory genitálního systému. PV 2013-1000, 13.12.2013. 24. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a DOHNAL, Jiří (VFU Brno). Využití (R)-alaptidu jako modifikátoru transdermální penetrace léčiv ve farmaceutických kompozicích pro humánní a veterinární aplikace. PV 2013-1001, 13.12.2013. 25. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ŘEZÁČOVÁ, Anna and OKTÁBEC, Zbyněk and DOHNAL, Jiří (University of Veterinary and Pharmaceutical Sciences Brno). Alaptide: Methods of Effecting its Solubility, Membrane Permeation and Pharmaceutical Compositions for Human and/or Veterinary Applications. WO/2014/019556 A1, 06.02.2014. 26. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a BOBÁĽ, Pavel (VFU Brno). Využití substituovaných analogů alaptidu jako modifikátorů transdermální penetrace ve farmaceutických kompozicích pro humánní a veterinární aplikace. PV 2014-416, 17.06.2014. 27. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a BRYCHTOVÁ, Kateřina a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace
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ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující nesteroidní antiflogistika a/nebo antipyretika-analgetika. CZ 304915 B6, 10.12.2014. AEG Abstrakty vědeckých prací v zahraničních karentovaných časopisech 1. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and RAICH, Ivan. Preparation of 2-(4-{[4(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propanoic acid (VUFB 20615) and 2-methyl-2-(4-{[4(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propanoic acid (VUFB 20623) as potential antileukotrienic agents. Book of Abstracts: The XVIIIth International Symposium on Medicinal Chemistry (ISMC 2004), Copenhagen, Denmark & Malmö, Sweden, August 15-19, 2004, Drug Future 2004, vol. 29, no. Suppl. A, 399. [ISSN 0377-8282, IF2004 = 0.548] 2. JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila. Structurelipophilicity Relationships in Series of Phenolic Moiety Ring-substituted Pyrazinecarboxanilides. Book of Abstracts: The XIXth International Symposium on Medicinal Chemistry (ISMC 2006), Istanbul, Turkey, August 29-September 2, 2006, Drug Future 2006, vol. 31, no. Suppl. A, 51. [ISSN 0377-8282, IF2006 = 0.777] 3. DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila and BUCHTA, Vladimír and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína. Preparation, Antimycobacterial, Antifungal and Photosynthesis-inhibiting Evaluation of Some Anilides of Substituted Pyrazinecarboxylic Acid. Book of Abstracts: The XIXth International Symposium on Medicinal Chemistry (ISMC 2006), Istanbul, Turkey, August 29-September 2, 2006, Drug Future 2006, vol. 31, no. Suppl. A, 53. [ISSN 0377-8282, IF2006 = 0.777] 4. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and MONREAL-FÉRRIZ, Juana and DOLEŽAL, Martin and JAMPÍLEK, Josef. Synthesis, Antituberculotic Activity and Stability of New Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The XIXth International Symposium on Medicinal Chemistry (ISMC 2006), Istanbul, Turkey, August 29-September 2, 2006, Drug Future 2006, vol. 31, no. Suppl. A, 60. [ISSN 0377-8282, IF2006 = 0.777] 5. JAMPÍLEK, Josef and DOLEŽAL, Martin and HOŠŤÁLKOVÁ, Anna and VINŠOVÁ, Jarmila. Structurelipophilicity Relationships in Series of New Substituted N-phenylpyrazine-2-carboxamides as Biologically Active Compounds. Book of Abstracts: The XXth International Symposium on Medicinal Chemistry (ISMC 2008), Vienna, Austria, August 31-September 4, 2008, Drug Future 2008, vol. 33, no. Suppl. A, 60. [ISSN 0377-8282, IF2008 = 0.468] 6. SKÓRSKA-STANIA, Agnieszka and ŚLIWA, Magdalena and OLEKSYN, Barbara and MUSÍLEK, Kamil and KUČA, Kamil and JAMPÍLEK, Josef and MUSIOŁ, Robert and DOHNAL, Jiří. Is It Possible to Guess Potential Drug Activity from Its Crystal Structure? Book of Abstracts: The 25th European Crystallographic Meeting (ECM-25), Istanbul, Turkey, August 16-21, 2009, Acta Cryst. A 2009, vol. A65, no. S., s148 (FA1-MS07-P04). [ISSN 2053-2733, IF2009 = 49.93] 7. DOLEŽAL, Martin and JAMPÍLEK, Josef and ZITKO, Jan and OSIČKA, Zdeněk and SERVUSOVÁ, Barbora. Structure-property Relationships in Series of Chlorine-substituted Pyrazinecarboxanilides as Biologically Active Compounds. Book of Abstracts: The XXIst International Symposium on Medicinal Chemistry (ISMC 2010), Brussels, Belgium, September 5-9, 2010, Drug Future 2010, vol. 35, no. Suppl. A, 76 (PO-60). [ISSN 0377-8282, IF2010 = 0.324] 8. JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and RAICH, Ivan. Preparation and Physico-chemical Properties of Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopiperidin-1yl)hexanoates. Book of Abstracts: The XXIst International Symposium on Medicinal Chemistry (ISMC 2010), Brussels, Belgium, September 5-9, 2010, Drug Future 2010, vol. 35, no. Suppl. A, 77 (PO-61). [ISSN 0377-8282, IF2010 = 0.324] 9. KOS, Jiří and GONĚC, Tomáš and BOBÁL, Pavel and JAMPÍLEK, Josef. Synthesis of Hydroxynaphthalene-2-carboxanilides as Biologically Active Compounds. Book of Abstracts: The XXIInd International Symposium on Medicinal Chemistry (ISMC 2012), Berlin, Germany, September 2-6, 2012, ChemMedChem 2012, vol. 7, no. Suppl. A, 194 (P256). [ISSN 1860-7179, IF2012 = 2.835] 10. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and ČÍŽEK, Alois and JAMPÍLEK, Josef. Bactericidal Activity of (S)-5-Chloro-2hydroxy-N-{3-methyl-1-oxo-1-[4-(trifluoromethyl)phenylamino]butan-2-yl}benzamide against MRSA in Dependence on Time and Concentration. Book of Abstracts: The XXIIIrd International Symposium on Medicinal Chemistry (ISMC 2014), Lisbon, Portugal, September 7-11, 2014, ChemMedChem 2014, vol. 9, no. Suppl. A, 103 (C017). [ISSN 1860-7179, IF2014 = 2.968]
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AEH Abstrakty vědeckých prací v domácích karentovaných časopisech 1. DOLEŽAL, Martin and JAMPÍLEK, Josef and KUTILOVÁ, Helena and KRÁĽOVÁ, Katarína. Synthesis and Biological Evaluation of Anilides Pyrazine-2-carboxylic Acid. Book of Abstracts: The 54th International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4, 2002, Chem. Listy 2002, vol. 96, no. 6, 398. [ISSN 0009-2770, IF2002 = 0.336] 2. DOLEŽAL, Martin and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Inhibition of Photosynthetic Electron Transport in Spinach Chloroplasts by Some Anilides of Pyrazine-2-Carboxylic Acids. Book of Abstracts: The 54th International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4, 2002, Chem. Listy 2002, vol. 96, no. 6, 399. [ISSN 0009-2770, IF2002 = 0.336] 3. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Studies of the Influence of Semiconductor Heterogeneous Catalysts on the Bis(4-methoxyphenyl)disulfide Formation. Book of Abstracts: The 54th International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4, 2002, Chem. Listy 2002, vol. 96, no. 6, 403. [ISSN 0009-2770, IF2002 = 0.336] 4. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří. Aliphatic Iodo Derivatives of Tetrahydrofuran Formation by means of Titanic Heterogeneous Catalyst as By-Products at the Synthesis of 2-Arylpropanoic Acids from Acetophenone Derivatives. Book of Abstracts: LIBLICE 2002 – The 37th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 22-24, 2002, Chem. Listy 2002, vol. 96, no. 11, 932. [ISSN 0009-2770, IF2002 = 0.336] 5. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří. Study of Radical Aroylation of the Pyrazine Nucleus Through Homogeneous Catalysis by Means of Salts of Transition Metals. Book of Abstracts: LIBLICE 2002 – The 37th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 22-24, 2002, Chem. Listy 2002, vol. 96, no. 11, 939. [ISSN 0009-2770, IF2002 = 0.336] 6. JAMPÍLEK, Josef and DOLEŽAL, Martin and HANIKA, Jiří. Double Bond Catalytic Hydrogenation on Palladium Heterogeneous Catalyst in Presence of Sulfanyl Group. Book of Abstracts: The 55th International Conference of Chemical Societies, Košice, Slovakia, September 8-12, 2003, Chem. Listy 2003, vol. 97, no. 9, 757. [ISSN 0009-2770, IF2003 = 0.345] 7. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and RAICH, Ivan. Synthesis of 5- or 6-[(3Methoxyphenyl)sulfanyl]pyrazine-2-carboxylic Acid and 5- or 6-[(4-Methoxyphenyl)sulfanyl]pyrazine-2carboxylic Acid Derivatives. Book of Abstracts: LIBLICE 2003 – The 38th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 28-30, 2003, Chem. Listy 2003, vol. 97, no. 11, 1108. [ISSN 0009-2770, IF2003 = 0.345] 8. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and ŠATÍNSKÝ, Dalibor. Novel Regioselective Preparation of 5-Chloropyrazine-2-carbonitrile from Pyrazine-2-carboxamide. Book of Abstracts: The 56th International Conference of Chemical Societies, Ostrava, Czech Republic, September 69, 2004, Chem. Listy 2004, vol. 98, no. 8, 670. [ISSN 0009-2770, IF2004 = 0.348] 9. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and JUN, Daniel. Preparation and Antiplatelet Activity of Glycidic Acid Derivatives. Book of Abstracts: LIBLICE 2004 – The 39th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 26-28, 2004, Chem. Listy 2004, vol. 98, no. 11, 1015. [ISSN 0009-2770, IF2004 = 0.348] 10. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK, Josef. New Derivatives of Isoniazide and Pyrazinamide. Book of Abstracts: LIBLICE 2005 – The 40th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 18-20, 2005, Chem. Listy 2005, vol. 99, no. 11, 845. [ISSN 0009-2770, IF2005 = 0.445] 11. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and GRAFNETTEROVÁ, Taťjana, and DOHNAL, Jiří. Hydrophobic Properties of Some Antimicrobially Active Esters of Salicylanilides. Book of Abstracts: LIBLICE 2005 – The 40th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 18-20, 2005, Chem. Listy 2005, vol. 99, no. 11, 846. [ISSN 0009-2770, IF2005 = 0.445] 12. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and JAMPÍLEK, Josef. Preparation and Antimycobacterial Activity of Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 58th International Conference of Chemical Societies, Ústí nad Labem, Czech Republic, September 4-8, 2006, Chem. Listy 2006, vol. 100, no. 8, 659. [ISSN 0009-2770, IF2006 = 0.431] 13. JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and DOHNAL, Jiří. Hydrophobic Properties of New Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 58th International Conference of Chemical Societies, Ústí nad Labem, Czech Republic, September 4-8, 2006, Chem. Listy 2006, vol. 100, no. 8, 659-660. [ISSN 0009-2770, IF2006 = 0.431]
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14. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana and DOHNAL, Jiří. Hydrophobic Properties of Substituted Salicylanilide Esters of Amino Acids. Book of Abstracts: LIBLICE 2007 – The 42nd Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 16-18, 2007, Chem. Listy 2007, vol. 101, no. 11, 977. [ISSN 0009-2770, IF2007 = 0.683] 15. DOHNAL, Jiří and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana and VINŠOVÁ, Jarmila. Preparation and Hydrophobic Properties of 5-Chloro-N-[1-(3,4dichlorophenylcarbamoyl)alkyl]-2-hydroxybenzamides. Book of Abstracts: The XXXVIIth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 8-10, 2008, Chem. Listy 2008, vol. 102, no. S, s214. [ISSN 0009-2770, IF2008 = 0.593] 16. DOLEŽEL, Jan and HIRŠOVÁ, Petra and OPLETALOVÁ, Veronika and VEJSOVÁ, Marcela and JAMPÍLEK, Josef. Synthesis and Biological Evaluation of Rhodanine and N-Substituted Rhodanine Derivatives. Book of Abstracts: The XXXVIIth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 8-10, 2008, Chem. Listy 2008, vol. 102, no. S, s215. [ISSN 0009-2770, IF2008 = 0.593] 17. JAMPÍLEK, Josef and MUSIOŁ, Robert and BUCHTA, Vladimír and DOHNAL, Jiří and FINSTER, Jacek and TABAK, Dominik and NIEDBALA, Halina and POLAŃSKI, Jarosław. Preparation and Antifungal Activity of Ring-Substituted 4-Hydroxy-1H-quinolin-2-ones. Book of Abstracts: The XXXVIIth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 8-10, 2008, Chem. Listy 2008, vol. 102, no. S, s222. [ISSN 0009-2770, IF2008 = 0.593] 18. IMRAMOVSKÝ, Aleš a VINŠOVÁ, Jarmila a MONREAL-FÉRRIZ, Juana a JAMPÍLEK, Josef. Decomposition Hydrolytic Study of Hydrazonoformamide Prodrugs of Isoniazide. Book of Abstracts: LIBLICE 2008 – The 43rd Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 14-16, 2008, Chem. Listy 2008, vol. 102, no. 11, 1041. [ISSN 00092770, IF2008 = 0.593] 19. IMRAMOVSKÝ, Aleš and BRITO, Alexandra Maria and PEJCHAL, Vladimír and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef. Syntesis and Antifungal Properties of New 2-Substituted Benzothiazoles. Book of Abstracts: LIBLICE 2010 – The 45th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 20-22, 2010, Chem. Listy 2010, vol. 104, no. 11, 10841085. [ISSN 0009-2770, IF2010 = 0.620] 20. RAICH, Ivan and KÁČEROVÁ, Sandra and JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina. Conformational Analysis of Substituted Alkyl-6-(2,5-dioxopyrrolidin-1-yl)hexanoates: Calculation study. Book of Abstracts: LIBLICE 2010 – The 45th Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 20-22, 2010, Chem. Listy 2010, vol. 104, no. 11, 10871088. [ISSN 0009-2770, IF2010 = 0.620] AFA Publikované vyžádané referáty na zahraničních vědeckých konferencích 1. JAMPÍLEK, Josef and ZADRAŽILOVÁ, Iveta and KOS, Jiří and GONĚC, Tomáš. Design, Synthesis and Anti-staphylococcus Activity of Hydroxynaphthalenecarboxanilides. Proceedings: International ScientificPractical Conference “Pharmaceutical Education, Scientific and Manufacturing as a Reference to the Strategy Kazakhstan-2020”, South Kazakhstan State Pharmaceutical Academy, Shymkent, Kazakhstan, October 23-24, 2014, Republican Scientific Journal 2014, vol. 68, no. 3, 3-7. [ISSN 2306-6822] 2. JAMPÍLEK Josef and KRÁĽOVÁ, Katarína. Applications of nanoformulations in Agricultural Production and Their Potential Impact on Food and Human Health. Proceedings: The 24th Annual Central European Conference (ECOpole’15), Opole – Jarnołtówek, Poland, October 14-17, 2015, Proceedings of ECOpole (PECO-2015), 2015, vol. 9, no. 2, 465-472. [ISSN 1898-617X] AFC Publikované příspěvky na zahraničních vědeckých konferencích 1. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Comparison of Influence of Conductor, Semiconductor and Insulator Copper Heterogeneous Catalysts on Bis(4methoxyphenyl)disulfide Formation. Proceedings: The 6th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-6), September 1-30, 2002, http://www.mdpi.net/ec/papers/ecsoc6/187/jamp2002.htm. Editors: Shu-Kun Lin and Julio A. Seijas, CD-ROM edition. Published in 2002 by MDPI, Basel, Switzerland. [ISBN 3-906980-11-1] 2. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří and KRÁĽOVÁ, Katarína. Substituted Pyrazine-2-carboxamides: Preparation and Their Photosynthesis-inhibiting Activity. Proceedings: The 7th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-7), November 1-30, 2003, http://www.mdpi.net/ec/ec_article.php?id=81&file=papers/ecsoc-7/C001/C001.htm. Editors: Julio A. Seijas, De-Chun Ji and Shu-Kun Lin, CD-ROM edition. Published in 2003 by MDPI, Basel, Switzerland. [ISBN 3-906980-13-8]
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JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and BUCHTA, Vladimír. Quinaldine Derivatives Preparation and Their Antifungal Activity. Proceedings: The 8th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-8), November 1-30, 2004, c005, http://www.usc.es/congresos/ecsoc/8/BOCNP/005/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2004 by MDPI, Basel, Switzerland. [ISBN 3-906980-15-4] JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří. Thiosemicarbazones of Acetylpyrazines: Preparation and Their Hydrophobic Properties. Proceedings: The 9th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005, http://www.usc.es/congresos/ecsoc/9/GOS/a001/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2] JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří. Synthesis and Hydrophobic Properties of Benzoxazoles. Proceedings: The 9th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005, http://www.usc.es/congresos/ecsoc/9/GOS/a008/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2] OPLETALOVÁ, Veronika and JAMPÍLEK, Josef and CHLUPÁČOVÁ, Marta and DOLEŽEL, Jan and GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří. Chromatographic and Computational study of Hydrophobic Properties of Ring Substituted Pyrazinecarbonitriles and Acetylpyrazines. Proceedings: The 9th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005, http://www.usc.es/congresos/ecsoc/9/BOCNP/c004/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2] MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and PODESZWA, Barbara and FINSTER, Jacek and NIEDBALA, Halina and PAŁKA, Anna and POLAŃSKI, Jarosław. New Quinoline Derivatives Possessing Herbicidal Activity. Proceedings: The 9th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005, http://www.usc.es/congresos/ecsoc/9/BOCNP/c005/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2] DOLEŽAL, Martin and ČMEDLOVÁ, Pavlína and PALEK, Lukáš and KUNEŠ, Jiří and BUCHTA, Vladimír and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína. Synthesis and Biological Evaluation of Pyrazinecarboxamides. Proceedings: The 9th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005, http://www.usc.es/congresos/ecsoc/9/BOCNP/c020/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2] JAMPÍLEK, Josef and VINŠOVÁ Jarmila and DOHNAL, Jiří. Synthesis and Hydrophobic Properties of Substituted 2-Aryl-5,7-di-tert-butylbenzoxazoles. Proceedings: The 10th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, a003, http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CDROM edition. Published in 2006 by MDPI, Basel, Switzerland. [ISBN 3-906980-18-9] JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and DOHNAL, Jiří. N,N-Dimethylthiosemicarbazones of Acetylpyrazines: Preparation and Their Hydrophobic Properties. Proceedings: The 10th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, a004, http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CDROM edition. Published in 2006 by MDPI, Basel, Switzerland. [ISBN 3-906980-18-9] JAMPÍLEK, Josef and PALEK, Lukáš and DOLEŽAL, Martin. Synthesis and Hydrophobic Properties of Some Substituted 3-Arylaminopyrazine-2,5-dicarbonitriles. Proceedings: The 10th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, a019, http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CDROM edition. Published in 2006 by MDPI, Basel, Switzerland. [ISBN 3-906980-18-9] MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and TABAK, Dominik and PODESZWA, Barbara and FINSTER, Jacek and POLAŃSKI, Jarosław. Substituted Amides of Quinoline Derivatives: Preparation and Their Photosynthesis-inhibiting Activity. Proceedings: The 10th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, c007, http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CDROM edition. Published in 2006 by MDPI, Basel, Switzerland. [ISBN 3-906980-18-9] JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and KADEŘÁVKOVÁ, Zuzana and DOHNAL, Jiří. Synthesis and Hydrophobic Properties of New 2-Aryl-5,7-di-tert-butylbenzoxazoles. Proceedings: The 11th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-11), November 1-30, 2007, a009, http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a009/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland. [ISBN 3-906980-19-7]
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14. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and TABAK, Dominik and FINSTER, Jacek and PODESZWA, Barbara and KOZIK, Violetta and DOHNAL, Jiří and POLAŃSKI, Jarosław. Preparation and Herbicidal Activities of Substituted Amides of Quinoline Derivatives. Proceedings: The 11th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-11), November 1-30, 2007, a011, http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a011/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland. [ISBN 3-90698019-7] 15. JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and DOLEZEL, Jan and DOHNAL, Jiří. Preparation and Hydrophobic Properties of 5-Arylalkylidenerhodanines. Proceedings: The 11th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-11), November 1-30, 2007, a012, http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a012/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland. [ISBN 3-906980-19-7] 16. DOLEŽAL, Martin and JAMPÍLEK, Josef and BIELESZ, Stanislav and KUNEŠ, Jiří. Substituted pyrazine-2,5-dicarboxamides: Synthesis, Hydrophobicity Parameters, and Antimycobacterial Evaluation. Proceedings: The 11th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-11), November 1-30, 2007, c005, http://www.usc.es/congresos/ecsoc/11/hall_cBCNP/c005/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland. [ISBN 3-906980-19-7] 17. DOLEŽAL, Martin and and LEŠŇANSKÁ, Katarína and PEŠKO, Matúš and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína. Pyrazinecarboxamides, Their Synthesis and Evaluation as Potential Herbicides. Proceedings: The 12th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-12), November 1-30, 2008, c0004, http://www.usc.es/congresos/ecsoc/12/ECSOC12.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2008 by MDPI, Basel, Switzerland. [ISBN 3-906980-20-0] 18. OPLETALOVÁ, Veronika and JAMPÍLEK, Josef and DOLEŽEL, Jan and HIRŠOVÁ, Petra and DOHNAL, Jiří. Rhodanineacetic Acid Derivatives as Potential Drugs: Preparation and Hydrophobic Properties of 5-Arylalkylidene-3-carboxymethylrhodanines. Proceedings: The 12th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-12), November 1-30, 2008, c0006, http://www.usc.es/congresos/ecsoc/12/ECSOC12.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CDROM edition. Published in 2008 by MDPI, Basel, Switzerland. [ISBN 3-906980-20-0] 19. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and FINSTER, Jacek and TABAK, Dominik and NIEDBALA, Halina and CSOLLEI, Jozef and DOHNAL, Jiří and POLAŃSKI, Jarosław. Ring-substituted 4-Hydroxy-1H-quinolin-2-ones: Preparation and Their Photosynthesis-inhibiting Activity. Proceedings: The 12th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-12), November 1-30, 2008, c0012, http://www.usc.es/congresos/ecsoc/12/ECSOC12.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2008 by MDPI, Basel, Switzerland. [ISBN 3-906980-20-0] 20. JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and ŘEZÁČOVÁ, Anna and PLAČEK, Lukáš and KOS, Jiří and HAVELKOVÁ, Lenka and DOHNAL, Jiří and KRÁL Vladimír. Preparation and Properties of New Co-crystals of Ibandronate. Proceedings: The 13th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-13), November 1-30, 2009, c001, http://www.sciforum.net/presentation/201. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2009 by MDPI, Basel, Switzerland. [ISBN 3-906980-23-5] 21. MUSIOŁ, Robert and JAMPÍLEK, Josef and PEŠKO, Matúš and CARROLL, James and KRÁĽOVÁ, Katarína and FINSTER, Jacek and O'MAHONY, Jim and COFFEY, Aidan and POLAŃSKI, Jarosław. Substituted 2-Styrylquinazoline Derivatives: Preparation and Their Biological Activities. Proceedings: The 13th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-13), November 1-30, 2009, c004, http://www.sciforum.net/presentation/204. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2009 by MDPI, Basel, Switzerland. [ISBN 3-906980-23-5] 22. BRYCHTOVÁ, Kateřina and DITTRICHOVÁ, Sylva and SLABÁ, Barbora and PLAČEK, Lukáš and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef and CSÖLLEI, Jozef. Synthesis of Esters of 6-(2,5Dioxopyrrolidin-1-yl)-2-(morpholin-4-yl)hexanoic Acid as Potential Transdermal Penetration Enhancers. Proceedings: The 13th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-13), November 1-30, 2009, c010, http://www.sciforum.net/presentation/210. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2009 by MDPI, Basel, Switzerland. [ISBN 3-906980-23-5] 23. BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and PLAČEK, Lukáš and JAMPÍLEK, Josef and CSÖLLEI, Jozef. Synthesis of Esters of 6-(2,5-Dioxopyrrolidin-1-yl)-2-(2-oxoazepan-1-yl)hexanoic Acid as Potential Transdermal Penetration Enhancers. Proceedings: The 14th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, A417,
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http://www.sciforum.net/conference/ecsoc-14/paper/417. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2010 by MDPI, Basel, Switzerland. [ISBN 3-906980-24-3] JAMPÍLEK, Josef and KOS, Jiří and OKTÁBEC, Zbyněk and MANDELOVÁ, Zuzana and PEKÁREK, Tomáš and TKADLECOVÁ, Marcela and HAVLÍČEK, Jaroslav and DOHNAL, Jiří and KRÁL Vladimír.. Co-crystal Screening Study of Risedronate and Unsubstituted Hexoses. Proceedings: The 14th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, A421, http://www.sciforum.net/conference/ecsoc-14/paper/421. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2010 by MDPI, Basel, Switzerland. [ISBN 3-906980-24-3] IMRAMOVSKÝ, Aleš and JAMPÍLEK, Josef and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and MONREAL-FÉRRIZ, Juana and VINŠOVÁ, Jarmila. Preliminary Study of Photosynthesis-Inhibiting Activity of Substituted Phenylcarbamoylphenyl N-alkylcarbamates. Proceedings: The 14th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, B375, http://www.sciforum.net/conference/ecsoc-14/paper/375. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2010 by MDPI, Basel, Switzerland. [ISBN 3-906980-24-3] DOLEŽAL, Martin and OSIČKA, Zdeněk and ZITKO, Jan and KUNEŠ, Jiří and JAMPÍLEK, Josef and VEJSOVÁ, Marcela and BUCHTA Vladimír and KRÁĽOVÁ, Katarína. Substituted N-phenylpyrazine-2carboxamides, Their Synthesis, Hydro-lipophilic Properties and Evaluation of Their Antimycobacterial, Antifungal and Photosynthesis-inhibiting Activity. Proceedings: The 14th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, B380, http://www.sciforum.net/conference/ecsoc-14/paper/380. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2010 by MDPI, Basel, Switzerland. [ISBN 3-906980-24-3] ŽELAZKOVÁ, Jana and JAMPÍLEK, Josef. Total Synthesis of Arctigenin Derivatives as Potential Anticancer Agents. Proceedings: The 15th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-15), November 1-30, 2011, A598, http://www.sciforum.net/conference/ecsoc15/paper/598. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2011 by MDPI, Basel, Switzerland. [ISBN 3-906980-25-1] MUSIOŁ, Robert and JAMPÍLEK, Josef and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and KOWALCZYK, Wioleta and FINSTER, Jacek and POLAŃSKI, Jarosław. Preparation and Herbicidal Properties of Ring-Substituted 4-Chloro-2-styrylquinazolines. Proceedings: The 15th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-15), November 1-30, 2011, B586, http://www.sciforum.net/conference/ecsoc-15/paper/586. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2011 by MDPI, Basel, Switzerland. [ISBN 3-906980-25-1] ŠUJAN, Josef and PEŠKO, Matúš and GONĚC, Tomáš and KOS, Jiří and BOBÁĽ, Pavel and IMRAMOVSKÝ, Aleš and PLAČEK, Lukáš and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Herbicidal Properties of Substituted Quinoline-2-carboxanilides. Proceedings: The 15th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-15), November 1-30, 2011, B588, http://www.sciforum.net/conference/ecsoc-15/paper/588. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2011 by MDPI, Basel, Switzerland. [ISBN 3-90698025-1] ŠUJAN, Josef and OTEVŘEL, Jan and IMRAMOVSKÝ, Aleš and JAMPÍLEK, Josef and BOBÁĽ, Pavel. Microwave-assisted synthesis of new substituted anilides of quinaldic acid. Proceedings: The 15th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-15), November 1-30, 2011, C681, http://www.sciforum.net/conference/ecsoc-15/paper/681. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2011 by MDPI, Basel, Switzerland. [ISBN 3-90698025-1] VACULÍKOVÁ, Eliška and GRÜNWALDOVÁ, Veronika and KRÁL, Vladimir and DOHNAL, Jiří and JAMPÍLEK, Josef. Preparation of Candesartan Cilexetil Nanoparticles by Precipitation. Proceedings: The 16th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-16), November 1-30, 2012, B1008, http://www.sciforum.net/conference/ecsoc-16/paper/1008. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2013 by MDPI, Basel, Switzerland. [ISBN 3906980-26-X] KOS, Jiří and ZADRAŽILOVÁ, Iveta and PEŠKO, Matúš and PAVLICA, Jiří and GONĚC, Tomáš and BOBÁL, Pavel and ORAVEC, Michal and ČÍŽEK, Alois and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Biological Properties of Ring-Substituted 3-Hydroxynaphthalene-2-carboxanilides. Proceedings: The 16th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-16), November 1-30, 2012, B1009, http://www.sciforum.net/conference/ecsoc-16/paper/1009. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2013 by MDPI, Basel, Switzerland. [ISBN 3-906980-26-X]
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33. ZADRAŽILOVÁ, Iveta and PAUK, Karel and IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and MASAŘÍKOVÁ, Martina and ČÍŽEK, Alois and JAMPÍLEK, Josef. 2-Hydroxy-N-[1-(2hydroxyphenylamino)-1-oxoalkan-2-yl]benzamides – Potential drugs of MRSA infections? Proceedings: The International Student Scientific Conference of Faculty of Natural Sciences of Comenius University 2013, Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 24, 2013, p. 857-862. [ISBN 978-80-223-3392-4] 34. KOS, Jiří and GONĚC, Tomáš and TENGLER, Jan and ZADRAŽILOVÁ, Iveta and PEŠKO, Matúš and ORAVEC, Michal and KRÁĽOVÁ, Katarína and ČÍŽEK, Alois and JAMPÍLEK, Josef: Synthesis of amides of hydroxynaphthoic acids as biologically active compounds. Proceedings: The International Student Scientific Conference of Faculty of Natural Sciences of Comenius University 2013, Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 24, 2013, p. 1044-1047. [ISBN 978-80223-3392-4] 35. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Preparation of atorvastatin nanoparticles by solvent evaporation method. Proceedings: The International Student Scientific Conference of Faculty of Natural Sciences of Comenius University 2013, Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 24, 2013, p. 1199-1204. [ISBN 978-80-223-3392-4] 36. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISÁRČIK Martin and JAMPÍLEK, Josef. Preparation of Risedronate Nanoparticles Using Selected Polymeric Excipients. Proceedings: The 17th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-17), November 1-30, 2013, B012, http://sciforum.net/conference/ecsoc-17/paper/2256. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, ShuKun Lin, CD-ROM edition. Published in 2014 by MDPI, Basel, Switzerland. [ISBN 3-906980-46-0] 37. KOS, Jiří and MACHALOVÁ, Petra and PEŠKO, Matúš and GONĚC, Tomáš and BOBÁL, Pavel and ORAVEC, Michal and LIPTAJ, Tibor and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Herbicidal Activity of Halogenated 8-Hydroxyquinoline-2-carboxanilides. Proceedings: The 17th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-17), November 1-30, 2013, B013, http://sciforum.net/conference/ecsoc-17/paper/2261. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2014 by MDPI, Basel, Switzerland. [ISBN 3-906980-46-0] 38. GONĚC, Tomáš and KOS, Jiří and ŠORAL, Michal and PEŠKO, Matúš and ORAVEC, Michal and LIPTAJ, Tibor and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and PhotosynthesisInhibiting Activity of N-(n-Alkoxy)phenylamides of 2-Hydroxynaphthalene-1-carboxylic acid. Proceedings: The 18th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-18), November 1-30, 2014, b010, http://www.sciforum.net/conference/ecsoc-18/paper/2538. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2015 by MDPI, Basel, Switzerland. [ISBN 978-3-906980-55-3] 39. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISÁRČIK Martin and JAMPÍLEK, Josef. Preparation of Glibenclamide Nanoparticles. Proceedings: The 18th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-18), November 1-30, 2014, b025, http://www.sciforum.net/conference/ecsoc18/paper/2573. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2015 by MDPI, Basel, Switzerland. [ISBN 978-3-906980-55-3] 40. GONĚC, Tomáš and STRÁNÍK, Josef and PEŠKO, Matúš and KOS, Jiří and ORAVEC, Michal and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Photosynthesis-Inhibiting Activity of 1-[(2Chlorophenyl)carbamoyl]naphthalen-2-yl Alkylcarbamates. Proceedings: The 19th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-19), November 1-30, 2015, b006, http://sciforum.net/conference/80/paper/3079. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2016 by MDPI, Basel, Switzerland. [ISBN 978-3-03842-145-0] 41. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISÁRČIK Martin and JAMPÍLEK, Josef. Preparation of Hydrochlorothiazide Nanoparticles. Proceedings: The 19th International Electronic Conference on Synthetic Organic Chemistry (ECSOC-19), November 1-30, 2015, b007, http://sciforum.net/conference/80/paper/3080. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2016 by MDPI, Basel, Switzerland. [ISBN 978-3-03842-145-0] AFD Publikované příspěvky na domácích vědeckých konferencích 1. ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro Antimicrobial Screening of N-(n-Alkoxy)phenylanilides of 2-Hydroxynaphthalene-1-carboxylic acid. Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and Pharmaceutical Sciences Brno, Brno, Czech Republic, October 2, 2014, p. 85-88. [ISBN 78-80-7305-740-4] 2. ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Rapid Screening of Rutin Skin Permeation. Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and Pharmaceutical Sciences Brno, Brno, Czech Republic, October 2, 2014, p. 94-98. [ISBN 78-80-7305-740-4]
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VACULÍKOVÁ, Eliška and JAMPÍLEK, Josef. Preparation of Glibenclamide Nanoparticles via Solvent Evaporation. Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and Pharmaceutical Sciences Brno, Brno, Czech Republic, October 2, 2014, p. 99-102. [ISBN 78-80-7305-740-4]
AFE Abstrakty vyžádaných referátů ze zahraničních konferencí 1. JAMPÍLEK, Josef. Advances in Investigation of Hydrophilic and Lipophilic Properties of Drugs. Book of Abstracts: The XXXVth Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, May 30 - June 1, 2012, OS-5. 2. JAMPÍLEK, Josef. Pharmaceutical nanoparticles and methods of their characterization. Book of Abstracts: The XXXVIth Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, June 5-7, 2013, OS-19. 3. JAMPÍLEK, Josef and MUSIOŁ, Robert and KOS, Jiří and GONĚC, Tomáš and BOBÁL, Pavel and POLAŃSKI, Jarosław. Design and Antimicrobial Screening of New Ring-Substituted Quinoline Analogues. Book of Abstracts: The BIT′s 4th Annual International Congress of Medichem 2013 (ICM2013), Haikou, China, November 13-16, 2013, p. 62. 4. JAMPÍLEK, Josef and COUFALOVÁ, Lenka and MRÓZEK, Lech. Investigation of Cholic Acid Derivatives as Transdermal Permeation Enhancers. Book of Abstracts: The XXXVIIth Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, June 11-14, 2014, OS-18. 5. JAMPÍLEK, Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and HRUBÁ, Michaela and MORAVCOVÁ, Marie and ŠTUJBER, Michal and LIPTAJ, Tibor. Synthesis and Antimicrobial Activity of Hydroxy(aza)naphthalenecarboxamides. Book of Abstracts: The 7th Central European Conference "Chemistry towards Biology", Katowice, Poland, September 9-12, 2014, p. O5. 6. JAMPÍLEK, Josef and CLEMENTS, Carol and KOS, Jiří and GONĚC, Tomáš and GRAY, Alexander I. Synthesis and In Vitro Anti-trypanosomal Screening of Hydroxynaphthalene-2-carboxanilides. Book of Abstracts: The VIth Conversatory on Medicinal Chemistry, Lublin, Poland, September 18-20, 2014, p. 24 (K5). [ISSN 978-83-63657-38-3] 7. JAMPÍLEK, Josef. Recent Advances in Design of Potential Quinoxaline Anti-Infectives. Book of Abstracts: The BIT′s 5th Annual International Congress of Medichem 2014 (ICM-2014), Suzhou, China, November 18-20, 2014, p. 197. 8. JAMPÍLEK, Josef. Azanaphthalenes as Potential Antimycobacterial Agents. Book of Abstracts: The 13th Ibn Sina International Conference on Pure and Applied Heterocyclic Chemistry, Hurghada, Egypt, February 14-17, 2015, p. 8 (PL-06). 9. ORAVEC, Michal and JAMPÍLEK, Josef. Determination of Drugs Loaded to Silica Nanoparticles in Brain Tissue. Book of Abstracts: The XXXVIIIth Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, May 27-29, 2015, OS-27. 10. JAMPÍLEK, Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta. Advances in Design of Potential Quinoline Antimycobacterial Agents. Book of Abstracts: The IXth Joint Meeting in Medicinal Chemistry (JMMC 2015), Athens, Greece, June 7-10, 2015, O6. 11. JAMPÍLEK, Josef and ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel. Design, Synthesis and Investigation of Aryl Derivatives of Alaptide as Potential Transdermal Permeation Enhancers. Book of Abstract: European Pharma Congress “Pharma Europe-2015”, Valencia, Spain, August 25-27, 2015, J. Pharma. Care Health Sys. 2015, vol. 2, no. 4, 63. [ISSN 2376-0419] 12. JAMPÍLEK Josef and ČERNÍKOVÁ, Aneta and TABIOVÁ, Katarína and BOBÁĽ, Pavel. In Vitro Evaluation of 8-Substituted 6,9-diazaspiro[4.5]decan-7,10-diones as Skin Permeation Modifiers. Book of Abstracts: The 4th World Conference on Physico-Chemical Methods in Drug Discovery and Development (PCMDDD-4), Rovinj – Red Island, Croatia, September 21-24, 2015, p. 10 (OP 08). 13. JAMPÍLEK Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and BOBÁĽ, Pavel. Design and Antimicrobial Activity of Ring-Substituted Hydroxynaphthalenecarboxamides and Their AzaAnalogues. Book of Abstracts: The BIT's 13th Annual World Congress of International Drug Discovery Science & Technology 2015 (IDDST 2015), Beijing, China, October 20-22, 2015, p. 109. 14. JAMPÍLEK Josef and ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel and DOHNAL, Jiří. Investigation of Alkyl Derivatives of Alaptide as Transdermal Permeation Modifier. Book of Abstracts: The BIT's 5th Annual World Symposium of Drug Delivery System 2015 (SDDS-2015), Beijing, China, October 20-22, 2015, p. 387.
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AFF Abstrakty vyžádaných referátů z domácích konferencí 1. JAMPÍLEK, Josef. Perspectives of nanoparticles in pharmacy. Book of Abstracts: The 1st International Symposium and Workshop on Environment and Health (ISEH 2012), Ostrava, Czech Republic, November 22-23, 2012, p. 44. [ISBN 978-80-248-2882-4] 2. JAMPÍLEK, Josef. Polymorphism and Its Influence to Biovailability. Book of Abstracts: The 2nd International Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech Republic, November 6-8, 2013, p. 20-21. [ISBN 978-80-248-3240-1] 3. JAMPÍLEK, Josef. Overcoming Blood-Brain Barrier Using Nanoparticles. Book of Abstracts: The 4th Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava, Czech Republic, May 18-21, 2015, p. 63. [ISBN 978-80-248-3745-1] 4. JAMPÍLEK, Josef. Nanoformulations of Antimicrobial Chemotherapeutics. Book of Abstracts: The International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering (NDDTE'16), Prague, Czech Republic, April 1-2, 2016, Keynote-2, http://nddte.com/paper/Keynote%20%20Dr.%20Jampilek.pdf. AFG Abstrakty příspěvků ze zahraničních konferencí 1. JAMPÍLEK, Josef and DOLEŽAL, Martin. Preparation and Biological Evaluation of 5-Aroylpyrazine-2carboxylic Acid Derivatives. Book of Abstracts: The 1st International Student Scientific Conference of Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 25-26, 2001, p. Po-2. 2. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Bis(4-methoxyphenyl)disulfide Preparation by Means of Copper Catalysts. Book of Abstracts: The 53th International Conference of Chemical Societies, Banská Bystrica, Slovakia, September 3-6, 2001, p. 268-269. 3. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Comparison of Effect of Semiconductor and Insulator Copper Heterogeneous Catalysts on Bis(4-methoxyphenyl)disulfide Formation. Book of Abstracts: The International Conference on Organic Synthesis “Balticum Organicum Syntheticum” (BOS 2002), Vilnius, Lithuania, June 23-27, 2002, p. 79. [ISBN 9986-19-485-7] 4. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and OSIČKA, Zdeněk. Preparation of Thiazol2-ylamide, or Pyrid-2-ylamide Pyrazine-2-carboxylic Acid Derivatives. Book of Abstracts: The XXXIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 11-13, 2002, p. 60. 5. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUCHAŘ, Miroslav. Synthesis of 2-Methyl-3-(4-{[4(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propionic Acid (VUFB 20584) as a Potential Antileukotrienic. Book of Abstracts: The 1st International SPECS and BioSPECS Symposium on The New Chemistries, Delft, the Netherlands, September 18-21, 2002, p. 98. 6. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří. Synthesis of (2E)-2-methyl-3-(4-{[4(quinolin-2-ylmethoxy)phenyl]sulphanyl}phenyl)acrylic Acid (VUFB 20609) as a Potential Antileukotrienic Agent. Book of Abstracts: The 9th European Symposium on Organic Reactivity (ESOR IX), Oslo, Norway, July 12-17, 2003, p.153. 7. JAMPÍLEK, Josef and DOLEŽAL, Martin and RAICH, Ivan and LIŠKA, František. 4-Substituted Aryland 6-Substituted Heteroarylhalides Coupling with 4-Methoxybenzenethiol by Means of Copper Heterogeneous Catalysts. Book of Abstracts: The 9th European Symposium on Organic Reactivity (ESOR IX), Oslo, Norway, July 12-17, 2003, p. 169. 8. JAMPÍLEK, Josef and CHLUPÁČOVÁ, Marta and DOLEŽAL, Martin and KRÁĽOVÁ, Katarína: Quinaldine Derivatives and Their Herbicidal Activities. Book of Abstracts: The International Conference “Jahrestagung – Joint Meeting 2004”, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, Germany, October 6-9, 2004, p. 111 (P-C63). [ISBN 3-00-014723-3] 9. JAMPÍLEK, Josef and DOLEŽAL, Martin and BROJEROVÁ Eliška and OPLETAL, Lubomír and JUN, Daniel. Substituted Diarylsulfides and Their Antiplatelet Activity. Book of Abstracts: The International Conference “The 4th Joint Meeting on Medicinal Chemistry 2005” (JMMC 2005), Vienna, Austria, June 2023, 2005, Sci. Pharm. 2005, vol. 73, no. 2 Suppl. 1, 83. [ISSN 0036-8709] 10. VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and BUCHTA, Vladimír and DOLEŽAL, Martin and JAMPÍLEK, Josef. Biodegradable Esters of Salicylanilides with Significant Antimicrobial Activity. Book of Abstracts: The 14th European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 258. [ISBN 952-10-2553-0] 11. JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš. Radical Aroylation of Pyrazine-2carboxylic Acid Derivatives. Book of Abstracts: The 14th European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 272. [ISBN 952-10-2553-0] 12. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK, Josef and DOLEŽAL, Martin. New Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 14th
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European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 295. [ISBN 952-10-2553-0] DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila and BUCHTA, Vladimír and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína. Substituted Amides of Pyrazinoic Acid, Synthesis and Biological Evaluation. Book of Abstracts: The 14th European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 350. [ISBN 952-10-2553-0] DOLEŽAL, Martin and BRUNER, Rudolf and BUCHTA, Vladimír and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína: Amides of Pyrazin-2-carboxylic acid: Synthesis, Antifungal Evaluation and Their Photosynthesis Inhibition. Book of Abstracts: The 57th International Conference of Chemical Societies, Tatranské Matliare, Slovakia, September 4-8, 2005, ChemZi 2005, vol. 1, no. 1, 206. [ISSN 1336-7242] JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš. Preparation and Antimycobacterial Activity of Pyrazine-2-carboxylic Acid Thiazol-2-ylamide Derivatives. Book of Abstracts: The International Conference “Frontiers in Medicinal Chemistry”, Frankfurt am Main, Germany, March 12-15, 2006, p. 90. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and DOLEŽAL, Martin and DOHNAL, Jiří. RP-HPLC Method for Determination of Isoniazide Prodrugs. Book of Abstracts: The International Conference “Drug Analysis 2006”, Namur, Belgium, May 16-19, 2006, PE-09. PALEK, Lukáš and JAMPÍLEK, Josef and DOLEŽAL, Martin. RP-HPLC Assay and Hydrophobic Properties of Novel Pyrazinamide Derivatives. Book of Abstracts: The International Conference “Drug Analysis 2006”, Namur, Belgium, May 16-19, 2006, PK-28. MUSIOŁ, Robert and JAMPÍLEK, Josef and PODESZWA, Barbara and FINSTER, Jacek and TABAK, Dominik and POLAŃSKI, Jarosław. Structure-lipophilicity Relationships in Series of Quinoline Derivatives. Book of Abstracts: The 18th International Conference on Physical Organic Chemistry (ICPOC-18), Warsaw, Poland, August 20-25, 2006, p. 76. [ISBN 83-89585-11-1] JAMPÍLEK, Josef and OPLETALOVÁ, Veronika, and POUR, Milan and KUNEŠ, Jiří and SILVA, Luís and BUCHTA, Vladimír and RICHARDSON, Des Robert and KALINOWSKI, Danuta and AL-HALLAK, Linda and HONCOVÁ, Dana. N,N-Dimethylthiosemicarbazones of Acetylpyrazines as Potential Drugs. Book of Abstracts: The International Conference “Joint Meeting of the Czech, German and Hungarian Pharmaceutical Societies”, Marburg, Germany, October 4-7, 2006, p. 122 (C076). [ISBN 3-89703-685-1] DOLEŽAL, Martin and MONKS, Kathryn and PLAŠOVÁ, Petra and VINŠOVÁ, Jarmila and JAMPÍLEK, Josef and SVOBODOVÁ, Michaela and BUCHTA, Vladimír. Synthesis, Antifungal and Antimycobacterial Properties of Pyrazine Analogues. Book of Abstracts: The International Conference “The 5th Joint Meeting on Medicinal Chemistry 2007” (JMMC 2007), Portorož, Slovenia, June 17-21, 2007, Farmacevtski vestnik 2007, vol. 58, no. Suppl. 1, 85 (PO031). [ISSN 0014-8229] JAMPÍLEK, Josef and DOLEŽAL, Martin and VINŠOVÁ, Jarmila. Structure-lipophilicity Relationships in Series of Methyl Moiety Ring-substituted Pyrazinecarboxanilides as New Antituberculotics. Book of Abstracts: The International Conference “The 5th Joint Meeting on Medicinal Chemistry 2007” (JMMC 2007), Portorož, Slovenia, June 17-21, 2007, Farmacevtski vestnik 2007, vol. 58, no. Suppl. 1, 112 (PO059). [ISSN 0014-8229] JAMPÍLEK, Josef and MUSIOŁ, Robert and BUCHTA, Vladimír and PODESZWA, Barbara and FINSTER, Jacek and NIEDBALA, Halina and PAŁKA, Anna and POLAŃSKI, Jarosław. Preparation and Antifungal Activity of 8-Hydroxyquinoline Derivatives. Book of Abstracts: The 8th Tetrahedron Symposium “50th Anniversary Meeting – Challenges in Organic Chemistry”, Berlin, Germany, June 27-29, 2007, P2.1. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana and DOHNAL, Jiří. Hydrophobic Properties of Some Novel Esters of Salicylanilides. Book of Abstracts: The 59th International Conference of Chemical Societies, Tatranské Matliare, Slovakia, September 2-6, 2007, ChemZi 2007, vol. 3, no. 1, 212. [ISSN 1336-7242] PETRIK, Pavel and VEJSOVÁ, Marcela and KUNEŠ, Jiří and JAMPÍLEK, Josef and ŠPANINGEROVÁ, Eliška and KEŠETOVIČOVÁ, Diana and VLČKOVÁ, Martina and MAJD, Morid and KALAFUTOVÁ, Stanislava and OPLETALOVÁ, Veronika. Antifungal and Antimycobacterial Properties of 5Arylmethylidenerhodanines and Their N3-Substituted Analogues. Book of Abstracts: The 5th International Postgraduate Research Symposium on Pharmaceutics (IPORSIP-2007), Istanbul, Turkey, September 1315, 2007, Acta Pharm. Sci. 2007, 49 (Suppl.), 77. [ISSN 1300-638X] JAMPÍLEK, Josef and DOLEŽAL, Martin and BIELESZ, Stanislav and VINŠOVÁ, Jarmila. RP-HPLC Determination of Hydrophobic Properties of New Pyrazindicarboxamide Derivatives. Book of Abstracts: The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA 2007), Island of Elba, Italy, September 23-26, p. 96.
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26. DOHNAL, Jiří and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and REČKOVÁ, Zuzana and VINŠOVÁ, Jarmila. Stability Study of Pyrazinamide Prodrugs as New Effective Antituberculotics. Book of Abstracts: The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA 2007), Island of Elba, Italy, September 23-26, p. 97. 27. REČKOVÁ, Zuzana and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and DOHNAL, Jiří. Stability Study of Isoniazid Prodrugs as New Effective Antituberculotics. Book of Abstracts: The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA 2007), Island of Elba, Italy, September 23-26, p. 98. 28. JAMPÍLEK, Josef and PEKÁREK, Tomáš and ZERZAŇOVÁ, Anna and MATĚJKA, Pavel and HAVLÍČEK, Jaroslav and BRUSOVÁ, Hana and DOHNAL, Jiří and KRÁL, Vladimír. Application of NIR for Characterization of Polymorph Purity and API-Excipient Cocrystals. Book of Abstracts: The XIXth Slovak - Czech Spectroscopic Conference, Častá-Papiernička, Slovakia, October 12-16, 2008, p. 96 (P-21). [ISBN 978-80-223-2557-8] 29. JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and RAICH, Ivan. Preparation and Physico-chemical Properties of Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1yl)hexanoates. Book of Abstracts: The International Conference “Frontiers in Medicinal Chemistry”, Heidelberg, Germany, March 15-18, 2009, p. 84. 30. JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and PEKÁREK, Tomáš and HAVLÍČEK, Jaroslav and DOHNAL, Jiří and KRÁL, Vladimír. Characterization of Polymorphs and API-Excipient Cocrystals Using Vibration Spectroscopy and Solid-state NMR. Book of Abstracts: The 11th International Workshop on Physical Characterization of Pharmaceutical Solids (IWPCPS ® 11), Stamford, Connecticut, USA, June 1419, 2009. 31. JAMPÍLEK, Josef and MUSIOŁ, Robert and CARROLL, James and O'MAHONY, Jim and COFFEY, Aidan and FINSTER, Jacek and TABAK, Dominik and NIEDBALA, Halina and DOHNAL, Jiří and POLAŃSKI, Jarosław. Synthesis and Antimycobacterial Activity of Styrylquinazolinone Derivatives. Book of Abstracts: The International Conference “The 6th Joint Meeting on Medicinal Chemistry 2009” (JMMC 2009), Budapest, Hungary, June 24-27, 2009, p. 73 (P-11). [ISBN 978-963-9319-95-0] 32. DOHNAL, Jiří and JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and ZERZAŇOVÁ, Anna and KRÁL, Vladimír. Utilization of NIR Spectroscopy in Candesartan Cilexetil Stability Study. Book of Abstracts: The 34th International Conference on Infrared, Millimeter, and Terahertz Waves (IRMMW-THz 2009), Busan, South Korea, September 21-25, 2009, p.59 (T5E25.0194). [ISBN 978-1-4244-5417-4] 33. OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and ZERZAŇOVÁ, Anna and DOHNAL, Jiří and KRÁL, Vladimír. Study of Interactions between API and Excipients in Solid Drug Formulation via NIR. Book of Abstracts: The 1st World Conference on Physico-Chemical Methods in Drug Discovery and Development, Rovinj, Croatia, September 27-October 1, 2009, p. 33 (OP-05). 34. ZERZAŇOVÁ, Anna and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and DOHNAL, Jiří and KRÁL, Vladimír. Absorption Study of Binary Mixtures. Book of Abstracts: The 1st World Conference on PhysicoChemical Methods in Drug Discovery and Development, Rovinj, Croatia, September 27-October 1, 2009, p. 48 (PP-06). 35. PAZOUREK, Jiří and DOHNAL, Jiří and JAMPÍLEK, Josef. Chiral Purity Determination of Z-alanine Using Capillary Electrophoresis. Book of Abstracts: The XXXIXth Conference “Synthesis and Analysis of Drugs”, Modra, Slovakia, September 2-4, 2010, p. 105 (P-58). [ISBN 978-80-7399-986-5] 36. OKTÁBEC, Zbyněk and IMRAMOVSKÝ, Aleš and PEJCHAL, Vladimír and JAMPÍLEK, Josef. RPHPLC Determination of Hydrophobic Properties of Novel Substituted Benzothiazole Derivatives. Book of Abstracts: The 28th International Symposium on Chromatography (ISC 2010), Valencia, Spain, September 12-16, 2010, p. 285 (P03-017). 37. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and PEJCHAL, Vladimír and JAMPÍLEK, Josef. Benzothiazole Derivates as Potent Acetylcholinesterase Inhibitors. Book of Abstracts: The International Conference “The 7th Joint Meeting on Medicinal Chemistry 2011” (JMMC 2011), Catania, Sicily, Italy, June 30-July 2, 2011. 38. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ŘEZÁČOVÁ, Anna and OKTÁBEC, Zbyněk and ČULEN, Martin and DOHNAL, Jiří. Approaches to Alaptide Water-Solubilization and Improvement of its Permeation Across Membranes. Book of Abstracts: The International Symposium on Advances in Synthetic and Medicinal Chemistry (ASMC 2011), St. Petersburg, Russia, August 21-25, 2011, p. 195 (P082). 39. JAMPÍLEK, Josef and MUSIOŁ, Robert and PÁVEK, Petr and KOWALCZYK, Wioleta and MAZUR, Paweł and POLAŃSKI, Jarosław. Investigation of Ring-substituted 3-(Benzylideneamino)-2-methylquinazolin-4(3H)-ones. Book of Abstracts: The International Symposium on Advances in Synthetic and Medicinal Chemistry (ASMC 2011), St. Petersburg, Russia, August 21-25, 2011, p. 196 (P083).
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40. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and MONREAL-FÉRRIZ, Juana and VINŠOVÁ, Jarmila and VANČO, Ján and JAMPÍLEK, Josef. New Carbamates of Salicylanilides as Potential Acetylcholinesterase Inhibitors and Their Molecular Docking. Book of Abstracts: The 63rd International Conference of Chemical Societies, Tatranské Matliare, Slovakia, September 5-9, 2011, ChemZi 2011, vol. 7, no. 13, 218. [ISSN 1336-7242] 41. ČULEN, Martin and DOHNAL, Jiří and JAMPÍLEK, Josef and ŘEZÁČOVÁ, Anna. Dynamic Dissolution Testing in R&D. Book of Abstracts: The 2nd World Conference on Physico-Chemical Methods in Drug Discovery and Development, Zadar, Croatia, September 18-22, 2011, p. 7 (OP-05). 42. BRYCHTOVÁ, Kateřina and JAMPÍLEK, Josef and DVOŘÁKOVÁ, Lenka and OPATŘILOVÁ, Radka and DOHNAL, Jiří. Investigating Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxoazepan-1-yl)hexanoates as Potential Transdermal Penetration Enhancers. Book of Abstracts: The 2nd World Conference on PhysicoChemical Methods in Drug Discovery and Development, Zadar, Croatia, September 18-22, 2011, p. 42 (PP02). 43. OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and DOHNAL, Jiří and ČULEN, Martin and KRÁL, Vladimír. Increasing of Drugs Water Solubility Using Pectines and Their Derivatives. Book of Abstracts: The 2nd World Conference on Physico-Chemical Methods in Drug Discovery and Development, Zadar, Croatia, September 18-22, 2011, p. 50 (PP-10). 44. JAMPÍLEK, Josef and VACULÍKOVÁ, Eliška and GRÜNWALDOVÁ, Veronika and KRÁL, Vladimír and DOHNAL, Jiří. Pilot Investigation of Nanoparticles Preparation by Precipitation. Book of Abstracts: The 48th International Conference on Medicinal Chemistry (RICT 2012), Poitiers, France, July 4-6, 2012, p. 103 (NA-03). 45. ČULEN, Martin and ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef and DOHNAL, Jiří. Dynamic dissolution using Golem apparatus – prediction of bioequivalence. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 79. [ISSN 0014-8172] 46. TENGLER, Jan and KAPUSTÍKOVÁ, Iva and BAĎO, Ondřej and RAČANSKÁ, Eva and JAMPÍLEK, Josef and MOKRÝ, Petr and CSÖLLEI, Jozef Preparation and study of physico-chemical and biological properties of new aryloxyaminopropanole derivatives. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 81-82. [ISSN 0014-8172] 47. GONĚC, Tomáš and CSÖLLEI, Jozef and MALÍK, Ivan and STOLAŘÍKOVÁ, Jiřina and COFFEY, Aidan and JAMPÍLEK, Josef and WAISSER, Karel. Phenylcarbamate derivatives with arylpiperazine fragment as antimycobacterial compounds. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 87. [ISSN 0014-8172] 48. KOS, Jiří and GONĚC, Tomáš and PEREIRA, Diogo and CHAMBEL, Bárbara and NĚMČÍKOVÁ, Ivana and MIKLASOVÁ, Hana and JAMPÍLEK, Josef. Synthesis of amides of hydroxynaphthalene acids as biologically active compounds. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 88. [ISSN 00148172] 49. DVOŘÁKOVÁ, Lenka and COUFAL, Libor and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Influencing penetration of corticoids through membranes using substance ALA. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 99. [ISSN 0014-8172] 50. FAJKUSOVÁ, Dagmar and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and VEJSOVÁ, Marcela and KELTOŠOVÁ, Stanislava and GUO, Jiahui and OKTÁBEC, Zbyněk and KOLLÁR, Peter and COFFEY, Aidan and CSÖLLEI, Jozef and JAMPÍLEK, Josef. Herbicidal and anti-infective activity of substituted 2aminobenzothiazoles. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 100. [ISSN 0014-8172] 51. ZITKO, Jan and DUFKOVÁ, Ida and PATEROVÁ, Pavla and JAMPÍLEK, Josef and KUBÍČEK, Vladimír and DOLEŽAL, Martin. Preparation, antimycobacterial and other biological effects of benzylamino derivatives of pyrazinamide. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 127. [ISSN 0014-8172] 52. ZADRAŽILOVÁ, Iveta and PAUK, Karel and MASAŘÍKOVÁ, Martina and IMRAMOVSKÝ, Aleš and ČÍŽEK, Alois and JAMPÍLEK, Josef. Antibacterial activity of salicylanilide esters against methicillinresistant Staphylococcus aureus (MRSA). Book of Abstracts: The IInd International Conference on Antimicrobial Research (ICAR 2012), Lisbon, Portugal, November 21-23, 2012, p. 481.
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53. ZADRAŽILOVÁ, Iveta and KOS, Jiří and POKORNÁ, Michaela and GONĚC, Tomáš and BOBÁL, Pavel and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro antimycobacterial activity of ring-substituted 3hydroxynaphthalene-2-carboxanilides. Book of Abstracts: The IInd International Conference on Antimicrobial Research (ICAR 2012), Lisbon, Portugal, November 21-23, 2012, p. 510. 54. ŽEMLIČKA, Milan and OPATŘILOVÁ, Radka and DOHNAL, Jiří and JAMPÍLEK, Josef. Internal differentiation of study, profiling of student according to choice of compulsory optional courses. Book of Abstracts: The 19th Annual Conference of the European Association of Faculties of Pharmacy (EAFP 2013), Ankara, Turkey, May 16-18, 2013, p. 106 (P-33). 55. ZADRAŽILOVÁ, Iveta and PAUK, Karel and IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and MASAŘÍKOVÁ, Martina and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro anti-MRSA activity of 2hydroxy-N-[1-(2-hydroxyphenylamino)-1-oxoalkan-2-yl]benzamides? Book of Abstracts: Antimicrobial Drug Conference, STARS EC FP7 Initial Training Network & TRAIN-ASAP ITN, Madrid, Spain, June 10-12, 2013, p. 70 (PO 19). 56. KOS, Jiří and GONĚC, Tomáš and JAMPÍLEK, Josef. Investigating the Spectrum of Biological Activity of Ring-Substituted 3-Hydroxynaphthalene-2-carboxanilides. Book of Abstracts: The 49th International Conference on Medicinal Chemistry (RICT 2013), Nice, France, July 3-5, 2013, p. 229 (HT-053). 57. ORAVEC, Michal and JAMPÍLEK, Josef and ZÁRUBA, Kamil and OPATŘILOVÁ, Radka and SUCHÝ, Pavel. Determination of Drugs in Silica Gel-Based Nanocarriers in Tissues. Book of Abstracts: The XVIIth euroANALYSIS, Warsaw, Poland, August 25–29, 2013, p. 183. [ISBN 978-83-7798-089-7] 58. ČERNÍKOVÁ, Aneta and COUFALOVÁ, Lenka and OPATŘILOVÁ, Radka and DOHNAL, Jiří and JAMPÍLEK, Josef. Evaluation of Alaptide as a Potential Modifier of Transdermal Penetration of Antimicrobial Agents. Book of Abstracts: The 9th Balaton Symposium on High-Performance Separation Methods, Siófok, Hungary, September 4-6, 2013, p. 15 (L-13). 59. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ČERNÍKOVÁ, Aneta and COUFALOVÁ, Lenka and DOHNAL, Jiří. In vitro evaluation of penetration of nanonized alaptide from semi-solid formulations. Book of Abstracts: The 3rd World Conference on Physico-Chemical Methods in Drug Discovery and Development, Dubrovnik, Croatia, September 22-26, 2013, p. 48 (PP-10). 60. PĚNTÁKOVÁ, Monika and MUSIOŁ, Robert and POLAŃSKI, Jarosław and JAMPÍLEK, Josef. Molecular Dynamics of the Newly Designed Inhibitors EGRF. Book of Abstracts: The BIT′s 4th Annual International Congress of Medichem 2013 (ICM-2013), Haikou, China, November 13-16, 2013, p. 94. 61. DOHNAL, Jiří and COUFALOVÁ, Lenka and ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Alaptide as Transdermal Penetration Modifier. Book of Abstracts: The BIT′s 3rd Annual Symposium of Drug Delivery Systems 2013 (SDDS-2013), Haikou, China, November 13-16, 2013, p. 244. 62. FAJKUSOVÁ, Dagmar and PEŠKO, Matúš and KELTOŠOVÁ, Stanislava and GUO, Jiahui and OKTÁBEC, Zbyněk and VEJSOVÁ, Marcela and KOLLÁR, Peter and COFFEY, Aidan and CSÖLLEI, Jozef and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Synthesis and Biological Activities of Substituted 2-Aminobenzothiazoles. Book of Abstracts: The 16th JCF-Frühjahrssymposium 2014, Friedrich-SchillerUniversität Jena, Jena, Germany, March 26-29, p. 70 (P-4). 63. KELTOŠOVÁ, Stanislava and JAMPÍLEK, Josef and KOLLÁR, Peter. In Vitro Biological Evaluation of New Potential Anticancer Drugs. Book of Abstracts: The 64th Pharmacological days and the 24th Martin Respiration Days, Martin, Slovakia, June 25-27, 2014, p. 40. [ISBN 978-80-89544-70-7] 64. GONĚC, Tomáš and ZADRAŽILOVÁ, Iveta and NEVIN, Eoghan and KOS, Jiří and COFFEY, Aidan and JAMPÍLEK, Josef. Synthesis and Biological Activity of N-(alkoxyphenyl)-2-hydroxynaphthalene-1carboxamides. Book of Abstracts: The XLIIIrd Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 4-6, 2014, Farm. Obzor 2014, vol. 83, no. 8-9, 182. [ISSN 0014-8172] 65. ČERNÍKOVÁ, Aneta and JAMPÍLEK, Josef. Modification of Transdermal Penetration of Different Drugs with Alaptide as Potential Enhancer. Book of Abstracts: The 7th Central European Conference "Chemistry towards Biology", Katowice, Poland, September 9-12, 2014, p. P19. 66. JAMPÍLEK, Josef and ORAVEC, Michal and ZÁRUBA, Kamil and ULBRICH, Pavel and BABULA, Petr and KUNEŠ, Martin and SUCHÝ, Pavel. Preparation and In Vivo Permeation of Drugs in Silica Gel-Based Nanocarriers through Blood–Brain Barrier. Book of Abstracts: The 7th Central European Conference "Chemistry towards Biology", Katowice, Poland, September 9-12, 2014, p. P21. 67. MALARZ, Joanna and KROMPIEC, Stanisław and PIETRASZUK, Cezary and JAMPÍLEK, Josef and VEJSOVÁ, Marcela. Synthesis of trisubstituted isoxazoles and their biological properties. Book of Abstracts: The 57th Meeting of the Polish Chemical Society and the Society of Engineers and Technicians of Chemical Industry, Częstochowa, Poland, September 14-18, 2014, p. 115 (S01-P121). [ISSN 978-83931072-6-1]
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68. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and ČÍŽEK, Alois and JAMPÍLEK, Josef. Time-kill curve kinetics of 4-chloro-N{(2S)-1-[(3,4-dichlorophenyl)amino]-3-methyl-1-oxobutan-2-yl}-2-hydroxybenzamide against multidrugresistant clinical isolates of methicillin-resistant Staphylococcus aureus (MRSA). Book of Abstracts: The 3rd International Conference on Antimicrobial Research (ICAR 2014), Madrid, Spain, October 1-3, 2014, p. 327 (T71). 69. DOHNAL, Jiří and ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Advances in Investigation of Alaptide as Transdermal Permeation Modifier. Book of Abstracts: The BIT′s 4th Annual Symposium of Drug Delivery Systems 2014 (SDDS-2014), Suzhou, China, November 18-20, 2014, p. 66. 70. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and IMRAMOVSKÝ, Aleš and ČÍŽEK, Alois and JAMPÍLEK, Josef. Antibacterial Activity of Novel Salicylanildes Against Vancomycinresistant Enterococcus faecalis (VRE). Book of Abstracts: The 25th European Congress of Clinical Microbiology and Infectious Diseases (ECCMID 2015), Copenhagen, Denmark, April 25-28, 2015, EV0211. 71. GONĚC, Tomáš and STRÁNÍK, Josef and KOS, Jiří and ORAVEC, Michal and JAMPÍLEK Josef. Synthesis of Substituted 1-(Phenylcarbamoyl)naphthalen-2-yl Alkylcarbamates with Potential Antimycobacterial Activity. Book of Abstracts: The 67th International Conference of Chemical Societies, Horný Smokovec, Slovakia, September 7-11, 2015, ChemZi 2015, vol. 11, no. 1, 144-145 (3Po09). [ISSN 1336-7242] 72. KOS, Jiří and GONĚC, Tomáš and NEVIN, Eoghan and COFFEY, Aidan and JAMPÍLEK Josef. RingSubstituted 8-Hydroxyquinoline-2-carboxanilides as Potential Antitubercular Agents. Book of Abstracts: The 67th International Conference of Chemical Societies, Horný Smokovec, Slovakia, September 7-11, 2015, ChemZi 2015, vol. 11, no. 1, 152 (3Po22). [ISSN 1336-7242] AFH Abstrakty příspěvků z domácích vědeckých konferencí 1. DOLEŽAL, Martin and JAMPÍLEK, Josef and BUCHTA, Vladimír. Synthesis and Biological Evaluation of 5-Aroylpyrazine-2-carboxylic Acid Derivatives. Book of Abstracts: The XXVIIIth Conference "Synthesis and Analysis of Drugs", Hradec Králové, Czech Republic, September 15-17, 1999, p. 40. 2. JAMPÍLEK, Josef and DOLEŽAL, Martin and DEIGNER, Hans-Peter. Sphingosine Preparation as Potential Antineoplastics by Optimized Tkaczuk-Thornton Method. Book of Abstracts: The XXXth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 17-19, 2001, p. 73. [ISBN 80-7305-416-7] 3. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří and BUCHTA, Vladimír. Preparation and Antimycotic Activity of Thiazol-2-ylamide pyrazine-2-carboxylic acid Derivatives. Book of Abstracts: The XXXIInd Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 16-19, 2003, p. 134. [ISBN 80-900306-5-3] 4. JUN, Daniel and JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and HRDINA, Radomír and OPLETAL, Lubomír. Antiplatelet Activity of Arylalkanoic Acid. Book of Abstracts: The XXXIInd Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 16-19, 2003, p. 135. [ISBN 80-900306-5-3] 5. OPLETALOVÁ, Veronika and POUR, Milan and KUNEŠ, Jiří and SILVA, Luís and BUCHTA, Vladimír and JAMPÍLEK, Josef and RICHARDSON, Des Robert and KALINOWSKI, Danuta. Thiosemicarbazones of Acetylpyrazines as Potential Drugs. Book of Abstracts: The 11th Blue Danube Symposium on Heterocyclic Chemistry, Brno, Czech Republic, August 28-September 1, 2005, PO-70. [ISBN 80-2103763-6] 6. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK Josef. Hydrazone Derivatives of Some Antituberculotics. Book of Abstracts: The XXXIVth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 12-14, 2005, p. 68. [ISBN 80-7305-533-3] 7. DOLEŽEL, Jan and OPLETALOVÁ, Veronika and BUCHTA, Vladimír and SILVA, Luís and JAMPÍLEK, Josef and DOHNAL, Jiří and RICHARDSON, Des Robert and KALINOWSKI, Danuta and KRÁĽOVÁ, Katarína. Synthesis and Biological Evaluation of Thiazole Derivatives. Book of Abstracts: The XXXVth Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 12-15, 2006, p. 85. [ISBN 80-7305-566-X] 8. OPLETALOVÁ, Veronika and DOLEŽEL, Jan and KUNEŠ, Jiří and JAMPÍLEK, Josef and SILVA, Luís and BUCHTA, Vladimír and ŠPANINGEROVÁ, Eliška and KEŠETOVIČOVÁ, Diana and VLČKOVÁ, Martina. Antifungal Activity of Benzylidenerhodanines. Book of Abstracts: The XXXVth Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 12-15, 2006, p. 120. [ISBN 80-7305-566-X]
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DOHNAL, Jiří and HAVLÍČEK, Jaroslav and JAMPÍLEK, Josef and BRUSOVÁ, Hana. Pharmaceutical Analysis in Solid State. Book of Abstracts: The XXXVIIIth Conference “Synthesis and Analysis of Drugs”, Hradec Králové, Czech Republic, September 14-16, 2009, p. 25-26 (L-2). [ISBN 978-80-7305-078-8] JAMPÍLEK, Josef and DOLEŽAL, Martin and KEŠETOVIČOVÁ, Diana. Structure-lipophilicity Relationships in Series of Methoxy Moiety Ring-substituted Pyrazinecarboxanilides. Book of Abstracts: The XXXVIIIth Conference “Synthesis and Analysis of Drugs”, Hradec Králové, Czech Republic, September 14-16, 2009, p. 90 (P-28). [ISBN 978-80-7305-078-8] SLABÁ, Barbora and PLAČEK, Lukáš and RIDVAN, Luděk and JAMPÍLEK, Josef. Identification of Almotriptan Impurity Using HPLC-MS/MS and HR-MS. Book of Abstracts: The XXXVIIIth Conference “Synthesis and Analysis of Drugs”, Hradec Králové, Czech Republic, September 14-16, 2009, p. 141 (P79). [ISBN 978-80-7305-078-8] DOHNAL, Jiří and HAVLÍČEK, Jaroslav and JAMPÍLEK, Josef and BRUSOVÁ, Hana and KREJČÍK, Lukáš. Position of Thermal Methods in Pharmaceutical Analysis of Solid State. Book of Abstracts: The 32nd International Czech and Slovak Calorimetric Meeting (Kalsem 2010), Lísek u Bystřice pod Pernštejnem, Czech Republic, May 24-28, 2010, p. 77-78. [ISBN 978-80-7395-259-4] JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and DOHNAL, Jiří. NIR and its Application in Pharmacy. Proceedings of lifelong learning lectures „Properties and Analysis of Solid Pharmaceutical Substances 2011“. Department of Solid State Chemistry, Faculty of Chemical Technology, Institute of Chemical Technology Prague, Czech Republic, April 28-29, 2011. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and MONREAL-FÉRRIZ, Juana and VINŠOVÁ, Jarmila and VANČO, Ján and JAMPÍLEK, Josef. Salicylanilide Carbamates as Acetylcholinesterase Inhibitors and Their Molecular Docking. Book of Abstracts: The 2nd French-Czech Vltava Chemistry Meeting, Pardubice, Czech Republic, August 30-31, 2011, p. 31. [ISBN 978-80-7395-412-3] GONĚC, Tomáš and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef and PAVLACKÁ, Lenka. Synthesis of Substituted 2-Naphthoylanilides as Potential Photosynthesis Inhibitors. Book of Abstracts: The XLth International Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 12-14, 2011, S-6. [ISBN 978-80-7305-593-6] ČULEN, Martin and DOHNAL, Jiří and JAMPÍLEK, Josef and ŘEZÁČOVÁ, Anna. Example of Dynamic Dissolution Testing Results Obtained with Golem Apparatus. Book of Abstracts: The XLth International Conference “ Synthesis and Analysis of Drugs ”, Brno, Czech Republic, September 12-14, 2011, P-11. [ISBN 978-80-7305-593-6] JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and PEJCHAL, Vladimír and OKTÁBEC, Zbyněk. RP-HPLC Determination of Hydrophobic Properties of Substituted Fluorobenzothiazole Derivatives. Book of Abstracts: The XLth International Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 12-14, 2011, P-32. [ISBN 978-80-7305-593-6] KOS, Jiří and JAMPÍLEK, Josef and GONĚC, Tomáš and BOBÁL, Pavel. Synthesis of NArylquinoxaline-2-carboxamides as Potential Antimicrobial Compounds. Book of Abstracts: The XLth International Conference “ Synthesis and Analysis of Drugs ”, Brno, Czech Republic, September 12-14, 2011, P-42. [ISBN 978-80-7305-593-6] OPATŘILOVÁ, Radka and BREZOVSKÁ, Monika, JAMPÍLEK, Josef. Study of Drug Penetration through a Barier. Book of Abstracts: The XLth International Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 12-14, 2011, P-61. [ISBN 978-80-7305-593-6] ČULEN, Martin and DOHNAL, Jiří and ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef. Artificial Digestive Tract – Golem. Book of Abstracts: Science and Research for Innovations (Part of net NINET realized with financial support of the program EUPRO-OK08003 of the Ministry of Education of the Czech Republic), Brno, Czech Republic, September 5, 2012, p. 12. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and ČECH-BARABASZOVÁ, Karla and JAMPÍLEK, Josef. Nanotechnologies in field of pharmacy. Book of Abstracts: The 3rd International Nanomaterials and Nanotechnology Meeting “NANO-Ostrava 2013”, Ostrava, Czech Republic, June 17-20, 2013, p. 61 (OP 12). [ISBN 978-80-7329-361-1] ZADRAŽILOVÁ, Iveta and PAUK, Karel and IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and POKORNÁ, Michaela and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro antimycobacterial activity of new synthesized salicylanilide esters. Book of Abstracts: The 26th Congress of the Czechoslovak Society for Microbiology, Brno, Czech Republic, June 24-26, 2013, p. 128. [ISBN 978-80-260-4507-6] VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Permeation/Penetration of Drug Nanoparticles through Skin and Their Potential Toxicity. Book of Abstracts: The 2nd International Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech Republic, November 6-8, 2013, p. 19. [ISBN 978-80-248-3240-1]
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24. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and MASAŘÍKOVÁ, Martina and IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and ČÍŽEK, Alois and JAMPÍLEK, Josef. Analysis of Bactericidal Effect of 4-Chloro-2-(4-chlorophenylcarbamoyl)phenyl Decylcarbamate against MRSA in Dependence on Time and Concentration under Conditions in Vitro. Book of Abstracts: The XXIIIrd Tomášek Days of Young Microbiologists 2014, Brno, Czech Republic, June 5-6, 2014, p. 39. [ISBN 97880-210-6508-6] 25. ČERNÍKOVÁ, Aneta and JAMPÍLEK, Josef. Evaluation of Alaptide as Potential Permeation Enhancer for Transdermal Delivery of Model Drug Theophylline. Book of Abstracts: The 4th Meeting of the Paul Ehrlich MedChem Euro-PhD Network, Hradec Králové, Czech Republic, June 20-22, 2014, p. 40 (O-21). 26. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Preparation of Risedronate Nanoparticles for Permeability Improvement. Book of Abstracts: The 4th Meeting of the Paul Ehrlich MedChem Euro-PhD Network, Hradec Králové, Czech Republic, June 20-22, 2014, p. 41 (O-22). 27. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISARČÍK, Martin and PEIKERTOVÁ, Pavlína and DĚDKOVÁ, Kateřina and JAMPÍLEK, Josef. Characterization of cimetidine nanoparticles for solubility test. Book of Abstracts: The 4th Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava, Czech Republic, May 18-21, 2015, p. 79. [ISBN 978-80-248-3745-1] 28. BÁBKOVÁ, Zuzana and POLÁŠKOVÁ, Alena and ADÁMIK, Matej and HELMA, Robert and KOS, Jiří and GONĚC Tomáš and JAMPÍLEK, Josef and BRÁZDOVÁ, Marie. Study of Biological Activity of Hydroxynaphthalene Carboxanilide Derivatives on Tumor Cell Lines. Book of Abstracts: The 20th Interdisciplinary Czech-Slovak Toxicology Conference (TOXCON 2015), Brno, Czech Republic, May 27-29, 2015, p. 26. [ISBN 978-80-263-0933-8] 29. KELTOŠOVÁ, Stanislava and JAMPÍLEK, Josef and KOLLÁR, Peter. Evaluation of Effect of Newly Synthesized Quinazolines on Proliferation and Cell Cycle of Human Tumor Cell Lines. Book of Abstracts: The 20th Interdisciplinary Czech-Slovak Toxicology Conference (TOXCON 2015), Brno, Czech Republic, May 27-29, 2015, p. 74. [ISBN 978-80-263-0933-8] 30. ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel and JAMPÍLEK, Josef. Analogues of Alaptide and Their Effect on the Penetration of Drugs. Book of Abstract: The XLIVth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 46 (P07). [ISBN 978-80-7305-760-2] 31. GONĚC, Tomáš and KMEŤKO, Juraj and KOS, Jiří and POSPÍŠILOVÁ, Šárka and ZADRAŽILOVÁ, Iveta and JAMPÍLEK Josef. Synthesis and Antimicrobial Activity of N-(halogenphenyl)-1hydroxynaphthalene-2-carboxamides. Book of Abstract: The XLIVth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 57 (P16). [ISBN 978-80-7305-760-2] 32. JĘDRZEJOWSKA, Agnieszka and MATUSSEK, Marek and KOZIK, Violetta and BĄK, Andrzej and ZADRAŽILOVÁ, Iveta and JAMPÍLEK Josef. Synthesis and Biological Properties of Chosen Symmetrical Amides and Thioamides of Terephthalic Acid. Book of Abstract: The XLIVth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 63 (P20). [ISBN 978-80-7305-760-2] 33. KOS, Jiří and GONĚC, Tomáš and ZADRAŽILOVÁ, Iveta and VALEŠOVÁ, Miroslava and POSPÍŠILOVÁ, Šárka and SPACZYŃSKA, Ewelina and JAMPÍLEK Josef. Ring-Substituted 1Hydroxynaphthalene-2-Carboxanilides as Potential Antibacterial Agents. Book of Abstract: The XLIVth Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 72 (P27). [ISBN 978-80-7305-760-2] 34. KAUEROVÁ, Tereza and GONĚC, Tomáš and KOS, Jiří and JAMPÍLEK Josef and KOLLÁR, Peter. In Vitro Analysis of Antiproliferative Effects of Newly Synthesized Nitro-substituted Hydroxynaphthanilides with Focus on Cell Cycle of Tumor Cell Lines. Book of Abstracts: The 65th Pharmacological Days, Prague, Czech Republic, September 16-18, 2015, p. 31. [ISBN 978-80-260-8027-5] 35. GONĚC, Tomáš and KOS, Jiří and ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and ŠORAL, Michal and LIPTAJ, Tibor and JAMPÍLEK Josef. Synthesis and Antibacterial Activity of N-(substituted phenyl)-1-hydroxynaphthalene-2-carboxamides. Book of Abstracts: LIBLICE 2015 – The 50th Conference: “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Olomouc, Czech Republic, November 6-8, 2015, p. 72 (Po20).
Výzkumné projekty obhájené nebo řešené (celkem 15 projektů) 1. 2.
Člen řešitelského kolektivu. HARTL, Jiří. „Biologicky aktivní deriváty pyrazinu a pyridinu“. Grantová agentura Univerzity Karlovy (GAUK 026/1998/B-CH/FaF) v letech 1998–2000. Člen řešitelského kolektivu. KARLÍČEK, Rolf. „Vývoj, příprava a technologie léčiv“. Výzkumné záměry Ministerstva školství, mládeže a tělovýchovy České republiky (MSM 111600001) v letech 1999–2004.
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Člen řešitelského kolektivu. KVASNIČKOVÁ, Eva. „Centrum pro výzkum struktury a mechanismu účinku potenciálních léčiv B5“. Ministerstvo školství, mládeže a tělovýchovy České republiky (LN00B125) v letech 2000–2004. JAMPÍLEK, Josef. „Dokončení přípravy série potenciálních antituberkulotik a antimykotik“. Fond rozvoje vysokých škol 2002 G4a – Tvůrčí činnost studentů – přírodovědné obory (FRVŠ 2245/G4/2002). JAMPÍLEK, Josef. „Pokračování přípravy potenciálně účinných antituberkulotik a antimykotik“. Fond rozvoje vysokých škol 2003 G6a – Tvůrčí činnost studentů – přírodovědné obory (FRVŠ 2998/G6/2003). CHLUPÁČOVÁ, Marta a JAMPÍLEK, Josef. „Chalkony a jejich analoga jako potenciální léčiva“. Fond rozvoje vysokých škol 2003 G3a – Tvůrčí činnost studentů – biomedicínské obory (FRVŠ 2970/G3/2003). JAMPÍLEK, Josef. „Cílený transport léčiva přes biologické membrány“. Grantová agentura České republiky (GAČR P304/11/2246) v letech 2011–2014. KOS, Jiří a JAMPÍLEK, Josef. „Syntéza amidů kyselin hydroxynaftoových jako biologicky aktivních látek“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 96/2012/FaF) v roce 2012. Člen řešitelského kolektivu. SEDMÍKOVÁ, Markéta a SALAŠOVÁ, Alena a VEČEREK, Vladimír. Centralizovaný rozvojový projekt Ministerstva školství, mládeže a tělovýchovy České republiky 2014 „Zvyšování kvalifikace studentů doktorských studijních programů a post-doktorandů zemědělských a veterinárních oborů zapojením do multidisciplinárních meziuniverzitních týmů.“ (MŠMT ČR, projekt č. C3) v roce 2014. JAMPÍLEK, Josef. „Syntéza amidů kyseliny kynureninové jako biologicky aktivních látek“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 37/2014/FaF) v roce 2014. ZADRAŽILOVÁ, Iveta a JAMPÍLEK, Josef. „Studium antimikrobiálních vlastností nově syntetizovaných potenciálních chemoterapeutik“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 52/2014/FaF) v roce 2014. Člen řešitelského kolektivu. SOPUCH, Tomáš. „Matricové systémy pro hojení kožních defektů pro humánní a veterinární použití“. Technologická agentura České republiky (TAČR TA04010065) v letech 2014–2017. ČERNÍKOVÁ, Aneta a JAMPÍLEK, Josef. „Hodnocení derivátů alaptidu jako potenciálních modifikátorů transdermální penetrace“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 302/2015/FaF) v roce 2015. JAMPÍLEK, Josef. „Protiinvazivní aktivita nových antimikrobiálních chemoterapeutik“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 304/2015/FaF) v roce 2015. Member of research group. SOBCZAK-KUPIEC, Agnieszka. “Innovative Composite Biomaterials Contained Bioactive Calcium Phosphates”. The National Centre for Research and Development, Warsaw, Poland (LIDER/037/481/L-5/13/NCBR) in 2015.
Vyžádané přednášky na konferencích a workshopech (celkem 26 přednášek) Vyžádané přednášky na vědeckých konferencích konaných v České republice 1. The 1st International Symposium and Workshop on Environment and Health (ISEH 2012), Ostrava, Czech Republic, November 22-23, 2012. (Invited plenary lecture “Perspectives of Nanoparticles in Pharmacy”, Book of Abstract: p. 44 [ISBN 978-80-248-2882-4]). 2. The 2nd International Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech Republic, November 6–8, 2013. (Invited plenary lecture “Polymorphism and Its Influence to Bioavailability”, Book of Abstract: pp. 20-21 [ISBN 978-80-248-3240-1]). 3. The 4th Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava, Czech Republic, May 18–21, 2015. (Invited lecture “Overcoming Blood-Brain Barrier Using Nanoparticles”, Book of Abstract: p. 63 [ISBN 978-80-248-3745-1]). 4. The International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering (NDDTE'16), Prague, Czech Republic, April 1-2, 2016. (Invited keynote lecture “Nanoformulations of Antimicrobial Chemotherapeutics”, Book of Abstracts: Keynote-2, http://nddte.com/keynote/#Prof.%20Josef%20Jampilek & http://nddte.com/paper/Keynote%20-%20Dr.%20Jampilek.pdf). Vyžádané přednášky na zahraničních vědeckých konferencích 1. The XXXV Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, May 30–June 1, 2012. (Invited plenary lecture “Advances in Investigation of Hydrophilic and Lipophilic Properties of Drugs”, Book of Abstract: OS-5).
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The XXXVI Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, June 5–7, 2013. (Invited plenary lecture “Pharmaceutical nanoparticles and methods of their characterization”, Book of Abstract: OS-19). The BIT′s 4th Annual International Congress of Medichem 2013 (ICM-2013), Haikou, China, November 13–16, 2013. (Invited lecture “Design and Antimicrobial Screening of New Ring-substituted Quinoline Analogues”, Book of Abstract: p. 62). The XXXVII Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, June 11–13, 2014. (Invited plenary lecture “Investigation of Cholic Acid Derivatives as Transdermal Permeation Enhancers”, Book of Abstract: OS-18). The 7th Central European Conference 'Chemistry towards Biology, Katowice, Poland, September 9–12, 2014. (Invited lecture “Synthesis and Antimicrobial Activity of Hydroxy(aza)naphthalenecarboxamides”, Book of Abstract: O5). The VI Conversatory on Medicinal Chemistry, Lublin, Poland, September 18–20, 2014. (Invited lecture “Synthesis and In Vitro Anti-trypanosomal Screening of Hydroxynaphthalene-2-carboxanilides”, Book of Abstract: p. 24 (K5) [ISSN 978-83-63657-38-3]). International Scientific-Practical Conference Pharmaceutical Education, Scientific and Manufacturing as a Reference to the Strategy Kazakhstan-2020, Faculty of Pharmacy, South Kazakhstan State Pharmaceutical Academy, Shymkent, Kazakhstan, October 23–24, 2014. (Invited opening lecture “Quality by Design: New Approach to Development of Drugs and Assurance of Their Quality”). International Scientific-Practical Conference Pharmaceutical Education, Scientific and Manufacturing as a Reference to the Strategy Kazakhstan-2020, Faculty of Pharmacy, South Kazakhstan State Pharmaceutical Academy, Shymkent, Kazakhstan, October 23–24, 2014. (Invited plenary lecture “Design, Synthesis and Anti-staphylococcus Activity of Hydroxynaphthalenecarboxanilides”, Book of Abstract: Republican Scientific Journal 2014, vol. 68, no. 3, 3–7 [ISSN 2306-6822]). The BIT′s 5th Annual International Congress of Medichem 2014 (ICM-2014), Suzhou, China, November 18–20, 2014. (Invited lecture “Recent Advances in Design of Potential Quinoxaline Anti-Infectives”, Book of Abstract: p. 197). The 13th Ibn Sina International Conference on Pure and Applied Heterocyclic Chemistry, Hurghada, Egypt, February 14–17, 2015. (Invited plenary lecture “Azanaphthalenes as Potential Antimycobacterial Agents”, Book of Abstract: p. 8 (PL-06)). The XXXVIII Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, May 27–29, 2015. (Invited plenary lecture “Determination of Drugs Loaded to Silica Nanoparticles in Brain Tissue”, Book of Abstract: OS-27). The IX Joint Meeting in Medicinal Chemistry (JMMC 2015), Athens, Greece, June 7–10, 2015. (Invited keynote lecture “Advances in Design of Potential Quinoline Antimycobacterial Agents”, Book of Abstract: O6). European Pharma Congress “Pharma Europe-2015”, Valencia, Spain, August 25-27, 2015. (Invited lecture “Design, Synthesis and Investigation of Aryl Derivatives of Alaptide as Potential Transdermal Permeation Enhancers”, Book of Abstract: J. Pharma. Care Health Sys. 2015, vol. 2, no. 4, 63. [ISSN 2376-0419]). The 4th World Conference on Physico-Chemical Methods in Drug Discovery and Development (PCMDDD4), Rovinj – Red Island, Croatia, September 21-24, 2015. (Invited lecture “In Vitro Evaluation of 8Substituted 6,9-diazaspiro[4.5]decan-7,10-diones as Skin Permeation Modifiers”, Book of Abstract: p. 10 (OP-08)). The 24th Annual Central European Conference (ECOpole’15), Jarnołtówek, Poland, October 14-17, 2015. (Invited keynote lecture “Applications of nanoformulations in Agricultural Production and Their Potential Impact on Food and Human Health” (http://ecopole.uni.opole.pl/index.php/invited-presentations). Proceedings: Proceedings of ECOpole 2015 (PECO-2015), 2015, vol. 9, no. 2, 465-472. [ISSN 1898617X] The BIT's 13th Annual World Congress of International Drug Discovery Science & Technology, Therapy and EXPO-2015 (IDDST 2015), Beijing, China, October 20-22, 2015. (Invited lecture “Design and Antimicrobial Activity of Ring-Substituted Hydroxynaphthalenecarboxamides and Their Aza-Analogues”, Book of Abstract: p. 109). The BIT's 5th Annual World Symposium of Drug Delivery System 2015 (SDDS-2015), Beijing, China, October 20-22, 2015. (Invited lecture “Investigation of Alkyl Derivatives of Alaptide as Transdermal Permeation Modifier”, Book of Abstract: p. 387).
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Vyžádané odborné přednášky na seminářích a workshopech 1. Zentiva Praha, Česká republika, 28. březen 2008 („Infračervená spektroskopie v blízké oblasti – NIR“, přednáška v rámci přednáškového cyklu „Science Forum” v délce 2 akademických hodin). 2. Ústav chemie pevných látek, Fakulta chemické technologie, Vysoká škola chemicko-technologická v Praze, 28.–29. duben 2011. („NIR a jeho využití ve farmacii“, přednáška v rámci kurzu celoživotního vzdělávání „Vlastnosti a analýza pevných farmaceutických substancí 2011” v délce 3 akademických hodin). 3. Státní ústav pro kontrolu léčiv (SÚKL), Praha, Česká republika, 19.–20. duben 2012. (“Polymorphism – What It Say?”, přednáška v rámci vzdělávací akce „EU Assessors Training on Efficient and Effective Quality Assessment“ v délce 3 akademických hodin). 4. Ústav analytické chemie, Akademie věd České republiky, Brno, 2. květen 2012. („Polymorfie léčiv a metody jejího stanovení“, přednáška v rámci cyklu „Kulatý stůl“ v délce 3 akademických hodin). 5. Centrum výzkumu globální změny Akademie věd České republiky, Brno, 4. listopad 2014 (“Application of Nanoparticles in Pharmacy – Overcoming BBB and Methods Analysis of Nanoparticles“, odborný seminář v délce 3 akademických hodin).
Členství v redakčních radách (celkem 6) Členství v redakčních radách (tuzemských) 1. Military Medical Science Letters [ISSN 0372-7025], Faculty of Military Health Sciences, University of Defense, http://www.mmsl.cz/editorial-board (od roku 2011) Členství v redakčních radách (zahraničních) 1. Journal of Bioequivalence & Bioavailability [ISSN 0975-0851], OMICS Group, http://www.omicsonline. org/editorialboard-bioequivalence-bioavailability-open-access.php (od roku 2013) 2. ADMET & DMPK [ISSN 1848-7718], IAPC Publishing, http://pub.iapchem.org/ojs/index.php/admet/ about/editorialTeam (od roku 2014) 3. Open Pharmaceutical Sciences Journal [ISSN 1874-8449], Bentham Science Publishers, http://benthamopen.com/PHARMSCI/editorial-board/ (od roku 2015) 4. ChemistrySelect [ISSN 2365-6549], Wiley-VCH, http://onlinelibrary.wiley.com/journal/10.1002/%28 ISSN%292365-6549/homepage/2766_edbd.html (od roku 2015) 5. Medicinal Chemistry [ISSN 1875-6638, IF2014 = 1.363], Bentham Science Publishers, http://benthamscience.com/journals/medicinal-chemistry/editorial-board/#top (od roku 2015) Redaktor speciálních čísel 1. Prodrugs: Pharmaceutical Design and Current Perspectives. Current Pharmaceutical Design 2011, vol. 17, no. 32, http://benthamscience.com/journal/contents.php?journalID=cpd&issueID=7364. [ISSN 1381-6128, IF2011 = 3.870] 2. Enhanced skin drug permeability: methodology, assessment and enhancement approaches. ADMET & DMPK 2014, vol. 2, no. 4, http://pub.iapchem.org/ojs/index.php/admet/issue/view/26. [ISSN 1848-7718] 3. Modern Approaches to Quality Assurance of Drug Formulations. BioMed Research International 2015, vol. 2015, http://www.hindawi.com/journals/bmri/si/970238/. [ISSN 2314-6133, IF2014 = 1.579] 4. Anti-Infective Drug Discovery Based on Diversified Plant Natural Compounds. Current Organic Chemistry 2016, http://benthamscience.com/journal-files/special-issue-details/COC-SII20151116-01.pdf. [ISSN 1875-5348, IF2014 = 2.157]
Členství v komisích výzkumných agentur a vědeckých výborech 1.
Člen hodnotícího panelu P207 „Chemické a biochemické přeměny” Grantové agentury České republiky (2015–2017), http://gacr.cz/poradni-organy/panely/
Členství ve vědeckých a odborných společnostech 1. 2. 3. 4.
Česká společnost chemická – sekce Organická, bioorganická a farmaceutická chemie (od roku 2002) Česká farmaceutická společnost – sekce Syntetických léčiv (od roku 2002) International Association of Physical Chemists (od roku 2014) Working Group on New TB Drugs (od roku 2015)
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Vypracování posudků Oponentské posudky na vědecké články (celkem 118 posuzovaných rukopisů) 1. Acta Chromatographica [ISSN 1233-2356, IF2014 = 0.577], Institute of Chemistry, University of Silesia, Katowice, Poland 1× 2. ADMET & DMPK [ISSN 1848-7718], IAPC Publishing 1× 3. African Journal of Pharmacy and Pharmacology [ISSN 1996-0816], Academic Journals 1× 4. Anti-Cancer Agents in Medicinal Chemistry [ISSN 1871-5206, IF2014 = 2.469], Bentham Science Publishers 2× 5. Arabian Journal of Chemistry [ISSN 1878-5352, IF2014 = 2.725], Elsevier 2× 6. ASC Combinatorial Science [ISSN 2156-8952, IF2014 = 3.032], American Chemical Society 1× 7. Biochemistry and Biophysics Reports [ISSN 2405-5808], Elsevier 1× 8. Bioinorganic Chemistry and Applications [ISSN 1565-3633, IF2014 = 2.081], Hindawi Publishing Corporation 1× 9. BioMed Research International [ISSN 2314-6133, IF2014 = 1.579], Hindawi Publishing Corporation 1× 10. Bioorganic & Medicinal Chemistry [ISSN 0968-0896, IF2014 = 2.793], Elsevier 8× 11. Bioorganic & Medicinal Chemistry Letters [ISSN 0960-894X, IF2014 = 2.420], Elsevier 4× 12. British Journal of Pharmaceutical Research [ISSN 2231-2919], Science Domain International 2× 13. Carbohydrate Polymers [ISSN 0144-8617, IF2014 = 4.074], Elsevier 1× 14. Central European Journal of Chemistry [ISSN 1895-1066, IF2013 = 1.329], Springer 3× 15. Chemical Biology & Drug Design [ISSN 1747-0277, IF2014 = 2.485], Wiley-Blackwell 1× 16. Chemical Engineering Journal [ISSN 1385-8947, IF2014 = 4.321], Elsevier 1× 17. Chemické listy [ISSN 0009-2770, IF2014 = 0.272], Czech Chemical Society 6× 18. ChemMedChem [ISSN 1860-7179, IF2014 = 2.968], Wiley-VCH 8× 19. Chemistry and Biodiversity [ISSN 1612-1880, IF2014 = 1.515], Wiley-VCH 1× 20. Chromatography Research International [ISSN 2090-3502], Hindawi Publishing Corporation 1× 21. Combinatorial Chemistry & High Throughput Screening [ISSN 1386-2073, IF2014 = 1.222], Bentham Science Publishers 2× 22. Current Pharmaceutical Design [ISSN 1381-6128, IF2014 = 3.452], Bentham Science Publishers 3× 23. Current Organic Synthesis [ISSN 1570-1794, IF2014 = 2.117], Bentham Science Publishers 1× 24. Česká a Slovenská Farmacie [ISSN 1803-6597], Czech Medical Association of J.E. Purkyne 2× 25. European Journal of Medicinal Chemistry [ISSN 0223-5234, IF2014 = 3.447], Elsevier 9× 26. European Journal of Organic Chemistry [ISSN 1434-193X, IF2014 = 3.065], Wiley-VCH 2× 27. Expert Opinion on Drug Discovery [ISSN 1746-0441, IF2014 = 3.539], Informa Healthcare 1× 28. Frontiers in Life Science [ISSN 2155-3769, IF2014 = 0.294], Taylor & Francis 1× 29. International Journal of Medicinal Chemistry [ISSN 2090-2069], Hindawi Publishing Corporation 1× 30. International Journal of Pharmaceutics [ISSN 0378-5173, IF2014 = 3.650], Elsevier 1× 31. Journal of Applied Biomedicine [ISSN 1214-021X, IF2014 = 1.302], Elsevier 3× 32. Journal of Biochemical and Molecular Toxicology [ISSN 1095-6670, IF2014 = 1.925], Wiley-Blackwell 1× 33. Journal of Bioequivalence & Bioavailability [ISSN 0975-0851], OMICS Group 5× 34. Journal of Biomolecular Structure & Dynamics [ISSN 0739-1102, IF2014 = 2.919], Taylor & Francis 1× 35. Journal of the Brazilian Chemical Society [ISSN 0103-5053, IF2014 = 1.129], Sociedade Brasileira de Química 2× 36. Journal of Microencapsulation [ISSN 0265-2048, IF2014 = 1.585], Informa Healthcare 2× 37. Journal of Molecular Structure [ISSN 0022-2860, IF2014 = 1.602], Elsevier 1× 38. Journal of Nanoscience and Nanotechnology [ISSN 1533-4880, IF2014 = 1.556], American Scientific Publishers 1× 39. Letters in Drug Design & Discovery [ISSN 1570-1808, IF2014 = 0.770], Bentham Science Publishers 3× 40. Letters in Organic Chemistry [ISSN 1570-1786, IF2014 = 0.664], Bentham Science Publishers 2× 41. Medicinal Chemistry [ISSN 1573-4064, IF2014 = 1.363], Bentham Science Publishers 3× 42. Military Medical Science Letters [ISSN 0372-7025], Faculty of Military Health Sciences, University of Defence 2× 43. Molecules [ISSN 1420-3049, IF2014 = 2.416], MDPI 7×
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44. 45. 46. 47. 48.
Monatshefte fur Chemie [ISSN 0026-9247, IF2014 = 1.222], Springer Pest Management Science [ISSN 1526-498X, IF2014 = 2.694], Wiley-VCH Pharmaceutical Research [ISSN 0724-8741, IF2014 = 3.420], Springer Steroids [ISSN 0039-128X, IF2014 = 2.639], Elsevier Tuberculosis [ISSN 1472-9792, IF2014 = 2.711], Elsevier
Externí hodnotitel projektů (celkem 65 grantových projektů) 1. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (2010–2011) 2. South African Medical Research Council (2010–2011) 3. Technologická agentura České republiky (2010–2013) 4. Interní grantová agentura Ministrstva zdravotnictví České republiky (2011–2013) 5. Agentúra na podporu výskumu a vývoja Slovenské republiky (2012, 2015, 2016) 6. Fulbright Visiting Scholar Program (2014–2015) 7. Hungarian Scientific Research Fund (2014–2015) 8. Grantová agentura České republiky (2015, 2016) 9. Vedecká grantová agentúra MŠ SR a SAV (2015) 10. Polish National Centre for Research and Development (2015)
4× 1× 2× 7× 1× 6× 2× 18× 2× 5× 1× 3× 25× 2× 1×
Člen hodnotící komise 1. Člen finálové výběrové poroty Ceny za nejlepší výzkumnou práci ve farmaceutických vědách 2010 „Ceny za farmacii 2010“ udílenou Francouzským velvyslanectvím v České republice a společností SanofiAventis, 17. červen 2010. 2. Člen finálové výběrové poroty (chemická sekce) „Nadnárodního kola studentské vědecké konference“ Praha, České republika, 12. květen 2015.
Organizování vědeckých konferencí (celkem 15) Člen organizačního výboru konferencí konaných v České republice 1. The XXXVIIth conference "Synthesis and Analysis of Drugs", Brno 2008 2. The XLth conference "Synthesis and Analysis of Drugs", Brno 2011 3. The 4th Nanomaterials and Nanotechnology Meeting "NanoOstrava 2015", Ostrava, 2015 4. The XLIVth conference "Synthesis and Analysis of Drugs", Brno 2015 Člen vědeckého výboru konferencí konaných v České republice 1. The 1st International Symposium and Workshop on Environment and Health, Ostrava, Czech Republic, 2012 2. The 2nd International Symposium and Workshop on Environment and Health, Ostrava, Czech Republic, 2013 3. International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering, Prague, Czech Republic, 2016 4. World Congress on Recent Advances in Nanotechnology (Chair of the Congress, http://rancongress.com/chair/), Prague, Czech Republic, 2016 Člen vědeckého výboru zahraničních konferencí 1. The XXXV Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice – Szczyrk, Poland, 2012 2. The XXXVI Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice – Szczyrk, Poland, 2013 3. The XXXVII Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice – Szczyrk, Poland, 2014 4. The 7th Central European Conference "Chemistry towards Biology", Katowice, Poland, 2014 5. The XXXVIII Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice – Szczyrk, Poland, 2015 6. The 4th World Conference on Physico-Chemical Methods in Drug Discovery and Development, Rovinj – Red Island, Croatia, 2015 7. The 5th IAPC Meeting “Emerging Technologies in Drug Discovery and Development”, Macau, China, 2016 (https://www.iapchem.org/page.php?page_id=73)
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Ocenění za vědecko-výzkumnou činnost (celkem 5) Vědecká ocenění 1. „PRIX DE PHARMACIE 2004” – 2. místo v celostátní soutěži „Cena za farmacii 2004” vyhlášené společností Aventis Pharma s.r.o., Praha, Česká republika. Uděleno: 11. červen 2004. Téma práce: „Quinlukast Analogues as Potential Antileukotrienic Agents: Synthesis and Study of Biological Properties”. 2.
„MOST CITED PAPER 2006–2009 AWARD“ udělena časopisem Bioorganic & Medicinal Chemistry, Elsevier BV, Amsterodam, Nizozemí za článek publikovaný v BMC 2006, 14 (10): 3592-3598.
3.
„2011 INDUSTRIAL AFFAIRS INNOVATION AWARD – TECHNOLOGY AND PROCESSES“ uděleno 1. místo v rámci Sanofi-Aventis korporátního „3. ročníku Industrial Innovation Awards 2011“. Uděleno: 22. červen 2011. Téma práce: „Artificial Digestive System GOLEM” (Reg. No. 2011TI-00082).
Ostatní ocenění 1. „OCENĚNÍ A PODĚKOVÁNÍ ZA DOSAVADNÍ SPOLUPRÁCI“ udělené děkanem Farmaceutické fakulty VFU Brno formou plakety při příležitosti 20. výročí založení Farmaceutické fakulty v rámci Veterinární a farmaceutické univerzity Brno. Uděleno: 14. září 2011. 2. „OUTSTANDING REVIEWER 2014–2015 AWARD“ uděleno vydavatelstvím Wiley-VCH dne 17.září 2015.
Spolupráce s praxí – aktivity v rámci aplikovaného výzkumu V letech 2004–2011 byl pracovníkem R&D divize Zentiva Praha, konkrétně „Centra pro výzkum a metodický rozvoj“, kde byl zodpovědný mimo jiné za vývoj/troubleshooting/portfolio care přípravků, resp. substancí, např.: Lozap H, Lindaxa, Coxtral, atorvastatin, Torvacard, tolterodin, Uroflow, risedronát, Risendros, klopidogrel, Trombex, levocetirizin, Zenaro, tibolon, Ladybon, kandesartan, Carzap, montelukast, Montelar, pregabalin, topiramát. V rámci aplikovaného výzkumu byly rovněž zkoumány možnosti přípravy, stability a využití kokrystalů a dalších krystalických, resp. amorfních forem substancí, např. agomelatin, aprepitant, risedronát, ibandronát, imatinib, gefitinib, erlotinib, sunitinib, dasatinib, sorafenib, lapatinib. Ve spolupráci s Vývojovými dílnami Ústavu organické chemie a biochemie AV ČR se podílel na vývoji unikátního přístroje pro dynamické disoluce pojmenovaný „Golem“, který byl posléze patentován a za jehož přínos pro usnadnění vývoje generických formulací v rámci celého korporátního R&D bylo celému týmu uděleno 1. místo v rámci korporátního 3. ročníku „Industrial Innovation Awards 2011“ Sanofi-Aventis za projekt „Artificial Digestive System GOLEM“. Dále se podílel na projektování laboratoří pro analýzu v pevné fázi, zaváděl metodiky NIR a THz spektroskopie ve vývojových a QC laboratořích v rámci celé společnosti Zentiva. Na základě řešení výše uvedených problematik je spoluautorem 15 patentů, resp. patentových přihlášek. Od roku 2012 vykonává externí poradenskou, resp. školící činnost pro různé farmaceutické firmy v České republice a Slovenské republice.
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Doklady o vyžádaných přednáškách na konferencích
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Doklady o vyžádaných přednáškách na seminářích a workshopech
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Doklady o získaných oceněních
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